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Rongliflozin

Phase 1

Healthy Adult Male Volunteers | Small molecule | Other |Sunshine Biopharma Inc.|Last Updated: Apr 12, 2023

Success Probability

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment6

FDA Designations

No designations recorded

Clinical trial landscape

Rongliflozin · 2 trials · 2 indications

Phase 1 2
NCT05497674Effects of Rifampicin and Probenecid On The Pharmacokinetic Profile Of Rongliflozin In Healthy SubjectsType 2 Diabetes Mellitus
COMPLETED28 Analytics
NCT05109078ADME Study of [14C]- Rongliflozin in Healthy Male SubjectsHealthy Adult Male Volunteers
COMPLETED6 Analytics
PHASE1COMPLETED
Effects of Rifampicin and Probenecid On The Pharmacokinetic Profile Of Rongliflozin In Healthy Subjects
Type 2 Diabetes MellitusUnlock trial analytics
PHASE1COMPLETED
ADME Study of [14C]- Rongliflozin in Healthy Male Subjects
Healthy Adult Male VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

rongliflozin: area under the drug-time curve (AUC) ratios of geometric means of rongliflozin+rifampicin relative to rongliflozin alone.
from 0 hour(pre-dose,within 30mins)to 5 days after rongliflozin dosing

To assess the effect of rifampicin on the AUC of rongliflozin

rongliflozin: The peak concentration (Cmax) ratios of geometric means of rongliflozin+rifampicin relative to rongliflozin alone.
from 0 hour(pre-dose,within 30mins)to 5 days after rongliflozin dosing

To assess the effect of rifampicin on the Cmax of rongliflozin

rongliflozin: AUC ratios of geometric means of rongliflozin+probenecid relative to rongliflozin alone.
from 0 hour(pre-dose,within 30mins)to 5 days after rongliflozin dosing

To assess the effect of probenecid on the AUC of rongliflozin

rongliflozin:Cmax ratios of geometric means of rongliflozin+probenecid relative to rongliflozin alone.
from 0 hour(pre-dose,within 30mins)to 5 days after rongliflozin dosing

To assess the effect of probenecid on the Cmax of rongliflozin

Cumulative excretion of 14C-labeled drug-related material (radioactivity in urine and fecal samples)
up to 14 days

Percent (%) of each radiolabeled drug-related material (parent and each metabolite) will be determined in urine and feces.

Identification of the Proportion of different metabolites to determine biotransformation pathway of Rongliflozin
up to 14 days

Proportion of different metabolites(Rongliflozin and main metabolites).

Distribution of radioactivity in whole blood and plasma and the pharmacokinetics of total radioactivity in plasma
up to 11 days

Radioactivity concentration in whole blood and plasma samples.

Secondary Endpoints

The time to peak (Tmax) of Rongliflozin.
from 0 hour(pre-dose,within 30mins)to 5 days after rongliflozin dosing
pharmacology (PD) of rongliflozin: cumulative urine glucose excretion every 24 hours
from 0 hour to 5 days after rongliflozin dosing
the number of participants with adverse events (AE) in Cohort A
from screening to 3 days after last dose of rifampicin
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
rongliflozin and/or rifampicinEXPERIMENTALon Day 1, subjects will receive a single dose administration of rongliflozin, followed by a washout period of 4 days. Starting On Day 5, subjects will administer rifampicin once a day (QD) for 10 consecutive days ( Day 5 to Study Day 14) , comprising of a single dose administration of rongliflozin on Study Day 11.
rongliflozin and/or probenecidEXPERIMENTALon Day 1, subjects will receive a single dose administration of rongliflozin, followed by a washout period of 4 days. Probenecid will be administrated twice a day from Day 5 to Day 9, and another single dose administration of rongliflozin on Day 6.
[14C]- RongliflozinEXPERIMENTALPatients will receive single dose of \[14C\]- Rongliflozin (Suspension, 50mg/100μCi)

Interventions

NameTypeDescription
RongliflozinDRUGoral administration, single dose on Day 1 and Day 11
RifampinDRUGQD for 10 days
ProbenecidDRUGtwice a day, for 5 days
[14C]- RongliflozinDRUGPatients will receive single dose of orally \[14C\]- Rongliflozin on Day 1
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Eligibility Criteria

Age Range18 Years to 45 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Sign the informed consent form before the trial and fully understand the trial content, process and possible adverse reactions; * Be able to complete the test according to the requirements of the protocol; * Subjects (including partners) are willing to take effective contracep...

Countries:China
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Frequently asked questions about Rongliflozin

What is Rongliflozin used for?

Rongliflozin is an investigational small molecule being studied for Type 2 Diabetes Mellitus and in healthy adult male volunteers. It is currently in Phase 1 clinical development and is not approved by the FDA.

Who makes Rongliflozin?

Rongliflozin is being developed by Sunshine Biopharma Inc., a company listed on the NASDAQ under the ticker SBFM. The drug is currently in Phase 1 clinical trials.

What phase is Rongliflozin in?

Rongliflozin is in Phase 1 clinical development. It is an investigational drug and has not been approved by the FDA. Clinical trials for Rongliflozin have been completed.

What clinical trials is Rongliflozin in?

Rongliflozin has been studied in two completed Phase 1 clinical trials: NCT05109078, an ADME study in healthy male subjects, and NCT05497674, a study of drug interactions in healthy subjects with Type 2 Diabetes Mellitus.

Is Rongliflozin the same as other drugs?

Rongliflozin is a distinct drug candidate developed by Sunshine Biopharma Inc. No alternative names for Rongliflozin have been identified in the available information.