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Relugolix

Phase 3

Uterine Fibroids | Small molecule | Endocrine |Takeda Pharmaceutical Company Limited|Last Updated: Mar 22, 2019

Success Probability

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials2
Total Enrollment346

FDA Designations

No designations recorded

Clinical trial landscape

Relugolix · 2 trials · 1 indication

Phase 3 2
NCT02655224A Placebo-Controlled, Phase 3 Study of Relugolix (TAK-385) 40 mg in the Treatment of Pain Symptoms Associated With Uterine FibroidsUterine Fibroids
COMPLETED65 Analytics
NCT02655237A Phase 3 Study to Evaluate the Efficacy and Safety of Relugolix (TAK-385) 40 mg Compared With Leuprorelin in the Treatment of Uterine FibroidsUterine Fibroids
COMPLETED281 Analytics
PHASE3COMPLETED
A Placebo-Controlled, Phase 3 Study of Relugolix (TAK-385) 40 mg in the Treatment of Pain Symptoms Associated With Uterine Fibroids
Uterine FibroidsUnlock trial analytics
PHASE3COMPLETED
A Phase 3 Study to Evaluate the Efficacy and Safety of Relugolix (TAK-385) 40 mg Compared With Leuprorelin in the Treatment of Uterine Fibroids
Uterine FibroidsUnlock trial analytics

Study Endpoints

Primary Endpoints

Percentage of Participants With a Maximum NRS Score of 1 or Less During the 28 Days Before the Final Dose of Study Drug
For 28 days before the final dose of study drug (up to Week 12)

Pain symptoms were evaluated using the NRS score. NRS score is a self-reported instrument assessing pain from 0 to 10. Higher scores reflect greater level of pain. The percentage of participants with a score of 1 or less is reported.

Percentage of Participants With Total PBAC Score of <10 From Week 6 to 12
Week 6 to 12

PBAC score was used to measure volume of menstrual blood loss. Participants used sanitary products designated by sponsor and recorded the numbers of tampons or towels used, clots and flooding in patient diary. Three diagrams used which represented a lightly, moderately stained or completely saturated pad/tampon. Following scores assigned: 1) 1, 5, or 20 points for each pad; 2) 1, 5, or 10 points for each tampon; 3) 1 or 5 points for each blood clot of \<1 cm/=1 cm/\>1 in longest diameter; 4) 5 points for each episode of flooding. The total PBAC score (sum of points) ranges from 0 to \>500.

Secondary Endpoints

Percentage of Participants With a Maximum NRS Score of 0 During the 28 Days Before the Final Dose of Study Drug
For 28 days before the final dose of study drug (up to Week 12)
Mean NRS Score During the 28 Days Before the Final Dose of Study Drug
For 28 days before the final dose of study drug (up to Week 12)
Percentage of Days Without Pain Symptoms (NRS = 0) During the 28 Days Before the Final Dose of Study Drug
For 28 days before the final dose of study drug (up to Week 12)
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Relugolix 40 mgEXPERIMENTALRelugolix placebo-matching tablet, orally, once daily before breakfast for 3 to 6 weeks in the run-in period, followed by relugolix 40 mg, tablet, orally once daily before breakfast for 12 weeks.
PlaceboPLACEBO_COMPARATORRelugolix placebo-matching tablet, orally, once daily before breakfast for 3 to 6 weeks in the run-in period, followed by relugolix placebo-matching tablet, orally once daily before breakfast for 12 weeks.
Leuprorelin 1.88 mg or 3.75 mgACTIVE_COMPARATORRelugolix placebo matching tablets, orally, once daily along with leuprorelin acetate placebo matching injection, SC, once in 4 weeks for 3 to 6 weeks in run-in period followed by leuprorelin acetate 1.88 mg or 3.75 mg, injection, SC, once in 4 weeks and relugolix placebo matching tablets, orally, once daily for 24 weeks in treatment period.

Interventions

NameTypeDescription
RelugolixDRUGRelugolix Tablets
Relugolix placeboDRUGRelugolix placebo-matching tablets
LeuprorelinDRUGLeuprorelin injection
Leuprorelin PlaceboDRUGLeuprorelin placebo-matching injections
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Eligibility Criteria

Age Range20 Years to N/A
SexFEMALE
Healthy VolunteersNo
Study Sites11

Inclusion Criteria: Inclusion Criteria for Entering the Screening Period (at VISIT 1) 1. In the opinion of the investigator or subinvestigator, the participant is capable of understanding and complying with protocol requirements. 2. The participant signs and dates a written, informed consent form ...

Countries:Japan
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