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CE/BZA

Phase 1

Healthy | Small molecule | Other |Pfizer, Inc.|Last Updated: Mar 25, 2015

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment24

FDA Designations

No designations recorded

Clinical trial landscape

CE/BZA · 1 trial · 1 indication

Phase 1 1
NCT02100553Study Evaluating Effects of Multiple-Dose Administration of Itraconazole on the Single Dose Pharmacokinetics of Conjugated Estrogens/Bazedoxifene in Non-Obese and Obese Postmenopausal WomenHealthy
COMPLETED24 Analytics
PHASE1COMPLETED
Study Evaluating Effects of Multiple-Dose Administration of Itraconazole on the Single Dose Pharmacokinetics of Conjugated Estrogens/Bazedoxifene in Non-Obese and Obese Postmenopausal Women
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Study Endpoints

Primary Endpoints

Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUC (0 - inf)] for BZA, total estrone adjusted for baseline and total equilin.
up to 96 hours

AUC (0 - inf)= Area under the plasma concentration versus time curve (AUC) from time zero (pre-dose) to extrapolated infinite time (0 - inf). It is obtained from AUC (0 - t) plus AUC (t - inf).

Maximum Observed Plasma Concentration (Cmax) for BZA, total estrone adjusted for baseline and total equilin.
up to 96 hours

Secondary Endpoints

Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUC (0 - inf)] for unconjugated estrone, unconjugated estrone adjusted for baseline, total estrone, and unconjugated equilin.
up to 96 hours
Maximum Observed Plasma Concentration (Cmax) for unconjugated estrone, unconjugated estrone adjusted for baseline, total estrone, and unconjugated equilin.
up to 96 hours
Apparent Oral Clearance (CL/F) for all analytes.
up to 96 hours
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Non-ObeseOTHERBMI \<30 kg/m\^2
ObeseOTHERBMI \>= 30 kg/m\^2

Interventions

NameTypeDescription
CE/BZADRUGCE 0.45mg/BZA 20mg tablets, single dose
ItraconazoleDRUGTwo 100 mg capsules, once daily for 7 days
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Eligibility Criteria

Age Range40 Years to 64 Years
SexFEMALE
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Generally healthy postmenopausal women, aged 40-64. Intact Uterus Exclusion Criteria: * The use of oral, vaginal, or transdermal estrogen, androgen or progestin-containing medications within 30 days before study drug administration.

Countries:United States
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Frequently asked questions about CE/BZA

What is CE/BZA used for?

CE/BZA is a small molecule drug being developed by Pfizer, Inc. It is being studied in healthy postmenopausal women. The drug is currently in Phase 1 clinical development, and it is investigational, meaning it has not been approved for any use.

Who makes CE/BZA?

CE/BZA is being developed by Pfizer, Inc., which is publicly traded under the ticker symbol PFE. The drug is currently in Phase 1 clinical development.

What phase is CE/BZA in?

CE/BZA is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed.

What clinical trials is CE/BZA in?

CE/BZA has one completed Phase 1 clinical trial, NCT02100553. This study evaluated the effects of multiple-dose administration of itraconazole on the single-dose pharmacokinetics of conjugated estrogens/bazedoxifene in non-obese and obese postmenopausal women.

Is CE/BZA the same as conjugated estrogens/bazedoxifene?

CE/BZA is a name for the combination of conjugated estrogens and bazedoxifene. The clinical trial NCT02100553 refers to the drug as conjugated estrogens/bazedoxifene, indicating that CE/BZA is an abbreviation for this combination.