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Tebipenem Pivoxil Hydrobromide

Phase 1

Diabetes | Small molecule | Metabolic |Spero Therapeutics, Inc.|Last Updated: Oct 23, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
ACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment12
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04919954Tebipenem (SPR994) Tissue Penetration in Diabetic Patients With Wound Infections and Healthy Volunteers Via In Vivo MicrodialysisPHASE1 COMPLETED 12Jul 1, 2021Dec 23, 2022Oct 23, 20231 United States
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Study Endpoints
Primary Endpoints
Tebipenem Pivoxil Hydrobromide Tissue Penetration
8 hours

The ratio of tebipenem tissue concentrations to blood concentrations following the final tebipenem dose

Secondary Endpoints
Tebipenem Pivoxil Hydrobromide Area Under the Curve (AUC) in Tissue
8 hours
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeOTHER
Treatment Arms
ArmTypeDescription
Diabetic Wound InfectionEXPERIMENTALParticipants with a documented medical history of Type 1 or Type 2 diabetes and a mild to moderate (Grade 2 or 3) wound infection of the lower limb will receive 3 to 7 doses of tebipenem, followed by sampling of interstitial tissue fluid at the margin of the wound by a microdialysis probe over 8 hours following the last dose.
Healthy VolunteersACTIVE_COMPARATORParticipants will be male or female healthy adult volunteers with no significant medical or medication history. Participants will receive 3 doses of tebipenem, followed by sampling of interstitial tissue fluid by a microdialysis probe inserted in a thigh over 8 hours following the last dose.
Interventions
NameTypeDescription
Tebipenem Pivoxil HydrobromideDRUGTebipenem 300 mg or 600 mg will be administered orally every 8 hours for total of 3 to 7 doses
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersYes
Study Sites1

Exclusion Criteria - All patients/participants Participants in the diabetic wound group or healthy volunteer group will be excluded if any of the following criteria are met: 1. Less than 18 years of age 2. History of hypersensitivity or allergy to tebipenem or its derivatives and any β-lactam anti...

Countries:United States
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