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nacubactam

Phase 1

Gram-negative Bacterial Infections | Small molecule | Infectious Disease |Roche Holding AG|Last Updated: Apr 23, 2018

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment21

FDA Designations

No designations recorded

Clinical trial landscape

nacubactam · 1 trial · 1 indication

Phase 1 1
NCT03182504A Study to Investigate the Intrapulmonary Lung Penetration of Nacubactam in Healthy ParticipantsGram-negative Bacterial Infections
COMPLETED21 Analytics
PHASE1COMPLETED
A Study to Investigate the Intrapulmonary Lung Penetration of Nacubactam in Healthy Participants
Gram-negative Bacterial InfectionsUnlock trial analytics

Study Endpoints

Primary Endpoints

Epithelial Lining Fluid (ELF) Concentration of Nacubactam to Plasma Concentration of Nacubactam Ratio
At 2, 3, 4, 6 and 8 hours after study drug administration

The ELF to plasma ratio will be calculated from the concentration of nacubactam in ELF and plasma as a measure of the intrapulmonary penetration of nacubactam in healthy participants.

Secondary Endpoints

ELF Concentration of Meropenem to Plasma Concentration of Meropenem Ratio
At 2, 3, 4, 6 and 8 hours after study drug administration
Area Under the Plasma Concentration-Time Curve from time 0 to 8 hours (AUC0-8) of Nacubactam in ELF
At 2, 3, 4, 6 and 8 hours after study drug administration
Maximum Concentration (Cmax) of Nacubactam in ELF
At 2, 3, 4, 6 and 8 hours after study drug administration
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Nacubactam Plus MeropenemEXPERIMENTALParticipants will receive a single dose of nacubactam co-administered with meropenem.

Interventions

NameTypeDescription
nacubactamDRUGParticipants will receive a single 2000 milligram (mg) intravenous (IV) infusion of nacubactam over 1.5 hours.
meropenemDRUGParticipants will receive a single 2000 mg IV infusion of meropenem over 1.5 hours.
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Eligibility Criteria

Age Range18 Years to 60 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * 18 to 60 years of age, inclusive * Healthy, as judged by the Investigator and defined by the absence of evidence of any active or clinically significant chronic disease identified from a detailed medical and surgical history, physical examination including vital signs and 12-l...

Countries:United States
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Frequently asked questions about nacubactam

What is nacubactam used for?

Nacubactam is an investigational small molecule being developed for Gram-negative bacterial infections. It is currently in Phase 1 clinical development and is not approved by the FDA. The drug is being studied for its ability to treat infections caused by Gram-negative bacteria.

Who makes nacubactam?

Nacubactam is being developed by Roche Holding AG, which trades under the ticker RHHBY. The company is conducting clinical trials to evaluate the drug's safety and pharmacokinetics in healthy volunteers.

What phase is nacubactam in?

Nacubactam is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and the drug remains in early-stage clinical testing.

What clinical trials is nacubactam in?

Nacubactam has one completed Phase 1 trial, NCT03182504, which investigated the intrapulmonary lung penetration of the drug in healthy participants. The study enrolled 21 participants in the United States and was an uncontrolled, open-label trial.

Is nacubactam FDA approved?

No, nacubactam is not FDA approved. It is an investigational drug currently in Phase 1 clinical development. The completed trial focused on lung penetration in healthy volunteers, and further studies would be needed to establish safety and efficacy.