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voriconazole

Phase 3

Aspergillosis | Small molecule | Infectious Disease |Pfizer, Inc.|Last Updated: May 5, 2016

Target and mechanism

ModalitySmall molecule

Also known as voriconazole (Vfend)

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLEDDMC
Total Trials2
Total Enrollment507

FDA Designations

No designations recorded

Clinical trial landscape

voriconazole · 9 trials · 9 indications

Phase 3 2Phase 2 4Phase 1 3
NCT00531479Anidulafungin Plus Voriconazole Versus Voriconazole For The Treatment Of Invasive AspergillosisAspergillosis
COMPLETED459 Analytics
NCT00150345Immediate vs. Deferred Empirical Antifungal Treatment With Voriconazole In Neutropenic PatientsPossible Fungal Infection
COMPLETED147 Analytics
PHASE3COMPLETED
Anidulafungin Plus Voriconazole Versus Voriconazole For The Treatment Of Invasive Aspergillosis
AspergillosisUnlock trial analytics
PHASE3COMPLETED
Immediate vs. Deferred Empirical Antifungal Treatment With Voriconazole In Neutropenic Patients
Possible Fungal InfectionUnlock trial analytics

Study Endpoints

Primary Endpoints

All-cause Mortality at Week 6 in Participants With Proven or Probable Invasive Aspergillosis
Day 1 to Day 42 (Week 6)

Number of deaths measured 6 weeks after start of treatment. Time to death defined as date of death minus first treatment date + 1.

Number of Participants With Proven or Probable Invasive Fungal Infections (IFI): Complete Case Analysis
Day 2 through Day 28

Number of participants with proven (deep tissue infection, fungemia, or endemic fungal infections) or probable IFI (at least 1 host criterion \[fever, body temperature \<36 or \>38 degrees Celsius, graft-versus-host disease, use of corticosteroids\]; and 1 microbiological criterion \[fungal or yeasts\]; or clinical criteria \[abnormal site consistent with infection\]) as defined by European Organization for Research and Treatment of Cancer Mycosis Study Group (EORTC/MSG) criteria. Complete case analysis: must be evaluable until Day 28 or had developed a proven or probable IFI by the final visit.

Area Under the Plasma Concentration-time Profile From Time Zero to Twelve Hours at Steady-State (AUC12,ss) Following IV Administration
Day 7 (up to Day 20): predose, 1 hour after the start of infusion, 10-20 minutes after the end of infusion, and 4, 6, 8, and 12 hours after the start of infusion

AUC12,ss was obtained by the Linear/Log trapezoidal method.

Maximum Observed Plasma Concentration at Steady State (Cmax,ss) Following IV Administration
Day 7 (up to Day 20): predose, 1 hour after the start of infusion, 10-20 minutes after the end of infusion, and 4, 6, 8, and 12 hours after the start of infusion
Time to Reach Maximum Observed Plasma Concentration (Tmax) Following IV Administration
Day 7 (up to Day 20): predose, 1 hour after the start of infusion, 10-20 minutes after the end of infusion, and 4, 6, 8, and 12 hours after the start of infusion
Area Under the Plasma Concentration-time Profile From Time Zero to Twelve Hours at Steady-State (AUC12,ss) Following Oral Administration
Day 14 (the 7th day of oral treatment) or later: predose, and 1, 2, 4, 6, 8, and 12 hours after dosing

AUC12,ss was obtained by the Linear/Log trapezoidal method.

Maximum Observed Plasma Concentration at Steady State (Cmax,ss) Following Oral Administration
Day 14 (the 7th day of oral treatment) or later: predose, and 1, 2, 4, 6, 8, and 12 hours after dosing
Time to Reach Maximum Observed Plasma Concentration (Tmax) Following Oral Administration
Day 14 (the 7th day of oral treatment) or later: predose, and 1, 2, 4, 6, 8, and 12 hours after dosing
Number of Participants Assessed Near Distance Visual Acuity Test
Screening, Day 7 (the 7th day of IV treatment), Day 8 (the 1st day of oral treatment), Day 14 (the 7th day of oral treatment), and the 30-day follow-up visit
Number of Participants Assessed Color Vision Test
Screening, Day 7 (the 7th day of IV treatment), Day 8 (the 1st day of oral treatment), Day 14 (the 7th day of oral treatment), and the 30-day follow-up visit
Number of Participants Assessed Visual Questionnaire
Screening, Day 7 (the 7th day of IV treatment), Day 8 (the 1st day of oral treatment), Day 14 (the 7th day of oral treatment), and the 30-day follow-up visit
Area Under the Curve Over Dosing Interval at Steady State (AUC12,ss) Following IV Administration
Day 7 (up to Day 20 or more) at predose, 60 and 138 minutes, 4, 6, 8 and 12 hours postdose

AUC12,ss = Area under the plasma concentration-time profile from time zero (predose) to twelve hours at steady-state. AUC12,ss was obtained by the Linear/Log trapezoidal method.

Peak Plasma Concentration at Steady State (Cmax,ss) Following IV Administration
Day 7 (up to Day 20 or more) at predose, 60 and 138 minutes, 4, 6, 8 and 12 hours postdose
Time to Reach Cmax (Tmax) Following IV Administration
Day 7 (up to Day 20 or more) at predose, 60 and 138 minutes, 4, 6, 8 and 12 hours postdose
AUC12,ss Following Oral Administration
Day 7 (or later) predose, 1, 2, 4, 6, 8 and 12 hours postdose

AUC12,ss = Area under the plasma concentration-time profile from time zero (predose) to twelve hours at steady-state. AUC12,ss was obtained by the Linear/Log trapezoidal method.

