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RO6864018

Phase 1

Healthy Volunteer | Small molecule | Other |Roche Holding AG|Last Updated: Mar 1, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment48

FDA Designations

No designations recorded

Clinical trial landscape

RO6864018 · 1 trial · 1 indication

Phase 1 1
NCT02015715A Study Evaluating the Safety, Pharmacokinetics, and Pharmacodynamics of RO6864018 in Male, Healthy, Asian ParticipantsHealthy Volunteer
COMPLETED48 Analytics
PHASE1COMPLETED
A Study Evaluating the Safety, Pharmacokinetics, and Pharmacodynamics of RO6864018 in Male, Healthy, Asian Participants
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Study Endpoints

Primary Endpoints

Number of Participants With Adverse Events
Baseline up to Day 29

Secondary Endpoints

Area Under the Plasma Concentration Time Curve From Time Zero to Infinity (AUC0-inf) of RO6864018
Pre-dose (0 hour), 0.25, 0.5, 1, 1.5, 2, 3, 4, 8, 12, 18, 24, 36 and 48 hours post-Day 1 dose
AUC0-inf of Active Metabolite RO6871765
Pre-dose (0 hour), 0.25, 0.5, 1, 1.5, 2, 3, 4, 8, 12, 18, 24, 36 and 48 hours post-Day 1 dose
AUC0-inf of Prodrug Metabolite RO6870868
Pre-dose (0 hour), 0.25, 0.5, 1, 1.5, 2, 3, 4, 8, 12, 18, 24, 36 and 48 hours post-Day 1 dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
RO6864018EXPERIMENTALAsian participants will receive a single oral dose of RO6864018 capsule on Day 1. The first dose escalation cohort will receive a single 400 mg oral dose. Dose will be escalated in subsequent cohorts (up to Cohort 4) up to a maximum of 1600 mg, based on safety, pharmacokinetic, and pharmacodynamic data available from lower dose cohorts. The Cohort 5 will include Caucasian participants who will receive a single 1200 mg (or the highest dose well-tolerated by Asian participants, if lower than 1200 mg) oral dose of RO6864018 capsules on Day 1.
PlaceboPLACEBO_COMPARATORParticipants will receive a single oral dose of placebo matching to RO6864018.

Interventions

NameTypeDescription
RO6864018DRUGA single oral ascending dose of RO6864018 capsules on Day 1.
PlaceboDRUGA single oral dose of placebo matching RO6864018 capsules on Day 1.
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Eligibility Criteria

Age Range21 Years to 65 Years
SexMALE
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Healthy male participants of ethnic Chinese, Korean, Japanese origin or Caucasian * No signs of any active or chronic disease following a detailed medical and surgical history, a complete physical examination including vital signs, 12-lead electrocardiogram (ECG), hematology, ...

Countries:Singapore
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Frequently asked questions about RO6864018

What is RO6864018?

RO6864018 is an investigational small molecule being developed by Roche Holding AG (RHHBY). It is currently in Phase 1 clinical development. The drug has been studied in a completed trial involving healthy volunteers, with a focus on evaluating its safety, pharmacokinetics, and pharmacodynamics.

What is RO6864018 used for?

RO6864018 is being studied for use in healthy volunteers. The completed Phase 1 trial assessed the drug's safety, pharmacokinetics, and pharmacodynamics in this population. It is not approved for any medical condition and remains in clinical development.

Who makes RO6864018?

RO6864018 is developed by Roche Holding AG, which trades under the ticker RHHBY. The company is conducting clinical research on this investigational small molecule, which is currently in Phase 1 development.

What phase is RO6864018 in?

RO6864018 is in Phase 1 clinical development. A single Phase 1 trial has been completed, and the drug is not yet approved. It remains an investigational agent under study.

What clinical trials is RO6864018 in?

RO6864018 has one completed clinical trial, identified as NCT02015715. This Phase 1 study evaluated the safety, pharmacokinetics, and pharmacodynamics of RO6864018 in male, healthy Asian participants in Singapore. The trial enrolled 48 participants and was placebo-controlled and double-blind.

Is RO6864018 the same as any other drug?

RO6864018 is the sole name provided for this investigational drug. No alternative names have been associated with it in the available clinical trial information.