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SAR247799

Phase 1

Microvascular Coronary Artery Disease | Small molecule | Cardiovascular |Sanofi|Last Updated: Apr 25, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment54
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03462017Pharmacodynamic Study to Assess the Effects of Repeated Dosing of SAR247799 on Endothelial Function in Patients With Type 2 Diabetes MellitusPHASE1 COMPLETED 54Mar 7, 2018Dec 22, 2018Apr 25, 20222 Germany
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Study Endpoints
Primary Endpoints
Change in Flow Mediated Dilation (FMD)
Baseline to Days 14, 21, 28, 35, and 42

Absolute change from baseline in the % FMD index of the brachial artery

Secondary Endpoints
Microvascular reactivity
Baseline to Days 14, 21, 28, 35, and 42
Number of adverse events
Up to Day 42
Assessment of pharmacokinetic (PK) parameter: Cmax
Days 1, 2, 3, 7, and 14
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
SAR247799EXPERIMENTALSAR247799 repeated doses once daily in the morning under fasted condition for 28 days according to a sequential dose design
PlaceboPLACEBO_COMPARATORIdentical matching placebo for SAR247799 and for sildenafil once daily in the morning under fasted condition for 28 days
SildenafilACTIVE_COMPARATORSildenafil once daily in the morning under fasted condition for 28 days
Interventions
NameTypeDescription
SAR247799DRUGPharmaceutical form:Capsule Route of administration: Oral
PlaceboDRUGPharmaceutical form:Capsule Route of administration: Oral
SildenafilDRUGPharmaceutical form:Encapsulated tablet Route of administration: Oral
AcetylcholineDRUGPharmaceutical form:Solution Route of administration: Transdermal
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Eligibility Criteria
Age Range18 Years — 64 Years
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion criteria : * Male and female stable Type 2 diabetes mellitus (T2DM) patients. * Body Mass Index between 18 and 35 kg/m\^2. * Stable T2DM patients, but otherwise healthy as assessed by a clinical and laboratory assessments and detailed medical history. * Diagnosis of T2DM for at least 6 mo...

Countries:Germany
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