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SAR260301

Phase 1

Neoplasm Malignant | Small molecule | Oncology |Sanofi|Last Updated: Apr 10, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment75
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01673737A Phase I/Ib Trial for the Evaluation of SAR260301 in Monotherapy or in Combination With Vemurafenib in Patients With Various Advanced CancerPHASE1 COMPLETED 75Aug 1, 2012Feb 1, 2015Apr 10, 20154 United States, Canada
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Study Endpoints
Primary Endpoints
Maximal tolerated dose (MTD) of SAR260301 in monotherapy (Study Part A)
Day 28
Maximal tolerated dose (MTD) of SAR260301 in combination with vemurafenib (Study Part B)
Day 28
Secondary Endpoints
Number of patients with treatment emergent events
Up to 2 years
Assessment of PK parameters for SAR260301 and vemurafenib, including tmax, Cmax, AUC, Rac (Day 28/Day1), half-life, CL, Ctrough
4 weeks
Assessment of PK parameters for SAR260301 including tmax, Cmax, AUC fasting and fed (food effect)(Only part A)
Up to 8 weeks
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part A MonotherapyEXPERIMENTALDose escalation of daily or twice daily SAR260301 within a 28-day cycle, followed by an expansion phase at the maximal tolerated dose
Part B CombinationEXPERIMENTALDose escalation of twice-daily SAR260301 within a 28-day cycle and in combination with 720 or 960 mg twice daily of Vemurafenib, followed by an expansion phase at the maximal tolerated dose of SAR260301 in combination
Interventions
NameTypeDescription
SAR260301DRUGPharmaceutical form: film-coated tablets Route of administration: oral
VemurafenibDRUGPharmaceutical form: film-coated tablets Route of administration: oral
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites4

Inclusion criteria : * Age ≥18 years old * Locally advanced or metastatic solid tumor disease as well as lymphoma for which no alternative therapy is available (Part A) * Unresectable / metastatic BRAF-mutated melanomas, progressing on BRAF inhibitor after no more than 4 months treatment or with on...

Countries:United StatesCanada
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