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GDC-0810 Phase II

Phase 1

Healthy Volunteer | Small molecule | Other |Roche Holding AG|Last Updated: Aug 22, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment45

FDA Designations

No designations recorded

Clinical trial landscape

GDC-0810 Phase II · 1 trial · 1 indication

Phase 1 1
NCT02722018Study to Investigate the Effect of Formulation and Food on the Pharmacokinetics of GDC-0810Healthy Volunteer
COMPLETED45 Analytics
PHASE1COMPLETED
Study to Investigate the Effect of Formulation and Food on the Pharmacokinetics of GDC-0810
Healthy VolunteerUnlock trial analytics

Study Endpoints

Primary Endpoints

Maximum Observed Plasma Concentration (Cmax) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Time to Reach Cmax (Tmax) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Area Under the Plasma Concentration Versus Time Curve From Time Zero to Time of Last Quantifiable Concentration (AUC0-t) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Area Under the Plasma Concentration Versus Time Curve From Time Zero to Extrapolated Infinite Time (AUC0-inf) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Apparent Terminal Elimination Rate Constant (lambda Z) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Apparent Terminal Elimination Half-Life (t1/2) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Apparent Oral Clearance (CL/F) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Apparent Volume of Distribution (Vz/F) of GDC-0810
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Relative Bioavailability Based on Cmax (Frel Cmax) of GDC-0810 (Test vs Reference)
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Relative Bioavailability Based on AUC0-t (Frel AUC0-t) of GDC-0810 (Test vs Reference)
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Relative Bioavailability Based on Cmax (Frel Cmax) of GDC-0810 (Fed vs Fasted)
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period
Relative Bioavailability Based on AUC0-t (Frel AUC0-t) of GDC-0810 (Fed vs Fasted)
Pre-dose (1 hour before dosing), 0.5, 1, 2, 3, 4, 6, 8, 12, 16 hours post-dose on Day 1, 24 and 36 hours post-dose (Day 2), 48 hours post-dose (Day 3) of each treatment period

Secondary Endpoints

Number of Participants With Adverse Events (AEs)
Baseline up to 28 days after last GDC-0810 dose (Up to 57 days)
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part 1: GDC-0810 dose level A - Low Fat MealEXPERIMENTALParticipants will receive a single dose of GDC-0810 dose level A on Day 1 of each treatment period. GDC-0810 will be administered with low fat meal in the form of Phase II tablet or one of three Phase III prototype tablets (Prototype 1, 2 or 3) in a crossover fashion.
Part 2 (Optional): GDC-0810 dose level A - Low Fat MealEXPERIMENTALParticipants will receive a single dose of GDC-0810 dose level A on Day 1 of each treatment period. GDC-0810 will be administered with low fat meal in the form of Phase II tablet or one of two Phase III prototype tablets (Prototype 4 or 5) in a crossover fashion.
Part 3: GDC-0810 dose level B - Low Fat Meal/FastedEXPERIMENTALParticipants will receive a single dose of GDC-0810 dose level B on Day 1 of each treatment period. GDC-0810 will be administered with low fat meal or under fasted condition either as Phase II tablet (with low fat meal) or as the Phase III prototype tablet selected from Parts 1 or 2 (with low fat meal or under fasted conditions), in a crossover fashion.

Interventions

NameTypeDescription
GDC-0810 Phase II TabletDRUGParticipants will receive dose level A (in Parts 1 and 2) or dose level B (in Part 3) tablets.
GDC-0810 Phase III Prototype TabletDRUGParticipants will receive dose level A (in Parts 1 and 2) or dose level B (in Part 3) tablets.
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Eligibility Criteria

Age Range40 Years to 70 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Female participants of non-childbearing potential including non-pregnant, non-lactating, and either postmenopausal or surgically sterile for at least 45 days post procedure * Body mass index (BMI) range 18.0 to 32.0 kilograms per square meter (kg/m\^2), inclusive * In good hea...

Countries:United Kingdom
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Frequently asked questions about GDC-0810 Phase II

What is GDC-0810 Phase II used for?

GDC-0810 Phase II is a small molecule being studied in healthy volunteers. It is currently in Phase 1 clinical development, not Phase 2, and is being investigated for its pharmacokinetic properties, including the effect of formulation and food on its absorption. The drug is not approved and remains investigational.

Who makes GDC-0810 Phase II?

GDC-0810 Phase II is being developed by Roche Holding AG, which trades under the ticker RHHBY. The company is conducting clinical trials to evaluate the drug's pharmacokinetics in healthy volunteers. Roche is the sole developer listed for this asset.

What phase is GDC-0810 Phase II in?

GDC-0810 Phase II is in Phase 1 clinical development, despite its name suggesting a later stage. It is an investigational small molecule being studied in healthy volunteers. The drug has not been approved by regulatory authorities and is still undergoing clinical trials.

What clinical trials is GDC-0810 Phase II in?

GDC-0810 Phase II is associated with one completed clinical trial, NCT02722018, titled 'Study to Investigate the Effect of Formulation and Food on the Pharmacokinetics of GDC-0810.' This Phase 1 study enrolled 45 healthy female volunteers in the United Kingdom and was controlled but not double-blinded.

Is GDC-0810 Phase II the same as GDC-0810?

GDC-0810 Phase II appears to be a designation for the drug GDC-0810, which is being studied in a Phase 1 trial. The name 'Phase II' may refer to a specific formulation or study stage, but the active ingredient is GDC-0810. No alternative names are provided for this asset.