Cmax,ss Following Oral Administration
Day 7 (or later) predose, 1, 2, 4, 6, 8 and 12 hours postdose
Tmax Following Oral Administration
Day 7 (or later) predose, 1, 2, 4, 6, 8 and 12 hours postdose
Number of Subjects With Successful Global Outcome at 6 Months: Chronic Bronchopulmonary Aspergillosis
at 6 months of treatment

Successful global outcome: composite assessment of radiological and mycological responses; defined as complete or partial radiological response and mycological eradication (absence of aspergillus); no success=criteria not met. Assessment was determined by the Data Review Committee (DRC). Complete response: resolution of radiographic and or bronchoscopic abnormalities attributable to aspergillosis present at baseline; partial response: reduction in diameter ≥ 50 percent on chest tomodensitometry (TDM) or regressed lesion on endoscopy witnessed by 2 different operators without any new lesion.

The pharmacokinetics of voriconazole following an intravenous to oral switch regimen in healthy adults
14 days
Assess brain levels of voriconazole in the brain using a non-evasive technique of MRS
The primary objective was to investigate the pharmacokinetics of voriconazole following intravenous (iv) to oral administration in immunocompromised children aged 2 to <12years.

Secondary Endpoints

Global Response at Week 6
Baseline, Day 42 (Week 6)
All-cause Mortality at Week 6 in Participants With Possible, Probable, or Proven Invasive Aspergillosis (IA)
Day 1 to Day 42 (Week 6)
All-cause Mortality at Week 12 in Participants With Probable or Proven Invasive Aspergillosis (IA)
Day 1 to Day 84 (Week 12)
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
VoriconazoleACTIVE_COMPARATORVoriconazole monotherapy
Voriconazole and AnidulafunginEXPERIMENTALCombination therapy with voriconazole and anidulafungin
Early treatmentEXPERIMENTALVoriconazole starts within 18 hours of onset of fever intravenously with a loading dose of 6 mg/kg q12h for the first two doses followed by 4 mg/kg q12h (maintenance dose). Switched to oral treatment (200 mg BID) is possible after at least four days. Treatment will be ended if the patient is afebrile (\< 38.0 °C) for 7 days with neutrophil counts \< 500/µL, or if the patient is afebrile (\< 38.0 °C) for 2 days with neutrophil counts \> 500/µL.
Deferred treatmentOTHERTreatment with voriconazole (for dosage see "early treatment arm") is initiated only if a patient is persistently febrile on day 5 after the onset of fever despite antibiotic treatment.
1.0EXPERIMENTALImmunocompromised children aged 2 to \<15 and 12 to \<15 years weighing \<50 kg who are at high risk for systemic fungal infection.
2.0EXPERIMENTALImmunocompromised children aged 12 to \<15 years weighing more than 50 kg who are at high risk for systemic fungal infection.
Children aged 2 to <12 yearsEXPERIMENTALImmunocompromised children aged 2 to \<12 years who are at high risk for systemic fungal infection.
1EXPERIMENTAL -

Interventions

NameTypeDescription
voriconazoleDRUGFirst week: Voriconazole 6 mg/kg IV bid for the first 24 hours, followed by 4 mg/kg IV BID plus anidulafungin placebo IV qd. Second week: Voriconazole 4 mg/kg IV bid or 300 mg PO bid plus anidulafungin placebo IV qd. Third and fourth weeks: Voriconazole 4 mg/kg IV bid OR 300 mg PO bid plus anidulafungin placebo IV qd, OR Voriconazole 4 mg/kg IV bid or 300 mg PO bid monotherapy. Fifth and sixth weeks: Voriconazole 4 mg/kg IV bid or 300 mg PO bid monotherapy.
anidulafunginDRUGFirst week: Voriconazole 6 mg/kg IV bid for the first 24 hours, followed by 4 mg/kg IV bid plus anidulafungin 200 mg IV on day 1, followed by 100 mg IV qd thereafter. Second week: Voriconazole 4 mg/kg IV bid or 300 mg PO bid plus anidulafungin 100 mg IV qd. Third and fourth weeks: Voriconazole 4 mg/kg IV bid OR 300 mg PO bid plus anidulafungin 100 mg IV qd, OR Voriconazole 4 mg/kg IV bid or 300 mg PO bid monotherapy. Fifth and sixth weeks: Voriconazole 4 mg/kg IV bid or 300 mg PO bid monotherapy.
voriconazole (Vfend)DRUGvoriconazole, early treatment
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Eligibility Criteria

Age Range16 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites107

Inclusion Criteria: * Immunocompromised state due to either 1. receipt of hematopoeitic stem cell transplantation or 2. hematologic malignancy; * Diagnosis of possible, probable, or proven invasive aspergillosis. Exclusion Criteria: * Patients with aspergilloma or chronic aspergillosis * Receipt ...

Countries:United StatesAustraliaBelgiumBrazilCanadaCzechiaFranceGermanyGreeceIndiaItalyNetherlandsPeruPolandPortugalRussiaSingaporeSouth KoreaSpainSwitzerlandTaiwanThailandTurkey (Türkiye)United KingdomJapan
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