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PvP001

Phase 1

Digestive System Disease | Small molecule | Other |Takeda Pharmaceutical Company Limited|Last Updated: Apr 4, 2023

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Trial Design

RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment139

FDA Designations

No designations recorded

Clinical trial landscape

PvP001 · 1 trial · 1 indication

Phase 1 1
NCT03701555A Study of PVP001, PVP002, and PVP003 in Healthy Adults and PVP001 and PVP002 in Adults With Celiac DiseaseDigestive System Disease
COMPLETED139 Analytics
PHASE1COMPLETED
A Study of PVP001, PVP002, and PVP003 in Healthy Adults and PVP001 and PVP002 in Adults With Celiac Disease
Digestive System DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Part 1: Number of Participants Reporting One or More Treatment Emergent Adverse Events (TEAEs) for PvP001 and PvP002
Cohort Treatment Day up to 5 days after 24-hour safety assessment on Day 2 (up to Day 7)
Part 4: Number of Participants Reporting One or More TEAEs for PvP003 After Multiple Doses
Day 1 of Cohort Treatment Period 1 up to 5 days after the Day 5 of Cohort Treatment Period 2 (up to Day 28)
Part 1: Number of Participants Reporting One or More Treatment Emergent Serious Adverse Events (TESAEs) for PvP001 and PvP002
Cohort Treatment Day up to 5 days after 24-hour safety assessment on Day 2 (up to Day 7)
Part 4: Number of Participants Reporting One or More TESAEs for PvP003 600 mg After Multiple Doses
Day 1 of Cohort Treatment Period 1 up to 5 days after the Day 5 of Cohort Treatment Period 2 (up to Day 28)
Part 2, Group 1, Cohort 2B: Median Percentage of Gluten Degradation by PvP001 in a Standardized 3 Gram (gm) Gluten-containing Study Meal After Administration of PvP001
Cohort Treatment Day

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using Enzyme-Linked Immunosorbent Assay (ELISA) based on the monoclonal R5 and G12 antibodies.

Part 2, Group 2, Cohort 2E: Median Percentage of Gluten Degradation by PvP002 in a Standardized 3 gm Gluten-containing Study Meal After Administration of PvP002
Cohort Treatment Day

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 1, Cohort 2C: Median Percentage of Gluten Degradation by PvP001 in a Standardized 3 gm Gluten-containing Study Meal Following 7 Days of Standard Dose PPI Treatment
Cohort Treatment Day

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2G and 2H: Median Percentage of Gluten Degradation by PvP001 300 mg and 600 mg in a Standardized 1 gm Gluten-containing Study Meal at 20 Minutes After Administration of PvP001
Cohort Treatment Day: at 20 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2G and 2H: Median Percentage of Gluten Degradation by PvP001 300 mg and 600 mg in a Standardized 1 gm Gluten-containing Study Meal at 35 Minutes After Administration of PvP001
Cohort Treatment Day: at 35 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2G and 2H: Median Percentage of Gluten Degradation by PvP001 300 mg and 600 mg in a Standardized 1 gm Gluten-containing Study Meal at 65 Minutes After Administration of PvP001
Cohort Treatment Day: at 65 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2J: Median Percentage of Gluten Degradation by PvP001 900 mg in a Standardized 6 gm Gluten-containing Study Meal at 20 Minutes After Administration of PvP001
Cohort Treatment Day: at 20 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2J: Median Percentage of Gluten Degradation by PvP001 900 mg in a Standardized 6 gm Gluten-containing Study Meal at 35 Minutes After Administration of PvP001
Cohort Treatment Day: at 35 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 2, Group 3, Cohort 2J: Median Percentage of Gluten Degradation by PvP001 900 mg in a Standardized 6 gm Gluten-containing Study Meal at 65 Minutes After Administration of PvP001
Cohort Treatment Day: at 65 minutes post-dose

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 3, Groups 1 to 5, Cohorts 3B, 3D, 3F, 3H and 3J: Median Percentage of Gluten Degradation by PvP003 150 mg and 600 mg in a Standardized 1 gm Gluten-containing Study Meal at 35 Minutes After Administration of PvP003
Cohort Treatment Day: at 35 minutes

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Part 3, Groups 1 to 5, Cohorts 3B, 3D, 3F, 3H and 3J: Median Percentage of Gluten Degradation by PvP003 150 mg and 600 mg in a Standardized 1 gm Gluten-containing Study Meal at 65 Minutes After Administration of PvP003
Cohort Treatment Day: at 65 minutes

Median percentage degraded relative to placebo was derived using the formula: (1 - \[active/placebo\])\*100. Gluten degradation was assessed using ELISA based on the monoclonal R5 and G12 antibodies.

