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RO5045337

Phase 1

Hematologic Neoplasms | Small molecule | Oncology |Roche Holding AG|Last Updated: Jul 7, 2017

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment116

FDA Designations

No designations recorded

Clinical trial landscape

RO5045337 · 6 trials · 4 indications

Phase 1 6
NCT01677780An Extension Study of RO5045337 in Participants Participating in Previous Roche-sponsored Cancer StudiesMyelogenous Leukemia, Chronic, Neoplasms, Myelogenous Leukemia, Acute
COMPLETED11 Analytics
NCT01605526A Study of RO5045337 in Combination With Doxorubicin in Patients With Soft Tissue SarcomaSarcoma
COMPLETED23 Analytics
NCT01164033A Study of RO5045337 in Patients With Solid TumorsNeoplasms
COMPLETED76 Analytics
NCT01143740A Study of RO5045337 in Patients With Liposarcomas Prior to Debulking SurgerySarcoma
COMPLETED20 Analytics
NCT00623870A Study of RO5045337 [RG7112] in Patients With Hematologic Neoplasms.Hematologic Neoplasms
COMPLETED116 Analytics
NCT00559533A Study of RO5045337 [RG7112] in Patients With Advanced Solid TumorsNeoplasms
COMPLETED106 Analytics
PHASE1COMPLETED
An Extension Study of RO5045337 in Participants Participating in Previous Roche-sponsored Cancer Studies
Myelogenous Leukemia, Chronic, Neoplasms, Myelogenous Leukemia, AcuteUnlock trial analytics
PHASE1COMPLETED
A Study of RO5045337 in Combination With Doxorubicin in Patients With Soft Tissue Sarcoma
SarcomaUnlock trial analytics
PHASE1COMPLETED
A Study of RO5045337 in Patients With Solid Tumors
NeoplasmsUnlock trial analytics
PHASE1COMPLETED
A Study of RO5045337 in Patients With Liposarcomas Prior to Debulking Surgery
SarcomaUnlock trial analytics
PHASE1COMPLETED
A Study of RO5045337 [RG7112] in Patients With Hematologic Neoplasms.
Hematologic NeoplasmsUnlock trial analytics
PHASE1COMPLETED
A Study of RO5045337 [RG7112] in Patients With Advanced Solid Tumors
NeoplasmsUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs)
Approximately 24 months
Maximum tolerated dose/dose-limiting toxicities
approximately 12 months
Safety: Incidence of adverse events
approximately 12 months
Examination of potential food-effect on pharmacokinetics of RO5045337
3 weeks
Evaluation of relative bioavailability of RO5045337
3 weeks
Biomarker evidence of MDM2 and p53 pathway alterations (histologic, molecular and imaging analyses)
from baseline to week 12
Comparison of daily versus twice daily dosing: Incidence of adverse events
approximately 4.5 years
MTD and associated dose schedule
Every 28 days

Secondary Endpoints

Pharmacokinetics of RO5045337 and doxorubicin in combination therapy: Area under the concentration-time curve (AUC)
Pre-dose and up to 72 hours post-dose Days 1 and 5 of Cycle 1
Pharmacodynamics: Serum macrophage inhibitory cytokine-1 (MIC-1) levels
Pre-dose and up to 72 hours post-dose on Days 1 and 5 of Cycle 1
Evaluation of safety and tolerability of RO5045337
3 weeks
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
RO5045337EXPERIMENTALParticipants will continue the most similar dose and formulation available (which does not exceed the MTD or the maximum safely administered dose for that formulation during Phase 1) and the same schedule of RO5045337 treatment that they were receiving at the time of transitioning from their respective parent clinical study protocols: NO21279 (NCT00623870), NO21280 (NCT00559533), NP25299 (NCT01164033), NP28021 (NCT01605526) or NP28023 (NCT01635296).
Single ArmEXPERIMENTAL -
AACTIVE_COMPARATOR -
BEXPERIMENTAL -
CEXPERIMENTAL -
DEXPERIMENTAL -
1EXPERIMENTAL -

Interventions

NameTypeDescription
RO5045337DRUGParticipants will receive RO5045337 orally in doses ranging from 20 milligram per square meter (mg/m\^2) to 1800 mg/m\^2 daily, and up to 1500 mg dose twice daily on a variety of schedules including daily for up to 20 days and weekly dosing for 3 weeks in 28 day cycles until disease progression or unacceptable toxicity with maximum treatment duration of 24 months.
doxorubicinDRUG60 mg/m2 (75 mg/m2, 50 mg/m2) iv on Day 1 of each 28-day cycle, up to 6 cycles
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites5

Inclusion Criteria: * Participants must meet the inclusion criteria outlined in the respective parent protocols: NO21279 (NCT00623870), NO21280 (NCT00559533), NP25299 (NCT01164033), NP28021 (NCT01605526) or NP28023 (NCT01635296) * Participants must have completed one of the following clinical study...

Countries:United StatesCanadaFranceItalyUnited Kingdom
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Frequently asked questions about RO5045337

What is RO5045337 used for?

RO5045337 is an investigational small molecule being studied for the treatment of various cancers, including solid tumors, hematologic neoplasms, chronic and acute myelogenous leukemia, and sarcoma. It is in Phase 1 clinical development and is not yet approved by regulatory authorities.

Who makes RO5045337?

RO5045337 is being developed by Roche Holding AG, a multinational healthcare company. Roche's stock is traded under the ticker symbol RHHBY on the OTC market.

What phase is RO5045337 in?

RO5045337 is in Phase 1 clinical development. All four clinical trials listed for the drug are Phase 1 studies and have been completed. The drug remains investigational and has not received regulatory approval.

What clinical trials is RO5045337 in?

RO5045337 has been studied in four completed Phase 1 trials: NCT00559533 in advanced solid tumors, NCT01143740 in liposarcomas prior to debulking surgery, NCT01164033 in solid tumors, and NCT01605526 in combination with doxorubicin for soft tissue sarcoma. These trials enrolled a total of 182 patients.

Is RO5045337 the same as RG7112?

Yes, RO5045337 is also known as RG7112. The clinical trial NCT00559533, titled 'A Study of RO5045337 [RG7112] in Patients With Advanced Solid Tumors,' confirms that both names refer to the same investigational drug.