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ARRY-142886, MEK inhibitor

Phase 1

Advanced Cancer | Small molecule | Oncology |Pfizer, Inc.|Last Updated: Oct 14, 2020

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment57

FDA Designations

No designations recorded

Clinical trial landscape

ARRY-142886, MEK inhibitor · 1 trial · 1 indication

Phase 1 1
NCT00085787A Study of ARRY-142886 in Patients With Advanced CancerAdvanced Cancer
COMPLETED57 Analytics
PHASE1COMPLETED
A Study of ARRY-142886 in Patients With Advanced Cancer
Advanced CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Characterize the safety profile of the study drug in terms of adverse events, clinical laboratory tests, vital signs and electrocardiograms.
Part 1
Establish the maximum tolerated dose (MTD) of study drug.
Part 1
Assess the biological activity of the study drug in tumors in terms of inhibition of extracellular signal-regulated kinase (ERK) phosphorylation.
Part 2

Secondary Endpoints

Characterize the pharmacokinetics (PK) of the study drug in terms of plasma concentrations.
Part 1 and Part 2
Characterize the pharmacodynamic (PD) activity of the study drug on biomarkers.
Part 1 and Part 2
Assess the efficacy of the study drug in terms of tumor dimension assessment.
Part 1 and Part 2
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ARRY-142886EXPERIMENTAL -

Interventions

NameTypeDescription
ARRY-142886, MEK inhibitor; oralDRUGPart 1: single dose and multiple dose, escalating; Part 2: multiple dose, single schedule
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites3

Key Inclusion Criteria (Part 2): * Histopathologically or cytologically confirmed solid tumor that is refractory to standard therapies, or for which no standard therapies exist, or for which the Investigator feels no other active therapy is required for the duration of the study. * Eastern Cooperat...

Countries:United States
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Competitive Landscape -Cancer 5 trials (matched to "Advanced Cancer")

Frequently asked questions about ARRY-142886, MEK inhibitor

What is ARRY-142886 used for?

ARRY-142886 is an investigational small molecule MEK inhibitor being studied for the treatment of advanced cancer. It is currently in Phase 1 clinical development and has not been approved by the FDA. The drug is being evaluated in patients with advanced cancer to assess its safety and potential efficacy.

What does ARRY-142886 target?

ARRY-142886 targets MEK, a protein kinase involved in cell signaling pathways that regulate cell growth and proliferation. By inhibiting MEK, the drug aims to disrupt cancer cell growth. This mechanism is being explored in the treatment of advanced cancer.

Who makes ARRY-142886?

ARRY-142886 is being developed by Pfizer, Inc., a biopharmaceutical company listed on the New York Stock Exchange under the ticker symbol PFE. The drug is currently in Phase 1 clinical trials for advanced cancer.

What phase is ARRY-142886 in?

ARRY-142886 is in Phase 1 clinical development. It is an investigational drug and has not been approved by the FDA. The Phase 1 trial has been completed, and the drug remains under investigation for the treatment of advanced cancer.

What clinical trials is ARRY-142886 in?

ARRY-142886 has one completed Phase 1 clinical trial, identified as NCT00085787, titled "A Study of ARRY-142886 in Patients With Advanced Cancer." The trial enrolled 57 participants in the United States and was an uncontrolled, open-label study.