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GDC-0032 Phase III

Phase 1

Healthy Volunteer | Small molecule | Other |Roche Holding AG|Last Updated: Feb 1, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment76

FDA Designations

No designations recorded

Clinical trial landscape

GDC-0032 Phase III · 1 trial · 1 indication

Phase 1 1
NCT01980953A Study to Evaluate the Effect of Particle Size, Formulation and Food on the Pharmacokinetics of GDC-0032 in Healthy VolunteersHealthy Volunteer
COMPLETED76 Analytics
PHASE1COMPLETED
A Study to Evaluate the Effect of Particle Size, Formulation and Food on the Pharmacokinetics of GDC-0032 in Healthy Volunteers
Healthy VolunteerUnlock trial analytics

Study Endpoints

Primary Endpoints

Area Under the Concentration-Time Curve From Hour 0 to the Last Measurable Concentration (AUC0-t)
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour post-dose
Area Under the Concentration-Time Curve Extrapolated to Infinity (AUC0-infinity)
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour post-dose
Maximum Plasma Concentration (Cmax)
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour postdose

Secondary Endpoints

Time to Maximum Plasma Concentration (tmax)
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour post-dose
Apparent Terminal Elimination Rate Constant
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour post-dose
Apparent Terminal Elimination Constant (t1/2)
Pre-dose (Hour 0), 0.5, 1, 2, 4, 6, 8, 12, 24, 48, 72, 96, 168, 192 hour post-dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Part 1: Food EffectEXPERIMENTALGDC-0032 will be administered orally over 3-Treatment Period (TP) in 6-sequence as one 3 milligrams (mg) capsule in TP-A after 10 hour fasting from food, one 3 mg Phase III tablet in TP-B after 10 hour fasting from food and one 3 mg Phase III tablet in TP-C following the start of standard Food and Drug Administration (FDA) high-fat breakfast. Washout period o 14 to 20 days will be given between each TP.
Part 2: Tablet Formulation ComparisonEXPERIMENTALDifferent formulations of tablets (Tablet A and Tablet B) of GDC-0032 will be administered orally over 2-TP having 10 hour fasting from food. Participants will receive one 3 mg Tablet A in TP-A and one 3 mg Tablet B in TP-B after 14 to 20 days washout period.
Part 3: Capsule API Lot ComparisonEXPERIMENTALTwo different lots of GDC-0032 active pharmaceutical ingredient (API) capsule formulation will be administered orally in crossover fashion over 2-TP to 20 participants having 10 hour fasting from food. Participants will receive one 3 mg capsule in TP-A and one 3 mg capsule in TP-B after 14 to 20 days washout period.
Part 4: Tablet Relative BioavailibityEXPERIMENTALGDC-0032 will be administered orally in crossover fashion over 2-TP to 20 participants having 10 hour fasting from food. Participants will receive one 3 mg capsule in TP-A and one 2 mg Phase III tablet in TP-B after 14 to 20 days washout period.

Interventions

NameTypeDescription
GDC-0032 Phase III TabletDRUGParticipants will receive 2 mg or 3 mg Phase III tablet after 10 hour fasting from food.
GDC-0032 TabletDRUGParticipants will receive 3 mg Tablet A or Tablet B formulation after 10 hour fasting from food.
GDC-0032 CapsuleDRUGParticipants will receive 3 mg GDC-0032 capsule formulation after 10 hour fasting from food.
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Males or females of non-childbearing potential, between 18 and 55 years of age, inclusive; females will meet the following criteria: they will be non-pregnant, non-lactating, and either postmenopausal for at least 1 year or surgically sterile for at least 90 days. * Body mass ...

Countries:United States
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Frequently asked questions about GDC-0032 Phase III

What is GDC-0032 Phase III used for?

GDC-0032 Phase III is an investigational small molecule being studied in healthy volunteers. It is not approved for any disease and is in clinical development to evaluate its pharmacokinetics, including the effects of particle size, formulation, and food on how the drug is processed in the body.

Who makes GDC-0032 Phase III?

GDC-0032 Phase III is being developed by Roche Holding AG, which trades under the ticker RHHBY. The company is conducting clinical research on this investigational small molecule in healthy volunteer studies.

What phase is GDC-0032 Phase III in?

GDC-0032 Phase III is in Phase 1 clinical development. It is an investigational drug, not yet approved, and is being studied in a completed Phase 1 trial involving healthy volunteers to assess its pharmacokinetic properties.

What clinical trials is GDC-0032 Phase III in?

GDC-0032 Phase III has one completed clinical trial, NCT01980953, titled 'A Study to Evaluate the Effect of Particle Size, Formulation and Food on the Pharmacokinetics of GDC-0032 in Healthy Volunteers.' This Phase 1 study enrolled 76 participants in the United States.

Is GDC-0032 Phase III the same as GDC-0032?

GDC-0032 Phase III is a designation for the drug GDC-0032, which is being studied in a Phase 1 trial. The name includes 'Phase III' but the current clinical development stage is Phase 1, as indicated by the completed trial NCT01980953.