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TAK-020 Captisol

Phase 1

Healthy | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Apr 13, 2018

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment25

FDA Designations

No designations recorded

Clinical trial landscape

TAK-020 Captisol · 1 trial · 1 indication

Phase 1 1
NCT02723201TAK-020 Relative Bioavailability and Food Effect Study in Healthy ParticipantsHealthy
COMPLETED25 Analytics
PHASE1COMPLETED
TAK-020 Relative Bioavailability and Food Effect Study in Healthy Participants
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax: Maximum Observed Plasma Concentration for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
AUC∞: Area Under the Plasma Concentration-time Curve From Time 0 to Infinity for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose
Terminal Disposition Phase Half-life (T1/2z) in Plasma for TAK-020
Day 1 pre-dose and at multiple time points (up to 24 hours) post-dose

Secondary Endpoints

Number of Participants Who Experience at Least One or More Treatment-emergent Adverse Event (TEAE)
Baseline up to 30 days after last dose of study drug (Day 58 in Part 1), (Day 40 in Part 2)
Number of Participants Who Meet the Takeda Markedly Abnormal Criteria for Clinical Laboratory Tests at Least Once Post Dose
Baseline up to Day 2
Number of Participants Who Meet the Takeda Markedly Abnormal Criteria for Vital Sign Measurements at Least Once Post Dose
Baseline up to Day 2
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeOTHER

Treatment Arms

ArmTypeDescription
Part-1, Period 1: TAK-020 17.5 mg Oral SolutionEXPERIMENTALSingle dose 17.5 milligram (mg), on Day 1, followed by 7 days of washout. Dose will be determined from TAK-020 single rising dose (SRD) trial.
Part-1, Period 2: TAK-020 17.5 mg Co-crystal Tablet (CCT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part-1, Period 3:TAK-020 17.5 mg Solid Dispersion Tablet (SDT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part-1, Period 4:TAK-020 17.5 mg Immediate Release Tablet(IRT)EXPERIMENTALSingle oral dose 17.5 mg, on Day 1, followed by 7 days of washout. Dose will be the same as Part 1, Period 1.
Part 2, Period 1: TAK-020 25 mg CCTEXPERIMENTALParticipants will be randomized to AB or BA crossover where A= Fasted, B =Fed. Sequence I: Single oral dose TAK-020 25 mg, Fasted (A), 7 days washout, single oral dose TAK-020 Fed (B) Sequence II: Single oral dose TAK-020 25 mg, Fed (B), 7 days washout, single oral dose TAK-020 Fasted (A) Dose will be determined from SRD trial and Part 1.
Part- 3 Cohort 1: TAK-020 Solid FormulationEXPERIMENTALSingle oral dose on Day 1. Dose will be determined from SRD trial and Parts 1 and 2
Part 3 Cohort 2: TAK-020 Solid FormulationEXPERIMENTALSingle oral dose on Day 1. Dose will be determined from SRD trial and Parts 1 and 2

Interventions

NameTypeDescription
TAK-020 Captisol Oral SolutionDRUGTAK-020 solution.
TAK-020 CCTDRUGTAK-020 co-crystal tablet
TAK-020 SDTDRUGTAK-020 Solid dispersion tablet.
TAK-020 IRTDRUGTAK-020 immediate release tablet.
TAK-020 Solid FormulationDRUGTAK-020 solid formulation
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Is capable of understanding and complying with protocol requirements. 2. Is legally acceptable representative signs and dates a written, informed consent form and any required privacy authorization prior to the initiation of any study procedures including requesting that a pa...

Countries:United Kingdom
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Frequently asked questions about TAK-020 Captisol

What is TAK-020 Captisol used for?

TAK-020 Captisol is an investigational small molecule being studied in healthy participants. It is not approved for any disease and is in Phase 1 clinical development. The completed trial evaluated its relative bioavailability and the effect of food on its absorption in healthy volunteers.

Who makes TAK-020 Captisol?

TAK-020 Captisol is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company conducted a Phase 1 study of the drug in healthy participants in the United Kingdom.

What phase is TAK-020 Captisol in?

TAK-020 Captisol is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and the drug is not currently in active clinical trials.

What clinical trials is TAK-020 Captisol in?

TAK-020 Captisol was studied in a completed Phase 1 trial with the identifier NCT02723201, titled "TAK-020 Relative Bioavailability and Food Effect Study in Healthy Participants." The trial enrolled 25 healthy participants in the United Kingdom and was a randomized, controlled study.

Is TAK-020 Captisol the same as TAK-020?

TAK-020 Captisol is a formulation of TAK-020 that uses Captisol, a solubilizing agent. The clinical trial NCT02723201 studied this specific formulation in healthy participants to assess its relative bioavailability and the effect of food on its absorption.