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TAK-020 Captisol

Phase 1

Healthy | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Apr 13, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment25
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02723201TAK-020 Relative Bioavailability and Food Effect Study in Healthy ParticipantsPHASE1 COMPLETED 25Apr 28, 2016Aug 24, 2016Apr 13, 20181 United Kingdom
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Study Endpoints
Primary Endpoints
Cmax: Maximum Observed Plasma Concentration for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
AUC∞: Area Under the Plasma Concentration-time Curve From Time 0 to Infinity for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
Terminal Disposition Phase Half-life (T1/2z) in Plasma for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
Secondary Endpoints
Number of Participants Who Experience at Least One or More Treatment-emergent Adverse Event (TEAE)
Baseline up to 30 days after last dose of study drug (Day 58 in Part 1), (Day 40 in Part 2)
Number of Participants Who Meet the Takeda Markedly Abnormal Criteria for Clinical Laboratory Tests at Least Once Post Dose
Baseline up to Day 2
Number of Participants Who Meet the Takeda Markedly Abnormal Criteria for Vital Sign Measurements at Least Once Post Dose
Baseline up to Day 2
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeOTHER
Treatment Arms
ArmTypeDescription
Part-1, Period 1: TAK-020 17.5 mg Oral SolutionEXPERIMENTALSingle dose 17.5 milligram (mg), on Day 1, followed by 7 days of washout. Dose will be determined from TAK-020 single rising dose (SRD) trial.
Part-1, Period 2: TAK-020 17.5 mg Co-crystal Tablet (CCT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part-1, Period 3:TAK-020 17.5 mg Solid Dispersion Tablet (SDT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part-1, Period 4:TAK-020 17.5 mg Immediate Release Tablet(IRT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part 2, Period 1: TAK-020 25 mg CCTEXPERIMENTALParticipants will be randomized to AB or BA crossover where A= Fasted, B =Fed. Sequence I: Single oral dose TAK-020 25 mg, Fasted (A), 7 days washout, single oral dose TAK-020 Fed (B) Sequence II: Single oral dose TAK-020 25 mg, Fed (B), 7 days washout, single oral dose TAK-020 Fasted (A) Dose will be determined from SRD trial and Part 1.
Part- 3 Cohort 1: TAK-020 Solid FormulationEXPERIMENTALSingle oral dose on Day 1. Dose will be determined from SRD trial and Parts 1 and 2
Part 3 Cohort 2: TAK-020 Solid FormulationEXPERIMENTALSingle oral dose on Day 1. Dose will be determined from SRD trial and Parts 1 and 2
Interventions
NameTypeDescription
TAK-020 Captisol Oral SolutionDRUGTAK-020 solution.
TAK-020 CCTDRUGTAK-020 co-crystal tablet
TAK-020 SDTDRUGTAK-020 Solid dispersion tablet.
TAK-020 IRTDRUGTAK-020 immediate release tablet.
TAK-020 Solid FormulationDRUGTAK-020 solid formulation
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Is capable of understanding and complying with protocol requirements. 2. Is legally acceptable representative signs and dates a written, informed consent form and any required privacy authorization prior to the initiation of any study procedures including requesting that a pa...

Countries:United Kingdom
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