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RO4998452

Phase 2

Diabetes Mellitus Type 2 | Small molecule | Metabolic |Roche Holding AG|Last Updated: Nov 18, 2020

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLED
Total Trials4
Total Enrollment507

FDA Designations

No designations recorded

Clinical trial landscape

RO4998452 · 4 trials · 1 indication

Phase 2 1Phase 1 3
NCT00800176A Dose-Finding Study of RO4998452 in Patients With Diabetes MellitusDiabetes Mellitus Type 2
COMPLETED394 Analytics
PHASE2COMPLETED
A Dose-Finding Study of RO4998452 in Patients With Diabetes Mellitus
Diabetes Mellitus Type 2Unlock trial analytics

Study Endpoints

Primary Endpoints

Absolute Change in HbA1c
Baseline, Week 4, Week 8 and Week 12
Effect on postprandial plasma glucose concentration
Following meal 13 hours after dosing
Creatinine clearance; Pk parameters; adverse events
Days 1-3
AEs, laboratory parameters, vital signs.
Throughout study
AUC0-24h, Cmax
Days 1 and 14

Secondary Endpoints

Change From Baseline in Fasting Plasma Glucose (mmol/L)
Baseline and Week 12
Change From Baseline in Mean Daily Glucose Concentration (mmol/L)
Baseline and Week 12
Change From Baseline in Fructosamine Concentration (μmol/L)
Baseline and 12 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
PlaceboPLACEBO_COMPARATORDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test.
RO4998452 10mgEXPERIMENTALDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test. The two capsules combined contained 10 mg of RO4998452.
RO4998452 2.5mgEXPERIMENTALDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test. The two capsules combined contained 2.5 mg of RO4998452.
RO4998452 20mgEXPERIMENTALDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test. The two capsules combined contained 20 mg of RO4998452.
RO4998452 40mgEXPERIMENTALDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test. The two capsules combined contained 40 mg of RO4998452.
RO4998452 5mgEXPERIMENTALDuring the single-blind run-in period, two placebo capsules were taken in the morning approximately 15 minutes prior to breakfast. During the 12-week double-blind treatment period, two capsules were taken in the morning approximately 15 minutes prior to breakfast, except on the days of the meal tolerance test. The two capsules combined contained 5 mg of RO4998452.
AEXPERIMENTAL -
BEXPERIMENTAL -
CPLACEBO_COMPARATOR -
1 (normal)EXPERIMENTAL -
2 (mild)EXPERIMENTAL -
3 (moderate)EXPERIMENTAL -
4 (severe)EXPERIMENTAL -
1EXPERIMENTAL -
2EXPERIMENTAL -
3EXPERIMENTAL -
4EXPERIMENTAL -
5EXPERIMENTAL -
6EXPERIMENTAL -
7EXPERIMENTAL -

Interventions

NameTypeDescription
PlaceboDRUGpo daily for 12 weeks
RO4998452DRUG2.5mg po daily for 12 weeks
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Eligibility Criteria

Age Range18 Years to 75 Years
SexALL
Healthy VolunteersNo
Study Sites67

Inclusion Criteria: * adult patients, 18-75 years of age; * type 2 diabetes, diagnosed for \>=3 months; * either treated with diet, exercise and stable metformin, or with diet and exercise alone. Exclusion Criteria: * type 1 diabetes mellitus; * currently or within 2 months prior to screening tre...

Countries:United StatesAustraliaBrazilCanadaGermanyHong KongJapanLatviaMexicoRomaniaRussiaSpainFrance
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Frequently asked questions about RO4998452

What is RO4998452 used for?

RO4998452 is an investigational small molecule being developed for the treatment of Type 2 Diabetes Mellitus. It is in Phase 2 clinical development and has been studied in patients with this condition across multiple trials.

Who makes RO4998452?

RO4998452 is being developed by Roche Holding AG, which trades under the ticker RHHBY. The company has sponsored clinical trials of this investigational drug in patients with Type 2 Diabetes Mellitus.

What phase is RO4998452 in?

RO4998452 is in Phase 2 clinical development. It has completed four clinical trials, including a Phase 2 dose-finding study, and is not yet approved by regulatory authorities.

What clinical trials is RO4998452 in?

RO4998452 has completed four clinical trials: NCT00682097, a Phase 1 multiple ascending dose study; NCT00800176, a Phase 2 dose-finding study; NCT00933972, a Phase 1 study in patients with renal impairment; and NCT01044017, a Phase 1 single dose study. All trials enrolled patients with Type 2 Diabetes Mellitus.

Is RO4998452 the same as any other drug?

No alternative names for RO4998452 have been identified in the available information. It is referred to solely by its code name RO4998452 in clinical trial records.