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TAK-020

Phase 1

Healthy Volunteers | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Jan 7, 2019

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment120

FDA Designations

No designations recorded

Clinical trial landscape

TAK-020 · 1 trial · 1 indication

Phase 1 1
NCT02413255Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Ascending Single- and Multiple-Doses of TAK-020 in Healthy VolunteersHealthy Volunteers
COMPLETED120 Analytics
PHASE1COMPLETED
Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Ascending Single- and Multiple-Doses of TAK-020 in Healthy Volunteers
Healthy VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

Percentage of Participants Who Experience at Least One Treatment-emergent Adverse Event (TEAE) in Part 1 Single-rising Dose (SRD)
First dose of study drug up to and including 30 days after last dose of study drug (Up to 31 days) for Part 1

An Adverse Event (AE) is defined as any untoward medical occurrence in a clinical investigation participant administered a drug; it does not necessarily have to have a causal relationship with this treatment. A TEAE is defined as an adverse event that occurred or worsened after receiving study drug.

Percentage of Participants With Markedly Abnormal Values (MAV) for Safety Laboratory Findings at Least Once Post-dose in Part 1 (SRD)
From Day 1 to Day 14 of Part 1

Safety laboratory tests includes hematology, serum chemistries, and urinalysis.

Percentage of Participants With MAV for Vital Sign Measurements at Least Once Post-dose in Part 1 (SRD)
From Day 1 to Day 14 of Part 1

Vital signs include oral temperature, respiratory rate, sitting blood pressure (after 5 minutes resting) and pulse beats per minute (bpm).

Percentage of Participants With MAV for Safety Electrocardiogram (ECG) Parameters at Least Once Post-dose in Part 1 (SRD)
From Day 1 to Day 14 in Part 1

A standard 12-lead ECG was performed. Change from baseline=CFB.

Percentage of Participants Who Experience at Least One Treatment-emergent Adverse Event (TEAE) in Part 2 Multiple-rising Dose (MRD)
First dose of study drug up to and including 30 days after last dose of study drug (Up to 39 days) in Part 2

An AE is defined as any untoward medical occurrence in a clinical investigation participant administered a drug; it does not necessarily have to have a causal relationship with this treatment. A TEAE is defined as an adverse event that occurred or worsened after receiving study drug.

Percentage of Participants With MAV for Safety Laboratory Findings at Least Once Post-dose in Part 2 (MRD)
From Day 1 to Day 17 in Part 2

Safety laboratory tests include hematology, and serum chemistries.

Percentage of Participants With MAV for Vital Sign Measurements at Least Once Post-dose in Part 2 (MRD)
From Day 1 to Day 17 in Part 2

Vital signs include oral temperature respiratory rate, sitting blood pressure (after 5 minutes resting) and pulse (bpm).

Percentage of Participants With MAV for Safety ECG Parameters at Least Once Post-dose in Part 2 (MRD)
From Day 1 to Day 17 in Part 2

A standard 12-lead ECG was performed.

