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REGN7999

Phase 2

Non-Transfusion Dependent Beta-Thalassemia (NTDT) | Small molecule | Hematology |Regeneron Pharmaceuticals, Inc.|Last Updated: Jul 1, 2026

Target and mechanism

Molecular targetTMPRSS6
Target classProtein
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment19

FDA Designations

No designations recorded

Clinical trial landscape

REGN7999 · 2 trials · 2 indications

Phase 2 1Phase 1 1
NCT06421636A Study to Test the Safety, Tolerability, and Efficacy of an Antibody, REGN7999, Injected Under the Skin for the Treatment of Iron Overload in Adult Participants With Non-Transfusion Dependent β-thalassemia, Using MRI Scans to Measure Iron Levels in the BodyNon-Transfusion Dependent Beta-Thalassemia (NTDT)
ACTIVE NOT_RECRUITING19 Analytics
PHASE2ACTIVE NOT_RECRUITING
A Study to Test the Safety, Tolerability, and Efficacy of an Antibody, REGN7999, Injected Under the Skin for the Treatment of Iron Overload in Adult Participants With Non-Transfusion Dependent β-thalassemia, Using MRI Scans to Measure Iron Levels in the Body
Non-Transfusion Dependent Beta-Thalassemia (NTDT)Unlock trial analytics

Study Endpoints

Primary Endpoints

Change from baseline in Liver Iron Concentration (LIC) by R2* Magnetic Resonance Imaging (MRI)
At week 24
Incidence of Treatment-Emergent Adverse Events (TEAEs)
Up to week 72
Severity of TEAEs
Up to week 72
Incidence and severity of treatment emergent adverse events (TEAEs) in participants treated with REGN7999 or placebo
Through the end of study visit, week 20

IV cohorts 1 to 4 SC cohorts 1 and 2

Incidence and severity of TEAEs in participants treated with REGN7999 or placebo
Through the end of study visit, week 26

IV cohort 5 and SC cohort 3

Secondary Endpoints

Achievement of ≥20% reduction from baseline in LIC by R2* MRI
Through week 52
Change from baseline in hemoglobin
To week 24
Change from baseline in LIC by R2* MRI
At week 52
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part A High DoseEXPERIMENTALRandomized 2:2:1
Part A Low DoseEXPERIMENTALRandomized 2:2:1
Part A PlaceboPLACEBO_COMPARATORRandomized 2:2:1
Part B High DoseEXPERIMENTALRandomized 2:2:1
Part B Low DoseEXPERIMENTALRandomized 2:2:1
Part B PlaceboPLACEBO_COMPARATORRandomized 2:2:1
IV Cohort 1EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
IV Cohort 2EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
IV Cohort 3EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
IV Cohort 4EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
IV Cohort 5EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
SC Cohort 1EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
SC Cohort 2EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1
SC Cohort 3EXPERIMENTALSingle dose REGN7999 or Placebo; randomized 3:1

Interventions

NameTypeDescription
REGN7999DRUGAdministered subcutaneous (SC)
PlaceboDRUGAdministered SC
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersNo
Study Sites26

Key Inclusion Criteria: 1. Clinical diagnosis of NTDT as described in the protocol 2. IOL, defined as LIC ≥ 5 mg Fe/g DW as measured by R2\* MRI at screening 3. Serum ferritin ≥ 300 ng/mL as described in the protocol Key Exclusion Criteria: 1. Hemoglobin ≤ 8 g/dL at screening 2. Any RBC transfusi...

Countries:United StatesGeorgiaGreeceIndiaItalyMalaysiaThailandTurkey (Türkiye)United KingdomBelgium
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Recent Changes (Last 90 Days)

HIGHJul 2, 2026NCT06421636Status: RECRUITING → ACTIVE_NOT_RECRUITING
HIGHJul 2, 2026NCT06421636Status: RECRUITING → ACTIVE_NOT_RECRUITING
HIGHJul 2, 2026NCT06421636Status: RECRUITING → ACTIVE_NOT_RECRUITING
HIGHJul 2, 2026NCT06421636Status: RECRUITING → ACTIVE_NOT_RECRUITING

Frequently asked questions about REGN7999

What is REGN7999 used for?

REGN7999 is an investigational small molecule being developed by Regeneron Pharmaceuticals for the treatment of iron overload in adult patients with Non-Transfusion Dependent Beta-Thalassemia (NTDT). It is also being studied in healthy participants to assess its safety and how it works in the body.

What does REGN7999 target?

REGN7999 targets TMPRSS6, a protein involved in iron regulation. By targeting TMPRSS6, the drug aims to reduce iron overload in patients with Non-Transfusion Dependent Beta-Thalassemia (NTDT). This mechanism is being evaluated in clinical trials to determine its safety and efficacy.

Who makes REGN7999?

REGN7999 is developed by Regeneron Pharmaceuticals, Inc., a biopharmaceutical company traded on NASDAQ under the ticker symbol REGN. The company is conducting clinical trials to evaluate the drug's safety, tolerability, and efficacy in healthy participants and patients with Non-Transfusion Dependent Beta-Thalassemia (NTDT).

What phase is REGN7999 in?

REGN7999 is in Phase 2 clinical development. A Phase 1 trial in healthy participants has been completed, and a Phase 2 study in patients with Non-Transfusion Dependent Beta-Thalassemia (NTDT) is active but not recruiting. The drug is investigational and has not been approved by regulatory authorities.

What clinical trials is REGN7999 in?

REGN7999 has two clinical trials. NCT05481333 is a completed Phase 1 study in healthy participants in Belgium, with 64 enrolled. NCT06421636 is an active Phase 2 study in adults with Non-Transfusion Dependent Beta-Thalassemia (NTDT) across multiple countries, including the US, Greece, India, and Italy, with 19 enrolled.

Is REGN7999 the same as another drug?

REGN7999 is not known to have alternative names. It is a unique investigational small molecule developed by Regeneron Pharmaceuticals. The drug is being studied under its code name REGN7999 in clinical trials for iron overload in Non-Transfusion Dependent Beta-Thalassemia (NTDT).