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RO5285119

Phase 1

Healthy Volunteer | Small molecule | Other |Roche Holding AG|Last Updated: Nov 2, 2016

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials4
Total Enrollment135

FDA Designations

No designations recorded

Clinical trial landscape

RO5285119 · 4 trials · 1 indication

Phase 1 4
NCT02179866A Single-center Study to Investigate How Quickly and to What Extent a Radioactive Dose of RO5285119 is Absorbed, Metabolized and Eliminated From the Body of Healthy Male VolunteersHealthy Volunteer
COMPLETED6 Analytics
NCT01967979A Study of the Effect of Multiple Doses of Itraconazole and Fluoxetine on the Pharmacokinetics of a Single Dose of RO5285119 in Healthy SubjectsHealthy Volunteer
COMPLETED28 Analytics
NCT01708616A Study of the Combination of Multiple Doses of RO5285119 With a Single Dose of Risperidone in Healthy VolunteersHealthy Volunteer
COMPLETED24 Analytics
NCT01418963A Study of RO5285119 in Healthy VolunteersHealthy Volunteer
COMPLETED77 Analytics
PHASE1COMPLETED
A Single-center Study to Investigate How Quickly and to What Extent a Radioactive Dose of RO5285119 is Absorbed, Metabolized and Eliminated From the Body of Healthy Male Volunteers
Healthy VolunteerUnlock trial analytics
PHASE1COMPLETED
A Study of the Effect of Multiple Doses of Itraconazole and Fluoxetine on the Pharmacokinetics of a Single Dose of RO5285119 in Healthy Subjects
Healthy VolunteerUnlock trial analytics
PHASE1COMPLETED
A Study of the Combination of Multiple Doses of RO5285119 With a Single Dose of Risperidone in Healthy Volunteers
Healthy VolunteerUnlock trial analytics
PHASE1COMPLETED
A Study of RO5285119 in Healthy Volunteers
Healthy VolunteerUnlock trial analytics

Study Endpoints

Primary Endpoints

Total recovery of radioactivity over time in urine and feces expressed as a percentage of the total radioactive dose administered
Up to Day 17
Pharmacokinetic profile of total drug-related material, RO5285119 and its metabolites, as appropriate in plasma, estimated Cmax
Up to Day 17
Effect of multiple doses of itraconazole and fluoxetine on the pharmacokinetics of a single dose of RO5285119 in healthy volunteers: Maximum concentration (Cmax) / Area under the concentration-time curve (AUC)
up to 5 and 7 days post-dose for cohort 1 and cohort 2, respectively
Pharmacokinetics of single dose risperidone in combination with multiple doses of RO5285119: Maximum plasma concentration (Cmax)
Pre-dose to 24 hours post-dose
Pharmacokinetics of single dose risperidone in combination with multiple doses of RO5285119: Area under the concentration-time curve (AUC)
Pre-dose to 24 hours post-dose
Safety: Incidence of adverse events
up to 5 weeks

Secondary Endpoints

Percent of dose recovered as total radioactivity, i.e. relative abundance of RO5285119 and its metabolite(s) in plasma, urine and feces
Up to Day 17
Incidence of adverse events
Up to 28 days after the last dose of study drug
Safety and tolerability of a single dose of RO5285119 administered in combination with itraconazole (cohort 1) and fluoxetine (cohort 2): Incidence of adverse events
up to 6 weeks
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP

Treatment Arms

ArmTypeDescription
[14C]-labeled RO5285119EXPERIMENTALSingle oral dose - drinking solution
Cohort 1 (Itraconazole DDI)EXPERIMENTAL -
Cohort 2 (Fluoxetine DDI)EXPERIMENTAL -
Placebo + risperidonePLACEBO_COMPARATOR -
Placebo +placeboPLACEBO_COMPARATOR -
RO5285119 + placeboACTIVE_COMPARATOR -
RO5285119 + risperidoneEXPERIMENTAL -
ActiveEXPERIMENTAL -
PlaceboPLACEBO_COMPARATOR -

Interventions

NameTypeDescription
RO5285119DRUGSingle oral dose of RO5285119 with approximately 2.1 MBq (56.6 uCi) \[14C\]-radiolabeled RO5285119 administered as a drinking solution under fasted conditions on Day -1
fluoxetineDRUGMultiple doses
itraconazoleDRUGMultiple doses
RO5285119 placeboDRUGmultiple doses
risperidoneDRUGsingle dose
risperidone placeboDRUGsingle dose
placeboDRUGsingle and multiple oral doses
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Eligibility Criteria

Age Range35 Years to 64 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male participants, 35 to 64 years of age, inclusive * For men with a female partner of child-bearing potential: Agreement to use two methods of contraception, including one barrier method e.g. condom, during the treatment period and for at least 3 months after the last...

Countries:NetherlandsFrance
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Frequently asked questions about RO5285119

What is RO5285119?

RO5285119 is an investigational small molecule being developed by Roche Holding AG (RHHBY). It has been studied in healthy volunteers in Phase 1 clinical trials. The drug is not approved and remains in clinical development.

What is RO5285119 used for?

RO5285119 has been studied in healthy volunteers, meaning it is not yet being tested in patients with a specific disease. Its intended therapeutic use has not been established, as it is still in early-stage clinical development.

Who makes RO5285119?

RO5285119 is being developed by Roche Holding AG, which trades under the ticker RHHBY. Roche has sponsored multiple Phase 1 clinical trials of the drug in healthy volunteers.

What phase is RO5285119 in?

RO5285119 is in Phase 1 clinical development. All four completed trials were Phase 1 studies, and the drug is still investigational. It has not been approved by regulatory authorities.

What clinical trials is RO5285119 in?

RO5285119 has been studied in four completed Phase 1 trials: NCT01418963, NCT01708616, NCT01967979, and NCT02179866. These trials enrolled a total of 135 healthy volunteers and were conducted in France and the Netherlands.

Is RO5285119 the same as risperidone?

No, RO5285119 is not the same as risperidone. One clinical trial, NCT01708616, studied the combination of multiple doses of RO5285119 with a single dose of risperidone in healthy volunteers, but they are distinct drugs.