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Insulin glargine HOE901

Phase 1

Type 1 Diabetes Mellitus | Small molecule | Metabolic |Sanofi|Last Updated: Aug 13, 2013

Target and mechanism

ModalitySmall molecule

Also known as Insulin glargine new formulation HOE901

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials3
Total Enrollment70

FDA Designations

No designations recorded

Clinical trial landscape

Insulin glargine HOE901 · 4 trials · 2 indications

Phase 1 4
NCT01838083Euglycemic Clamp Study Comparing Two New Insulin Glargine Formulations in Subjects With Type 1 Diabetes MellitusType1 Diabetes
COMPLETED50 Analytics
NCT01493115Single Dose Study With a New Insulin Glargine Formulation and Lantus® in Japanese Patients With Type 1 Diabetes MellitusType 1 Diabetes Mellitus
COMPLETED18 Analytics
NCT01349855Repeated Dosing Study With a New Insulin Glargine Formulation and Lantus® in Patients With Type 1 Diabetes MellitusType 1 Diabetes Mellitus
COMPLETED30 Analytics
NCT01146678Relative Bioavailability and Activity of Different Formulations of Insulin Glargine and Lixisenatide in Patients With Diabetes Mellitus Type 1Type 1 Diabetes Mellitus
COMPLETED22 Analytics
PHASE1COMPLETED
Euglycemic Clamp Study Comparing Two New Insulin Glargine Formulations in Subjects With Type 1 Diabetes Mellitus
Type1 DiabetesUnlock trial analytics
PHASE1COMPLETED
Single Dose Study With a New Insulin Glargine Formulation and Lantus® in Japanese Patients With Type 1 Diabetes Mellitus
Type 1 Diabetes MellitusUnlock trial analytics
PHASE1COMPLETED
Repeated Dosing Study With a New Insulin Glargine Formulation and Lantus® in Patients With Type 1 Diabetes Mellitus
Type 1 Diabetes MellitusUnlock trial analytics
PHASE1COMPLETED
Relative Bioavailability and Activity of Different Formulations of Insulin Glargine and Lixisenatide in Patients With Diabetes Mellitus Type 1
Type 1 Diabetes MellitusUnlock trial analytics

Study Endpoints

Primary Endpoints

Area under the serum insulin concentration curve within 24 hours (INS-AUC0-24) after dosing on Day 6
24-hours (D6 to D7)
Glucose infusion rate
up to day 2 of each period
Safety in terms of adverse and serious adverse events, vital signs, ECG, safety laboratory
up to day 10 of each period
Area under the plasma lixisenatide concentration curve (LIX-AUClast)
1 day (D1 to D2) in the first treatment period and 1 day (D1 to D2) during the second treatment period
Lixisenatide maximum plasma/serum peak concentration (LIX-Cmax)
1 day (D1 to D2) in the first treatment period and 1 day (D1 to D2) during the second treatment period

Secondary Endpoints

Maximum insulin concentration (INS-Cmax)
24-hours (D6 to D7)
Time to INS-Cmax (INS-tmax)
24-hours (D6 to D7)
Time to reach 50% of INS-AUC0-24 (T50%-INS-AUC0-24)
24-hours (D6 to D7)
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Insulin glargine new formulation (test T formulation)EXPERIMENTALOnce daily for 6 days
Insulin glargine new formulation (reference R formulation)EXPERIMENTALOnce daily for 6 days
Sequence 1EXPERIMENTALReference (insulin glargine) - Test1 (insulin glargine - new formulation dose 1) - Test2 (insulin glargine - new formulation dose 2)
Sequence 2EXPERIMENTALTest1 (insulin glargine - new formulation dose 1) - Test2 (insulin glargine - new formulation dose 2) - Reference (insulin glargine)
Sequence 3EXPERIMENTALTest2 (insulin glargine - new formulation dose 2) - Reference (insulin glargine) - Test1 (insulin glargine - new formulation dose 1)
Cohort 1EXPERIMENTALDose Level 1
Cohort 2EXPERIMENTALDose Level 2
Lantus(insulin glargine)/lixisenatide on-site mixEXPERIMENTALSingle dose injection of an on site mix of Lantus U100 and lixisenatide (800µg/mL in Lantus U100) at one peri-umbilical site under fasting conditions
lixisenatide + Lantus (insulin glargine)ACTIVE_COMPARATORSingle dose, separate injection simultaneous injections of Lantus U100 and lixisenatide (100µg/mL) at opposite peri-umbilical sites within 1 minute under fasting conditions

Interventions

NameTypeDescription
Insulin glargine new formulation HOE901DRUGPharmaceutical form: solution Route of administration: subcutaneous
Insulin glargine HOE901DRUGPharmaceutical form:solution for injection Route of administration: subcutaneous
Insulin glargine - New formulation HOE901DRUGPharmaceutical form:solution for injection Route of administration: subcutaneous
Lixisenatide AVE0010DRUGPharmaceutical form:solution for injection Route of administration: subcutaneous
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Eligibility Criteria

Age Range18 Years to 64 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion criteria : * Male or female subjects, between 18 and 64 years of age, inclusive, with diabetes mellitus type 1 for more than one year * Total insulin dose of \< 1.2 U/kg/day * Minimum usual basal insulin dose ≥ 0.2 U/kg/day * Body weight between 50.0 kg and 110.0 kg, Body Mass Index betwe...

Countries:GermanyJapan
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