Recent Updates
Recently added Catalysts

HEC113995PA•H2O

Phase 1

Healthy | Small molecule | Other |Sunshine Biopharma Inc.|Last Updated: May 13, 2021

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment69

FDA Designations

No designations recorded

Clinical trial landscape

HEC113995PA•H2O · 1 trial · 1 indication

Phase 1 1
NCT03943251The Study of a Selective Serotonin Partial Agonist and Reuptake Inhibitors, HEC113995PA•H2O,in Healthy SubjectsHealthy
COMPLETED69 Analytics
PHASE1COMPLETED
The Study of a Selective Serotonin Partial Agonist and Reuptake Inhibitors, HEC113995PA•H2O,in Healthy Subjects
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Adverse events of the single ascending-dose
From the baseline to day4

To assess the safe and tolerability of the single ascending-dose

Secondary Endpoints

Maximum Plasma Concentration(Cmax)
Prior to dosing(0.5h)and 0.5h,1h,1.5h,2h,2.5h,3h,4h,5h,6h,8h,10h,12h,24h,36h,48h,72h after dosing
Area Under the Curve(AUC)
Prior to dosing(0.5h)and 0.5h,1h,1.5h,2h,2.5h,3h,4h,5h,6h,8h,10h,12h,24h,36h,48h,72h after dosing
Maximum Peak Time(Tmax)
Prior to dosing(0.5h)and 0.5h,1h,1.5h,2h,2.5h,3h,4h,5h,6h,8h,10h,12h,24h,36h,48h,72h after dosing
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
HEC113995PA•H2O tabletEXPERIMENTALIncluding 7 dose groups(2.5-、5、10-、20-、40-、60-、80mg).Each dose group was given only once.After an overnight stay of at least 10h on an empty stomach, 240mL of water was administered in the morning under the condition of an empty stomach. Water was forbidden for 1h before and 1h after administration, and fasting for 4h after administration.
placebo tabletPLACEBO_COMPARATORIncluding 7 dose groups(2.5-、5、10-、20-、40-、60-、80mg).Each dose group was given only once.After an overnight stay of at least 10h on an empty stomach, 240mL of water was administered in the morning under the condition of an empty stomach. Water was forbidden for 1h before and 1h after administration, and fasting for 4h after administration.

Interventions

NameTypeDescription
HEC113995PA•H2O tabletDRUG2.5-、5-、10-、20-、40-、60-、80mg HEC113995PA•H2O tablet in day1.
Placebo tabletDRUG2.5-、5-、10-、20-、40-、60-、80mg Placebo tablet in day1.
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 45 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Willing to participate in the study, able to understand and sign the informed consent, and able to complete the the study in accordance with the requirements of the study. * Female subjects who are not pregnant or lactating and male subjects whose female partners are fertile s...

Countries:China
Unlock Eligibility Criteria

Frequently asked questions about HEC113995PA•H2O

What is HEC113995 PA•H2O used for?

HEC113995 PA•H2O is an investigational small molecule being studied for the treatment of Major Depressive Disorder. It is also being evaluated in healthy subjects to assess its safety, tolerability, and pharmacokinetics. The drug is currently in Phase 1 clinical development and is not yet approved by regulatory authorities.

What does HEC113995 PA•H2O target?

HEC113995 PA•H2O is described as a selective serotonin partial agonist and reuptake inhibitor. This means it is designed to interact with serotonin pathways in the brain, acting as a partial agonist at serotonin receptors and inhibiting serotonin reuptake, which may help regulate mood in Major Depressive Disorder.

Who makes HEC113995 PA•H2O?

HEC113995 PA•H2O is being developed by Sunshine Biopharma Inc., a company listed on the stock exchange under the ticker symbol SBFM. The company is conducting clinical trials to evaluate the drug's safety and efficacy in treating Major Depressive Disorder.

What phase is HEC113995 PA•H2O in?

HEC113995 PA•H2O is in Phase 1 clinical development. Two Phase 1 trials have been completed, both involving healthy subjects. The drug is still investigational and has not received FDA approval. It is being studied for its safety, tolerability, and pharmacokinetic profile.

What clinical trials is HEC113995 PA•H2O in?

HEC113995 PA•H2O has been studied in two completed Phase 1 clinical trials. The first, NCT03943251, evaluated the drug in healthy subjects in China. The second, NCT04591301, assessed the safety, tolerability, and pharmacokinetics of HEC113995 PA•H2O tablets in healthy subjects, also in China. Both trials were randomized, double-blind, and placebo-controlled.

Is HEC113995 PA•H2O the same as HEC113995?

HEC113995 PA•H2O is a specific form of the drug HEC113995, where PA•H2O refers to the particular salt or hydrate form used in the clinical trials. The trials listed for this drug use the name HEC113995 PA•H2O, indicating it is the active pharmaceutical ingredient in this specific formulation.