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pyroglutamate rongliflozin

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |Sunshine Biopharma Inc.|Last Updated: May 5, 2026

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment32

FDA Designations

No designations recorded

Clinical trial landscape

pyroglutamate rongliflozin · 2 trials · 2 indications

Phase 1 2
NCT05374343A Study of the Pharmacokinetics, Pharmacodynamics, and Safety of Rongliflozin in Type 2 Diabetic Subjects With Renal ImpairmentType 2 Diabetes
COMPLETED32 Analytics
NCT05427682A Clinical Trial to Evaluate the Pharmacokinetics and Safety of Pyroglutamate Rongliflozin Capsules in Subjects With Mild and Moderate Liver DamageDiabetes Mellitus, Type 2
COMPLETED32 Analytics
PHASE1COMPLETED
A Study of the Pharmacokinetics, Pharmacodynamics, and Safety of Rongliflozin in Type 2 Diabetic Subjects With Renal Impairment
Type 2 DiabetesUnlock trial analytics
PHASE1COMPLETED
A Clinical Trial to Evaluate the Pharmacokinetics and Safety of Pyroglutamate Rongliflozin Capsules in Subjects With Mild and Moderate Liver Damage
Diabetes Mellitus, Type 2Unlock trial analytics

Study Endpoints

Primary Endpoints

Plasma concentrations of rongliflozin
0 hour(pre-dose) to 96 hours after administration

Plasma concentrations of rongliflizin following the administration of a single dose of rongliflozin, the pharmacokinetic parameters for rongliflozin will be measured in varying degrees of kidney function.

Cmax
0 hour(pre-dose) to 96 hours after administration

Maximum plasma concentration of study drugs

AUC
0 hour(pre-dose) to 96 hours after administration

Maximum plasma concentration of study drugs

Adverse Events
Day -1 (Baseline) to Day 5

Incidence of adverse events

Secondary Endpoints

Change from baseline in 24-hour urine glucose excretion in varying degrees of kidney function
Day -1 (Baseline) to Day 5
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Group A and C (normal kidney function)ACTIVE_COMPARATOREach subject will receive a single dose of rongliflozin on Day 1
Group B (mild renal impairment)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1
Group D (moderate renal impairment)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1
Group A (normal liver function)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1
Group B (mild liver damage)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1
Group C (normal liver function)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1
Group D (moderate liver damage)EXPERIMENTALEach subject will receive a single dose of rongliflozin on Day 1

Interventions

NameTypeDescription
pyroglutamate rongliflozin capsulesDRUGSubjects will receive one 50mg capsule orally (by mouth) on Day 1
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Eligibility Criteria

Age Range18 Years to 75 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Type 2 diabetes patients. * The subject is willing to take effective contraceptive measures without a pregnancy plan within 4 weeks after signing the informed consent form to taking the test drug. * When screening, 19.0 kg/m2 \< or = body mass index (BMI) \< or = 35.0 kg/m2. *...

Countries:China
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Frequently asked questions about pyroglutamate rongliflozin

What is pyroglutamate rongliflozin used for?

Pyroglutamate rongliflozin is an investigational small molecule being developed for the treatment of Type 2 Diabetes Mellitus. It is currently in Phase 1 clinical development and has not been approved by regulatory authorities.

Who makes pyroglutamate rongliflozin?

Pyroglutamate rongliflozin is being developed by Sunshine Biopharma Inc., a company listed on the stock exchange under the ticker SBFM. The drug is in Phase 1 clinical development for Type 2 Diabetes.

What phase is pyroglutamate rongliflozin in?

Pyroglutamate rongliflozin is in Phase 1 clinical development. It is an investigational drug and has not been approved for any use. Two Phase 1 studies have been completed, with a total of 32 participants enrolled in each trial.

What clinical trials has pyroglutamate rongliflozin been in?

Pyroglutamate rongliflozin has been studied in two completed Phase 1 trials. NCT05374343 evaluated pharmacokinetics, pharmacodynamics, and safety in Type 2 diabetic subjects with renal impairment. NCT05427682 evaluated pharmacokinetics and safety in subjects with mild and moderate liver damage.

Is pyroglutamate rongliflozin the same as rongliflozin?

Pyroglutamate rongliflozin is a form of rongliflozin, as indicated by the clinical trial title for NCT05374343, which refers to rongliflozin. The drug is being developed for Type 2 Diabetes and is currently in Phase 1 trials.