Recent Updates
Recently added Catalysts

PF 06252616

Phase 1

LGMD2I | Small molecule | Other |Pfizer, Inc.|Last Updated: Oct 19, 2020

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

ACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment19

FDA Designations

No designations recorded

Clinical trial landscape

PF 06252616 · 1 trial · 1 indication

Phase 1 1
NCT02841267A Trial of PF-06252616 in Ambulatory Participants With LGMD2ILGMD2I
COMPLETED19 Analytics
PHASE1COMPLETED
A Trial of PF-06252616 in Ambulatory Participants With LGMD2I
LGMD2IUnlock trial analytics

Study Endpoints

Primary Endpoints

Incidence of Dose Limiting or Intolerability Treatment Related Adverse Events
Baseline through 64 weeks

Adverse events include subject-reported symptoms as well as clinically-significant changes in laboratory testing, vital signs, and suicide screening (based on the Columbia Suicide Severity Rating Scale).

Secondary Endpoints

Maximum Observed Serum Concentration at Steady State (Cmax, ss) of GDF-8
Day 337 and Day 393 for Cohort 1; Day 113 and 169 for Cohorts 2 and 3
Minimum Observed Serum Trough Concentration at Steady State (Ctrough,ss) of GDF-8
Day 337 and Day 393 for Cohort 1; Day 113 and 169 for Cohorts 2 and 3
Maximum Observed Serum Concentration (Cmax) of PF-06252616
Day 113 and Day 169
Unlock Study Endpoints

Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Low Dose, Cohort 1ACTIVE_COMPARATOR4 subjects will be enrolled in cohort 1 and will receive an initial dose of 5mg/kg PF 06252616 IV every 4 weeks. Following 32 weeks of treatment and a safety review, if no stopping rules have been met, subjects will be receive an additional 32 weeks of treatment with 40 mg/kg PF 06252616 IV every 4 weeks.
Middle dose, Cohort 2ACTIVE_COMPARATOR8 subjects will be enrolled in cohort 2 and receive 20 mg/kg of PF 06252616 IV every 4 weeks for 32 weeks.
High dose, Cohort 3ACTIVE_COMPARATOR8 subjects will be enrolled in cohort 3 and receive 40 mg/kg of PF06252616 IV every 4 weeks for 32 weeks.

Interventions

NameTypeDescription
PF 06252616DRUG -
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 99 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. Male and female patients age ≥ 18 2. Diagnosis of LGMD2I as defined by clinical presentation consistent with LGMD2I and FKRP gene testing showing biallelic alterations known or likely to be pathogenic. Diagnosis must be confirmed in subject's medical history and by genetic te...

Countries:United States
Unlock Eligibility Criteria

Frequently asked questions about PF 06252616

What is PF 06252616?

PF 06252616 is an investigational small molecule being developed by Pfizer, Inc. (PFE). It has been studied in Phase 1 clinical trials for the treatment of LGMD2I, a form of limb-girdle muscular dystrophy, as well as in healthy volunteers. The drug is not approved and remains in clinical development.

What is PF 06252616 used for?

PF 06252616 is being investigated for use in LGMD2I, a genetic muscle disorder, and has also been studied in healthy subjects to evaluate its safety and tolerability. It is an investigational drug and has not been approved for any indication.

Who makes PF 06252616?

PF 06252616 is developed by Pfizer, Inc., a biopharmaceutical company listed on the New York Stock Exchange under the ticker symbol PFE. The company has conducted clinical trials to evaluate the drug's safety and tolerability.

What phase is PF 06252616 in?

PF 06252616 is in Phase 1 clinical development. Two Phase 1 trials have been completed, one in healthy subjects and one in participants with LGMD2I. The drug is investigational and has not received FDA approval.

What clinical trials is PF 06252616 in?

PF 06252616 has been studied in two completed Phase 1 trials: NCT01616277, which evaluated safety and tolerability in healthy subjects, and NCT02841267, which assessed the drug in ambulatory participants with LGMD2I. Both trials were conducted in the United States.

Is PF 06252616 the same as PF-06252616?

Yes, PF 06252616 and PF-06252616 refer to the same investigational drug developed by Pfizer. The hyphenated version is the standard naming format used in clinical trial registries and scientific literature.