Secondary Endpoints

Cmax: Maximum Observed Plasma Concentration for TAK-020 in Part 1 (SRD)
Pre-dose and multiple timepoints (up to 96 hours) post-dose in Part 1
Cmax: Maximum Observed Plasma Concentration for TAK-020 in Part 2 (MRD)
Pre-dose and multiple timepoints (up to 48 hours) post-dose on Day 1 and pre-dose and multiple timepoints (up to 24 hours) post-dose on Day 9 in Part 2
Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for TAK-020 in Part 1 (SRD)
Pre-dose and multiple timepoints (up to 96 hours) post-dose in Part 1
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part 1 Cohort 1-9: PlaceboPLACEBO_COMPARATORTAK-020 placebo-matching solution, orally, once on Day 1.
Part 1 Cohort 1: TAK-020 0.1 mgEXPERIMENTALTAK-020 0.1 mg, solution, orally once on Day 1.
Part 1 Cohort 2: TAK-020 0.5 mgEXPERIMENTALTAK-020 0.5 mg, solution, orally, once on Day 1 following review of safety, tolerability and pharmacokinetic (PK) data from Cohort 1.
Part 1 Cohort 3: TAK-020 2.5 mgEXPERIMENTALTAK-020 2.5 mg, solution, orally once on Day 1 following review of safety, tolerability and PK data from Cohort 2.
Part 1 Cohort 4: TAK-020 4.4 mgEXPERIMENTALTAK-020 4.4 mg, solution, orally once on Day 1 following review of safety, tolerability and PK data from Cohort 3.
Part 1 Cohort 5: TAK-020 8.8 mgEXPERIMENTALTAK-020 8.8 mg, solution, orally once on Day 1 following review of safety, tolerability and PK data from Cohort 4.
Part 1 Cohort 6: TAK-020 17.5 mgEXPERIMENTALTAK-020 17.5 mg, solution, orally once on Day 1 following review of safety, tolerability and PK data from Cohort 5.
Part 1 Cohort 7: TAK-020 35 mgEXPERIMENTALTAK-020 35 mg, solution, orally once on Day 1. TAK-020 dose will be determined based on review of safety, tolerability and PK data from Cohort 6.
Part 1 Cohort 8: TAK-020 70 mgEXPERIMENTALTAK-020 70 mg, solution, orally once on Day 1. TAK-020 dose will be determined based on review of safety, tolerability and PK data from Cohort 7.
Part 1 Cohort 9: TAK-020 105 mgEXPERIMENTALTAK-020 105 mg, solution, orally once on Day 1. TAK-020 dose will be determined based on review of safety, tolerability and PK data from Cohort 8.
Part 2 Cohort 1-6: PlaceboPLACEBO_COMPARATORTAK-020 placebo-matching solution, orally, once on Day 1 and Days 3 to 9.
Part 2 Cohort 1: TAK-020 3.75 mgEXPERIMENTALTAK-020 3.75 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose are determined based on data from Part 1 of the study.
Part 2 Cohort 2: TAK-020 5.75 mgEXPERIMENTALTAK-020 5.75 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose will be determined based on data from Part 1 and review of safety, tolerability and PK data from Cohort 1 in Part 2.
Part 2 Cohort 3: TAK-020 13 mgEXPERIMENTALTAK-020 13 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose will be determined based on data from Part 1 and review of safety, tolerability and PK data from Cohort 2 in Part 2.
Part 2 Cohort 4: TAK-020 25 mgEXPERIMENTALTAK-020 25 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose will be determined based on data from Part 1 and review of safety, tolerability and PK data from Cohort 3 in Part 2.
Part 2 Cohort 5: TAK-020 45 mgEXPERIMENTALTAK-020 45 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose was determined based on data from Part 1 and review of safety, tolerability and PK data from Cohort 4 in Part 2.
Part 2 Cohort 6: TAK-020 60 mgEXPERIMENTALTAK-020 60 mg, solution, orally once on Day 1 and Days 3-9. TAK-020 dose was determined based on data from Part 1 and review of safety, tolerability and PK data from Cohort 5 in Part 2.

Interventions

NameTypeDescription
TAK-020DRUGTAK-020 oral solution
TAK-020 PlaceboDRUGTAK-020 placebo-matching oral solution
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria Participant eligibility is determined according to the following criteria prior to entry into the study: 1. In the opinion of the investigator, the participant is capable of understanding and complying with protocol requirements. 2. Participant or, when applicable, the participa...

Countries:United States
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Frequently asked questions about TAK-020

What is TAK-020?

TAK-020 is an investigational small molecule being developed by Takeda Pharmaceutical Company Limited. It is currently in Phase 1 clinical development, studied in healthy volunteers. The drug is not approved and remains under clinical investigation.

What is TAK-020 used for?

TAK-020 is being studied for use in healthy volunteers, as part of early-phase clinical trials to evaluate its safety, tolerability, pharmacokinetics, and pharmacodynamics. It is not approved for any disease or condition and is in Phase 1 development.

Who makes TAK-020?

TAK-020 is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company is conducting clinical trials to evaluate the drug's safety and tolerability in healthy volunteers.

What phase is TAK-020 in?

TAK-020 is in Phase 1 clinical development. A completed Phase 1 trial assessed ascending single and multiple doses of the drug in healthy volunteers. It is an investigational drug and has not been approved by regulatory authorities.

What clinical trials is TAK-020 in?

TAK-020 has one completed Phase 1 trial, NCT02413255, titled "Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Ascending Single- and Multiple-Doses of TAK-020 in Healthy Volunteers." The trial enrolled 120 participants in the United States and was placebo-controlled, randomized, and double-blind.