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PF-04937319 once-daily

Phase 1

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Pfizer, Inc.|Last Updated: Sep 27, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment33
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01933672Study Of Two Dosing Regimens Of PF-04937319 Compared To An Approved Agent (Sitagliptin) In Patients With Type 2 DiabetesPHASE1 COMPLETED 33Oct 1, 2013Mar 1, 2014Sep 27, 20168 United States
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Study Endpoints
Primary Endpoints
Change From Baseline in Weighted Mean Daily Glucose (WMDG) at Day 14
Prior to morning dose (Hour 0) and at 1.5, 3, 5, 6.5, 8, 11, 12.5, 14, 16, 20, and 24 hours post morning dose on Days 0 (baseline) and Day 14

Plasma glucose concentration was determined predose (Hour 0) and at 1.5, 3, 5, 6.5, 8, 11, 12.5, 14, 16, 20, and 24 hours postdose on Days 0 (baseline) and 14. WMDG was calculated as the area under the curve (AUC) of the 12-point plasma glucose concentration-time profile divided by 24 hours.

Secondary Endpoints
Change From Baseline in Fasting Plasma Glucose (FPG) at Day 14
Day 14
Change From Baseline in Pre-meal C-Peptide on Day 14
Day 14
Change From Baseline in Pre-meal Insulin on Day 14
Day 14
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
PF-04937319 once-dailyEXPERIMENTAL -
PF-04937319 split-doseEXPERIMENTAL -
Sitagliptin once-dailyACTIVE_COMPARATOR -
Interventions
NameTypeDescription
PF-04937319 once-dailyDRUGTablets, 300 mg once-daily with breakfast, 14-days
PF-04937319 split-doseDRUGtablets, 150 mg with breakfast plus 100 mg with lunch, 14-days
Sitagliptin once-dailyDRUGtablets, 100 mg once-daily with breakfast, 14-days
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites8

Inclusion Criteria: * Patients with type 2 diabetes, on background metformin therapy either alone or with 1 other oral anti-diabetic agent (excluding Actos) Exclusion Criteria: * Patients with cardiovascular event within 6-months of screening * Patients with diabetic complications * Female subjec...

Countries:United States
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