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Vupanorsen

Phase 2

Dyslipidemias | Small molecule | Metabolic |Pfizer, Inc.|Last Updated: Oct 4, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment286
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04516291A Dose-Ranging Study With Vupanorsen (TRANSLATE-TIMI 70)PHASE2 COMPLETED 286Sep 28, 2020Dec 6, 2021Oct 4, 2022114 United States, Canada +1
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Study Endpoints
Primary Endpoints
Percent Change From Baseline in Non-High-Density Lipoprotein-Cholesterol (Non-HDL-C) at Week 24
Baseline, Week 24

Fasting was required at least 10 hours before blood sample collection. Baseline was calculated using the average of all values obtained at Screening and on Day 1 prior to dosing.

Secondary Endpoints
Percent Change From Baseline in Triglyceride (TG), Apolipoprotein B (ApoB), Low-Density Lipoprotein-Cholesterol (LDL-C), and Non-HDL-C at Week 16
Baseline, Week 16
Percent Change From Baseline in TG, ApoB, and LDL-C at Week 24
Baseline, Week 24
Percent Change From Baseline in Angiopoietin-like Protein 3 (ANGPTL3) at Week 16
Baseline, Week 16
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
PlaceboPLACEBO_COMPARATORNo drug
Vupanorsen 80 mg every 4 weeksEXPERIMENTAL80 milligrams (mg) given subcutaneously every 4 weeks.
Vupanorsen 60 mg every 2 weeksEXPERIMENTAL60 mg given subcutaneously every 2 weeks.
Vupanorsen 120 mg every 4 weeksEXPERIMENTAL120 mg given subcutaneously every 4 weeks.
Vupanorsen 80 mg every 2 weeksEXPERIMENTAL80 mg given subcutaneously every 2 weeks.
Vupanorsen 160 mg every 4 weeksEXPERIMENTAL160 mg given subcutaneously every 4 weeks.
Vupanorsen 120 mg every 2 weeksEXPERIMENTAL120 mg given subcutaneously every 2 weeks.
Vupanorsen 160 mg every 2 weeksEXPERIMENTAL160 mg given subcutaneously every 2 weeks.
Interventions
NameTypeDescription
VupanorsenDRUGVupanorsen and placebo will be provided as prefilled syringes packaged and dispensed in cartons with tamper-evident seals. Only single-use syringes will be used.
PlaceboDRUGVupanorsen and placebo will be provided as prefilled syringes packaged and dispensed in cartons with tamper-evident seals. Only single-use syringes will be used.
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Eligibility Criteria
Age Range40 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites114

Inclusion Criteria: 1. Male or female participants aged ≥40 years at Screening. 2. Fasting non-HDL-C at Screening ≥100 mg/dL. 3. Fasting TG at Screening of 150 to 500 mg/dL, inclusive, which may be repeated once if deemed necessary. 4. Participants must be on a stable dose of a statin for at least ...

Countries:United StatesCanadaPoland
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