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Glasdegib Therapeutic Exposure

Phase 1

Healthy Volunteers | Small molecule | Other |Pfizer, Inc.|Last Updated: Sep 6, 2019

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials1
Total Enrollment36
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03162900A Phase 1 Study To Evaluate The Effect Of Glasdegib On The Cardiac Repolarization In Healthy SubjectsPHASE1 COMPLETED 36Jun 9, 2017Oct 16, 2017Sep 6, 20191 Belgium
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Study Endpoints
Primary Endpoints
QTcF interval
120 hours per period

Post-dose placebo corrected QTcF intervals from ECG traces following glasdegib dosing.

Secondary Endpoints
QTcF interval (Moxifloxacin)
120 hours
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Glasdegib QT Therapeutic ExposureEXPERIMENTALRandomized sequence of Glasdegib clinical exposure, Placebo and moxifloxacin active control administration. This treatment will be in four separate sequences with four periods per sequence. Each period will be separated by a washout of atleast 6 days.
Glasdegib QT Supra-therapeutic ExposureEXPERIMENTALRandomized sequence of glasdegib supra-therapeutic exposure, Placebo and moxifloxacin active control administration. This treatment will be in four separate sequences with four periods per sequence. Each period will be separated by a washout of atleast 6 days.
Interventions
NameTypeDescription
Glasdegib Therapeutic ExposureDRUGSubjects Receive a single 150 mg dose of Glasdegib followed by ECG and PK assessments.
Glasdegib Supra-therapeutic ExposureDRUGSubjects receive a single 300 mg dose of glasdegib followed by ECG and PK assessments.
Positive Control (Moxifloxacin)DRUGSubjects will receive a single 400 mg dose of moxifloxacin followed by ECG and PK assessments.
Placebo ControlOTHERSubjects will receive placebo dose followed by ECG and PK assessments.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * 1\. Healthy male and/or female subjects of non child bearing potential who, at the time of screening, are between the ages of 18 and 55 years, inclusive. Healthy is defined as no clinically relevant abnormalities identified by a detailed medical history, full physical examinat...

Countries:Belgium
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