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SYR-472

Phase 3

Diabetes Mellitus | Small molecule | Metabolic |Takeda Pharmaceutical Company Limited|Last Updated: Dec 14, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials5
Total Enrollment1,694
FDA Designations
No designations recorded
Clinical Trials (5)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01751360SYR-472 Open-label StudyPHASE3 COMPLETED 14Apr 1, 2013Aug 1, 2013Dec 11, 20231 Japan
NCT01632007Double-blind Comparative Study of SYR-472PHASE3 COMPLETED 245May 1, 2012Jul 1, 2013Dec 11, 202322 Japan
NCT01431807Long-term Study of SYR-472PHASE3 COMPLETED 680Sep 1, 2011Jun 1, 2013Dec 14, 202341 Japan
NCT00653185Efficacy of SYR-472 in Subjects With Type 2 Diabetes MellitusPHASE2 COMPLETED 369May 1, 2007Mar 1, 2008Jun 22, 201687 United States, Chile +10
NCT00760344Efficacy and Safety of SYR-472 in Subjects With Type 2 Diabetes MellitusPHASE2 COMPLETED 386Mar 1, 2007Mar 1, 2008Jun 22, 2016112 United States, Mexico
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Study Endpoints
Primary Endpoints
Blood Glucose
7 days
Glycosylated hemoglobin (HbA1c)
24 weeks.

Measurement of change in HbA1c (ratio of hemoglobin bound to glucose).

Adverse events
52 weeks.
Change from baseline in glycosylated hemoglobin
Weeks 12 or Final Visit.
Secondary Endpoints
Change from baseline in glycosylated hemoglobin
Weeks 4, 8, and 12 or Final Visit.
Change from baseline in fasting plasma glucose
Weeks 1, 2, 4, 8, and 12 or Final Visit.
1,5-Anhydroglucitol
Weeks 2, 4, 8, and 12 or Final Visit.
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Study Design & Arms
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
SYR-472 100mgEXPERIMENTALSYR-472 100mg
SYR-472 100 mgEXPERIMENTAL -
Alogliptin 25 mgACTIVE_COMPARATOR -
PlaceboPLACEBO_COMPARATOR -
SYR-472 groupEXPERIMENTAL(long-term monotherapy or long-term combination therapy with anti-diabetic drugs)
SYR-472 25 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin therapy)
SYR-472 50 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin therapy)
SYR-472 100 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin therapy)
SYR-472 200 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin therapy)
Placebo QDPLACEBO_COMPARATOR(with lifestyle modification and/or metformin therapy)
SYR-472 3.125 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin stable dose therapy)
SYR-472 12.5 mg QDEXPERIMENTAL(with lifestyle modification and/or metformin stable dose therapy)
Sitagliptin 100 mg QDACTIVE_COMPARATOR(with lifestyle modification and/or metformin stable dose therapy)
Interventions
NameTypeDescription
SYR-472DRUG -
Alogliptin 25 mgDRUG -
PlaceboDRUG -
SitagliptinDRUGSitagliptin 100 mg, tablets, orally, once daily with lifestyle modification and/or metformin stable dose therapy for up to 12 weeks.
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Eligibility Criteria
Age Range20 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: -1. The participant is judged to be capable of understanding and complying with protocol requirements by the investigator or subinvestigator. 2\. The participant can sign and date a written, informed consent form prior to the initiation of any study procedures. Exclusion Crite...

Countries:JapanUnited StatesChileCzechiaGuatemalaHungaryLatviaLithuaniaPuerto RicoRomaniaRussiaSlovakiaUkraineMexico
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