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Alfimeprase

Phase 3

Arterial Occlusive Diseases | Small molecule | Cardiovascular |Oruka Therapeutics, Inc.|Last Updated: Feb 3, 2010

Development status

Highest phase Phase 3
Registered trials 7 across 1 sponsor since Nov 2003

Target and mechanism

Molecular targetFGA, FGB, FGG
Target classHydrolytic Enzyme
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindUNCONTROLLEDDMC
Total Trials2
Total Enrollment400

FDA Designations

No designations recorded

Clinical trial landscape

Alfimeprase · 5 trials · 6 indications

Phase 3 3Phase 2 2
NCT00322270Safety and Efficacy Study of Alfimeprase in Subjects With Occluded CathetersThrombosis
COMPLETED- Analytics
NCT00346424Safety and Efficacy Study of Alfimeprase in Subjects With Occluded Central CathetersThrombosis
COMPLETED300 Analytics
NCT00115999Study of Alfimeprase to Rapidly Dissolve Blood Clots in the Leg and Help Prevent the Need for Surgery on Leg ArteriesArterial Occlusive Diseases
COMPLETED300 Analytics
PHASE3COMPLETED
Safety and Efficacy Study of Alfimeprase in Subjects With Occluded Catheters
ThrombosisUnlock trial analytics
PHASE3COMPLETED
Safety and Efficacy Study of Alfimeprase in Subjects With Occluded Central Catheters
ThrombosisUnlock trial analytics
PHASE3COMPLETED
Study of Alfimeprase to Rapidly Dissolve Blood Clots in the Leg and Help Prevent the Need for Surgery on Leg Arteries
Arterial Occlusive DiseasesUnlock trial analytics

Study Endpoints

Primary Endpoints

Safety and efficacy
up to120 minutes post study drug dosing
Catheter function restoration at fifteen minutes after initial instillation of study drug.
15 minutes
30 day open vascular surgery free rate

Secondary Endpoints

Adverse events, serious adverse events and bleeding events
24 hours post dosing
Adverse events up to day 30 visit(day 28-45) after instillation of study drug
approximately 28-45 days post dosing
Catheter function restoration at 30 minutes after initial instillation of study drug.
30 minutes
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Interventions

NameTypeDescription
AlfimepraseDRUGsingle-dose of alfimeprase, 10 mg.administered intracatheter to an occluded CVAD
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites18

Inclusion Criteria: * Must give written informed consent * Ages 18 or older * Unable to withdraw at least 3 mL of blood from a central venous access device * Hemodynamically stable * Available for follow-up assessments Exclusion Criteria: * Inability to infuse at least 2 mL of saline through the ...

Countries:United States
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Frequently asked questions about Alfimeprase

What is Alfimeprase used for?

Alfimeprase is being developed to treat thrombosis, including occluded central and indwelling catheters and arterial occlusive diseases. It is intended to dissolve blood clots in these settings. The clinical program has studied it in adults with catheter occlusion and with acute peripheral arterial occlusion, where clot removal may help avoid surgery on leg arteries.

What does Alfimeprase target?

Alfimeprase targets fibrinogen alpha, beta, and gamma chains, known as FGA, FGB, and FGG. It is a hydrolytic enzyme, meaning it acts by cleaving these fibrinogen chain substrates. This fibrinogen-directed activity underlies its use in breaking down clot material in occluded catheters and occluded peripheral arteries.

Who is developing Alfimeprase?

Alfimeprase is being developed by Oruka Therapeutics, Inc., which trades under the ticker ORKA. The company is the sponsor associated with the drug's clinical development program in cardiovascular and thrombosis indications, including occluded catheters and arterial occlusive diseases.

What phase is Alfimeprase in?

Alfimeprase has reached Phase 3 clinical development. Its Phase 3 program includes completed studies in occluded central catheters and in arterial occlusive disease, along with an earlier Phase 2 study in acute peripheral arterial occlusion. It is an investigational agent and is not described as approved.

What clinical trials is Alfimeprase in?

Alfimeprase has been studied in completed trials including NCT00346424 and NCT00322270, both Phase 3 studies in subjects with occluded catheters, and NCT00115999, a Phase 3 study in arterial occlusive disease of the leg. A Phase 2 trial, NCT00073554, evaluated thrombolysis in acute peripheral arterial occlusion. All are completed.

How many patients were enrolled in Alfimeprase trials?

Across the Alfimeprase clinical program, total enrollment is approximately 400 participants. The Phase 3 catheter occlusion study NCT00346424 enrolled 300 subjects, and the Phase 3 arterial occlusive disease study NCT00115999 also enrolled 300, while the Phase 2 trial NCT00073554 enrolled 100. Trials enrolled adults aged 18 years and older.