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REGN4461

Phase 1

Healthy Volunteers | Small molecule | Other |Regeneron Pharmaceuticals, Inc.|Last Updated: Mar 9, 2020

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLED
Total Trials1
Total Enrollment113

FDA Designations

No designations recorded

Clinical trial landscape

REGN4461 · 1 trial · 1 indication

Phase 1 1
NCT03530514A Study to Examine the Safety, Tolerability and Biological Effects of REGN4461 in Healthy VolunteersHealthy Volunteers
COMPLETED113 Analytics
PHASE1COMPLETED
A Study to Examine the Safety, Tolerability and Biological Effects of REGN4461 in Healthy Volunteers
Healthy VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of treatment-emergent adverse events (TEAEs)
Up to week 27

Secondary Endpoints

Concentrations of REGN4461 in serum over time
Up to week 27
Percent change from baseline to week 12 in body weight in overweight or obese participants
Baseline to week 12
Absolute change from baseline to week 12 in body weight in overweight or obese participants
Baseline to week 12
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Part A: Single dose cohort 1EXPERIMENTALCohort 1 will receive a single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 2EXPERIMENTALCohort 2 will receive a sequential ascending single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 3EXPERIMENTALCohort 3 will receive a sequential ascending single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 4EXPERIMENTALCohort 4 will receive a sequential ascending single SC dose of REGN4461 or matching placebo
Part A: Single dose cohort 5EXPERIMENTALCohort 5 will receive a sequential ascending single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 6EXPERIMENTALCohort 6 will receive a sequential ascending single SC dose of REGN4461 or matching placebo
Part A: Single dose cohort 7EXPERIMENTALCohort 7 will receive a sequential ascending single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 8EXPERIMENTALCohort 8 will receive a single IV dose of REGN4461 or matching placebo
Part A: Single dose cohort 9EXPERIMENTALCohort 9 will receive a single IV dose of REGN4461 or matching placebo
Part B: Repeated dose cohort 10EXPERIMENTALCohort 10 will receive repeated IV or SC doses of REGN4461 or matching placebo

Interventions

NameTypeDescription
REGN4461DRUGREGN4461
PlaceboDRUGPlacebo-matching REGN4461
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Key Inclusion Criteria Part A: * Males and females 18 to 50 years of age, inclusive * Body mass index (BMI) from 18.5 to \<30.0 kg/m\^2 * Participant is judged by the investigator to be in good health and free from major comorbidities based on medical history, physical examination, laboratory safe...

Countries:Belgium
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Frequently asked questions about REGN4461

What is Low-Dose REGN4461 used for?

Low-Dose REGN4461 is an investigational drug being studied for generalized lipodystrophy, a rare metabolic condition, and has also been evaluated in healthy volunteers. It is being developed by Regeneron Pharmaceuticals, Inc. (REGN) and is currently in Phase 2 clinical development.

What does Low-Dose REGN4461 target?

Low-Dose REGN4461 is a leptin receptor agonist antibody, meaning it targets and activates the leptin receptor. This mechanism is relevant to its potential use in generalized lipodystrophy, a condition characterized by fat loss and metabolic abnormalities.

Who makes Low-Dose REGN4461?

Low-Dose REGN4461 is being developed by Regeneron Pharmaceuticals, Inc., a biopharmaceutical company traded on the Nasdaq under the ticker symbol REGN. The drug is currently in Phase 2 clinical trials for generalized lipodystrophy.

What phase is Low-Dose REGN4461 in?

Low-Dose REGN4461 is in Phase 2 clinical development for generalized lipodystrophy. It is an investigational drug and has not been approved by regulatory authorities. A Phase 1 study in healthy volunteers has been completed.

What clinical trials is Low-Dose REGN4461 in?

Low-Dose REGN4461 has been studied in two completed trials. NCT03530514 was a Phase 1 study in healthy volunteers with 113 participants in Belgium. NCT04159415 was a Phase 2 study in patients with generalized lipodystrophy, enrolling 16 participants across the United States, Peru, Russia, and Turkey.

Is Low-Dose REGN4461 the same as REGN4461?

Yes, Low-Dose REGN4461 is the same drug as REGN4461. The name 'Low-Dose' refers to the specific dosage being studied, but the active agent is REGN4461, a leptin receptor agonist antibody developed by Regeneron Pharmaceuticals.