Secondary Endpoints

Part 1 and Part 2, Cmax: Maximum Observed Plasma Concentration for PvP001 and PvP002
Cohort Treatment Day pre-dose and at multiple time points (up to 480 minutes) post-dose
Part 1 and Part 2, Tmax: Time to Reach the Maximum Plasma Concentration (Cmax) for PvP001 and PvP002
Cohort Treatment Day pre-dose and at multiple time points (up to 480 minutes) post-dose
Part 1 and Part 2, T(1/2): Terminal Disposition Phase Half-life of PvP001 and PvP002
Cohort Treatment Day pre-dose and at multiple time points (up to 480 minutes) post-dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Part 1, Cohort 1A-1 to 1D-1 Healthy ParticipantsEXPERIMENTALA single dose of PvP001 placebo, PvP001 100 mg, PvP001 300 mg, or PvP001 900 mg will be administered in ascending order to healthy participants in Cohorts 1A-1, 1B-1, 1C-1, and 1D-1.
Part 1, Cohort 1E-1 Healthy ParticipantsEXPERIMENTALA single dose of the maximum feasible dose (MFD) of PvP002 will then be administered to healthy participants in Cohort 1E-1.
Part 1, Cohort 1A-2 - 1D-2 Celiac Disease (CeD)EXPERIMENTALA single dose of PvP001 placebo, PvP001 100 mg, PvP001 300 mg, or PvP001 900 mg will be administered in ascending order to participants with CeD in Cohorts 1A-2, 1B-2, 1C-2, and 1D-2.
Part 1, Cohort 1E-2 CeDEXPERIMENTALA single dose of the MFD of PvP002 will then be administered to participants with CeD in Cohort 1E-2.
Part 2, Cohort 2A - Cohort 2C Healthy ParticipantsEXPERIMENTALParticipants will be blinded to the PvP001 dose (placebo or MTD of PvP001) and will also receive MTD of PvP001 following 7 days of PPI treatment.
Part 2, Cohort 2D Healthy ParticipantsEXPERIMENTALParticipants will receive PvP001 placebo or MFD of PvP001.
Part 2, Cohort 2E Healthy ParticipantsEXPERIMENTALParticipants will receive PvP002 placebo or MFD of PvP002.
Part 2, Cohort 2F- Cohort 2H Healthy ParticipantsEXPERIMENTALParticipants will receive the PvP001 placebo and either 300 mg or 600 mg of PvP001.
Part 2, Cohort 2I and Cohort 2J Healthy ParticipantsEXPERIMENTALParticipants will receive the PvP001 placebo and 900 mg of PvP001.
Part 3, Cohorts 3A and 3B Healthy ParticipantsEXPERIMENTALParticipants will receive single dose of PvP003 placebo and 600 mg of PvP003 with pretreatment buffer solution before a standardized 1 gm gluten-containing study meal.
Part 3, Cohorts 3C and 3D Healthy ParticipantsEXPERIMENTALParticipants will receive single dose of PvP003 placebo and 600 mg of PvP003 without pretreatment buffer solution before a standardized 1 gm gluten-containing study meal.
Part 3, Cohorts 3E and 3F Healthy ParticipantsEXPERIMENTALParticipants will receive single dose of PvP003 placebo and 600 mg of PvP003 without pretreatment buffer solution after an approximately 50 milliliter (mL) portion of a standardized 1 gm gluten-containing study meal.
Part 3, Cohorts 3G and 3H Healthy ParticipantsEXPERIMENTALParticipants will receive single dose of PvP003 placebo and 600 mg of PvP003 without pretreatment buffer solution before a standardized gluten-free study meal followed approximately 30 minutes later by a standardized 1 gm gluten-containing study meal.
Part 4, Cohorts 4A and 4B Healthy ParticipantsEXPERIMENTALParticipants will receive multiple dose of PvP003 placebo and 600 mg of PvP003.
Part 3, Cohorts 3I and 3J Healthy ParticipantsEXPERIMENTALParticipants will receive single dose of PvP003 placebo and 150 mg of PvP003 without pretreatment buffer solution before a standardized 1 gm gluten-containing study meal.

Interventions

NameTypeDescription
PvP001 placeboOTHERplacebo
PvP001 100 mgDRUGPvP001 100 mg
PvP001 300 mgDRUGPvP001 300 mg
PvP001 900 mgDRUGPvP001 900 mg
Maximum Feasible Dose (MFD) of PvP002DRUGMFD of PvP002
Maximum Tolerated Dose (MTD) of PvP001DRUGMaximum Tolerated Dose (MTD) of PvP001
MTD of PvP001 following 7 days of PPI treatmentDRUGMaximum Tolerated Dose (MTD) of PvP001 following 7 days of PPI (Proton Pump Inhibitor) treatment
PvP002 placeboOTHERPlacebo
PvP001 600 mgDRUGPvP001 600 mg
PvP003 placeboDRUGPlacebo tablet orally.
PvP003DRUGPvP003 tablet orally.
PvP003 150 mgDRUGPvP003 150 mg
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Eligibility Criteria

Age Range18 Years to 64 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: Part 1, Part 2, Part 3 and Part 4 1. Male or female age 18- 64 years, inclusive 2. No relevant gastrointestinal symptoms 3. Able to abstain from alcohol for 72 hours prior to the Screening Visit; for 72 hours prior to and after the Cohort Treatment Day (Part 1, Part 2, and Part...

Countries:United States
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Frequently asked questions about PvP001

What is PvP001 used for?

PvP001 is an investigational small molecule being studied for the treatment of digestive system disease, specifically in adults with celiac disease. It is currently in Phase 1 clinical development and has not been approved by the FDA.

Who makes PvP001?

PvP001 is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. The company is conducting clinical trials to evaluate the safety and efficacy of this investigational drug.

What phase is PvP001 in?

PvP001 is in Phase 1 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities and is still undergoing clinical trials to assess its safety and potential efficacy.

What clinical trials is PvP001 in?

PvP001 has been studied in a Phase 1 clinical trial with the identifier NCT03701555. This completed trial enrolled 139 participants and evaluated PvP001, along with PVP002 and PVP003, in healthy adults and adults with celiac disease.

Is PvP001 the same as PVP002 or PVP003?

No, PvP001 is a distinct investigational drug from PVP002 and PVP003. However, all three were studied together in a single Phase 1 clinical trial (NCT03701555) that evaluated their safety and tolerability in healthy adults and adults with celiac disease.