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ARRY-142886, MEK inhibitor

Phase 1

Advanced Cancer | Small molecule | Oncology |Pfizer, Inc.|Last Updated: Oct 14, 2020

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment57

FDA Designations

No designations recorded

Clinical trial landscape

ARRY-142886, MEK inhibitor · 1 trial · 1 indication

Phase 1 1
NCT00085787A Study of ARRY-142886 in Patients With Advanced CancerAdvanced Cancer
COMPLETED57 Analytics
PHASE1COMPLETED
A Study of ARRY-142886 in Patients With Advanced Cancer
Advanced CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Characterize the safety profile of the study drug in terms of adverse events, clinical laboratory tests, vital signs and electrocardiograms.
Part 1
Establish the maximum tolerated dose (MTD) of study drug.
Part 1
Assess the biological activity of the study drug in tumors in terms of inhibition of extracellular signal-regulated kinase (ERK) phosphorylation.
Part 2

Secondary Endpoints

Characterize the pharmacokinetics (PK) of the study drug in terms of plasma concentrations.
Part 1 and Part 2
Characterize the pharmacodynamic (PD) activity of the study drug on biomarkers.
Part 1 and Part 2
Assess the efficacy of the study drug in terms of tumor dimension assessment.
Part 1 and Part 2
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ARRY-142886EXPERIMENTAL -

Interventions

NameTypeDescription
ARRY-142886, MEK inhibitor; oralDRUGPart 1: single dose and multiple dose, escalating; Part 2: multiple dose, single schedule
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites3

Key Inclusion Criteria (Part 2): * Histopathologically or cytologically confirmed solid tumor that is refractory to standard therapies, or for which no standard therapies exist, or for which the Investigator feels no other active therapy is required for the duration of the study. * Eastern Cooperat...

Countries:United States
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Competitive Landscape -Cancer 5 trials (matched to "Advanced Cancer")

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Frequently asked questions about ARRY-142886, MEK inhibitor

What is ARRY-142886 used for?

ARRY-142886 is an investigational oral small molecule being studied in advanced cancer. It was evaluated in a Phase 1 trial in patients with advanced cancer. It is not an approved therapy and remains in clinical development.

What does ARRY-142886 target?

ARRY-142886 is a MEK inhibitor. It targets MEK, a kinase in the MAPK signaling pathway. By inhibiting MEK, the drug aims to block signals that drive cancer cell growth. This mechanism is being explored in advanced cancer.

Who is developing ARRY-142886?

Pfizer, Inc. (ticker: PFE) is the developer of ARRY-142886. The company is responsible for its clinical development in advanced cancer.

What phase is ARRY-142886 in?

ARRY-142886 is in Phase 1 clinical development. It is investigational and has not been approved by the FDA for any indication. The Phase 1 program has been completed.

What clinical trials is ARRY-142886 in?

ARRY-142886 was studied in a Phase 1 trial, NCT00085787, titled "A Study of ARRY-142886 in Patients With Advanced Cancer." The trial enrolled 57 patients in the United States and is completed. No active trials are ongoing.

Is ARRY-142886 the same as MEK inhibitor?

ARRY-142886 is also known as a MEK inhibitor, which describes its drug class. It is an oral small molecule. The names ARRY-142886 and MEK inhibitor refer to the same investigational agent.