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Olutasidenib Investigational Agent Administration

Phase 1

Acute Myeloid Leukemia | Small molecule | Oncology |Rigel Pharmaceuticals, Inc.|Last Updated: Feb 6, 2026

Target and mechanism

Molecular targetIDH1
Target classInhibitor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment15

FDA Designations

No designations recorded

Clinical trial landscape

Olutasidenib Investigational Agent Administration · 1 trial · 1 indication

Phase 1 1
NCT07130695Olutasidenib Single Plus Combo Therapy in IDH1mut AML After Induction and ConsolidationAcute Myeloid Leukemia
RECRUITING15 Analytics
PHASE1RECRUITING
Olutasidenib Single Plus Combo Therapy in IDH1mut AML After Induction and Consolidation
Acute Myeloid LeukemiaUnlock trial analytics

Study Endpoints

Primary Endpoints

Assess the feasibility of olutasidenib after upfront acute myeloid leukemia (AML) therapy with intensive induction and/or consolidation in IDH1 mutant AML.
Up to 2 years

Feasibility defined as the number of participants with 75% protocol treatment compliance for a duration of at least 4 cycles (to include protocol defined dose delays), or until disease relapse or allogeneic hematopoietic stem cell transplant (alloHCT).

Assess the tolerability of olutasidenib after upfront AML therapy with intensive induction and/or consolidation in IDH1 mutant AML
Up to 2 years

Incidence of grade ≥4 adverse events (AEs) attributable to study drug for duration of treatment on study

Secondary Endpoints

Measure progression free survival
Up to 2 years following end of treatment
Estimate overall survival (OS)
Up to 2 years following end of treatment
Assess mean residual disease (MRD) negativity rates by both PCR based and flow cytometric methodologies
Baseline, Cycle 3 Day 15, and End of Treatment (Each cycle is 28 days)
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Olutasidenib Investigational Agent AdministrationEXPERIMENTAL150 mg by mouth twice daily.

Interventions

NameTypeDescription
Olutasidenib Investigational Agent AdministrationDRUGTwice daily olutasidenib maintenance therapy
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Histologically or cytologically confirmed non-acute promyelocytic isocitrate dehydrogenase (1 IDH1) mutant acute myeloid leukemia (AML). IDH1 mutation may be identified by NGS or PCR based methods and identified at time of diagnosis or any other time point prior to enrollment....

Countries:United States
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Frequently asked questions about Olutasidenib Investigational Agent Administration

What is Olutasidenib Investigational Agent Administration used for?

Olutasidenib Investigational Agent Administration is an investigational small molecule being studied for the treatment of Acute Myeloid Leukemia (AML). It is currently in Phase 1 clinical development and is not yet approved by the FDA. The drug is being evaluated in patients with IDH1-mutant AML.

What does Olutasidenib Investigational Agent Administration target?

Olutasidenib Investigational Agent Administration is a kinase inhibitor, as indicated by its '-nib' suffix. It is being studied in biomarker-selected patients with IDH1 mutations. The drug is intended to target the mutated IDH1 enzyme in Acute Myeloid Leukemia, though specific molecular details are not provided.

Who is developing Olutasidenib Investigational Agent Administration?

Olutasidenib Investigational Agent Administration is being developed by Rigel Pharmaceuticals, Inc., a biopharmaceutical company traded on the NASDAQ under the ticker symbol RIGL. The company is conducting clinical trials to evaluate the drug's safety and efficacy in patients with Acute Myeloid Leukemia.

What phase is Olutasidenib Investigational Agent Administration in?

Olutasidenib Investigational Agent Administration is in Phase 1 clinical development. It is an investigational drug, meaning it has not been approved by the FDA for any use. The ongoing Phase 1 trial is currently recruiting participants to study the drug in Acute Myeloid Leukemia.

What clinical trials is Olutasidenib Investigational Agent Administration in?

Olutasidenib Investigational Agent Administration is being studied in one active Phase 1 clinical trial with the identifier NCT07130695. The trial, titled 'Olutasidenib Single Plus Combo Therapy in IDH1mut AML After Induction and Consolidation,' is recruiting 15 participants in the United States. It is an uncontrolled, non-randomized, open-label study.

Is Olutasidenib Investigational Agent Administration the same as olutasidenib?

Olutasidenib Investigational Agent Administration is a formulation or administration method of the drug olutasidenib. The clinical trial NCT07130695 evaluates olutasidenib as a single agent and in combination therapy. The drug is being developed by Rigel Pharmaceuticals for Acute Myeloid Leukemia.