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PF-04937319 IR MST

Phase 1

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Pfizer, Inc.|Last Updated: Mar 4, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment39
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02206607Study To Compare Single Dose Of Three Modified Release Formulations Of PF-04937319 With Immediate Release Material-Sparing-Tablet (IR MST) Formulation Previously Studied In Adults With Type 2 Diabetes Mellitus.PHASE1 COMPLETED 39Sep 1, 2014Jan 1, 2015Mar 4, 20162 United States
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Study Endpoints
Primary Endpoints
Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUCinf]
0 (pre-dose) and 1, 2, 3, 4, 5, 6, 7, 8, 11, 12.5, 14, 16, 20, 24, 36, 48, and 72 hours post-dose

AUCinf is the area under the plasma concentration versus time curve (AUC) from time zero (pre-dose) to extrapolated infinite time.

Change From Reference in Weighted-Mean-Daily-Glucose (WMDG) on Day 1
0 (pre-dose) and 1, 2, 3, 4, 5, 6, 7, 8, 11, 12.5, 14, 16, 20, and 24 hours post-dose

MWG was calculated as the area under the curve (AUC) for the full 24 hours expressed.

Secondary Endpoints
Maximum Observed PF-04937319 Plasma Concentration (Cmax)
0 (pre-dose) and 1, 2, 3, 4, 5, 6, 7, 8, 11, 12.5, 14, 16, 20, 24, 36, 48, and 72 hours post-dose
PF-04937319 Plasma Concentration at 5 Hours After Morning Dose (C5)
0 (pre-dose) and 1, 2, 3, 4, 5, 6, 7, 8, 11, 12.5, 14, 16, 20, 24, 36, 48, and 72 hours post-dose
PF-04937319 Plasma Concentration at 16 Hours After Morning Dose (C16)
0 (pre-dose) and 1, 2, 3, 4, 5, 6, 7, 8, 11, 12.5, 14, 16, 20, 24, 36, 48, and 72 hours post-dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
PF-04937319 IR MSTEXPERIMENTALReference formulation
PF-04937319 MR 1EXPERIMENTALTest MR #1
PF-04937319 MR 2EXPERIMENTALTest MR #2
PF-04937319 MR 3EXPERIMENTALTest MR #3
Interventions
NameTypeDescription
PF-04937319 IR MSTDRUGImmediate release material sparing tablet (IR MST) administered as 150 mg with morning meal and 100 mg with lunch
PF-04937319 MR 1DRUGModified release formulation #1 administered with the morning meal at a dose predicted to yield exposure (AUC24) equivalent to 300 mg IR MST
PF-04937319 MR 2DRUGModified release formulation #2 administered with the morning meal at a dose predicted to yield exposure (AUC24) equivalent to 300 mg IR MST
PF-04937319 MR 3DRUGModified release formulation #3 administered with the morning meal at a dose predicted to yield exposure (AUC24) equivalent to 300 mg IR MST
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion Criteria: * Adults with type 2 diabetes, on stable background metformin therapy either alone or in combination with another oral anti-diabetic agent (OAD) excluding thiazolidinediones (TZDs) Exclusion Criteria: * Patients with cardiovascular event within 6 months of screening * Patients...

Countries:United States
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