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OPN-375

Phase 3

Bilateral Nasal Polyposis | Small molecule | ENT |OptiNose, Inc.|Last Updated: May 8, 2026

Success Probability

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment72

FDA Designations

No designations recorded

Clinical trial landscape

OPN-375 · 4 trials · 3 indications

Phase 3 4
NCT06850805Efficacy and Safety of 186 mcg of OPN-375 Nasal Spray Twice a Day (BID) in Adolescents With Chronic Rhinosinusitis Without Nasal PolypsChronic Rhinosinusitis Without Nasal Polyps
RECRUITING84 Analytics
NCT03960580Study Evaluating the Efficacy and Safety of Intranasal Administration of OPN-375 in Subjects With Chronic Rhinosinusitis Without the Presence of Nasal PolypsChronic Rhinosinusitis
COMPLETED223 Analytics
NCT03747458OPN-375 Efficacy and Safety in Adolescents With Bilateral Nasal PolypsBilateral Nasal Polyposis
ACTIVE NOT_RECRUITING72 Analytics
NCT03781804Study Evaluating the Efficacy and Safety of Intranasal Administration of OPN-375 in Subjects With Chronic Rhinosinusitis With or Without the Presence of Nasal PolypsChronic Rhinosinusitis
COMPLETED332 Analytics
PHASE3RECRUITING
Efficacy and Safety of 186 mcg of OPN-375 Nasal Spray Twice a Day (BID) in Adolescents With Chronic Rhinosinusitis Without Nasal Polyps
Chronic Rhinosinusitis Without Nasal PolypsUnlock trial analytics
PHASE3COMPLETED
Study Evaluating the Efficacy and Safety of Intranasal Administration of OPN-375 in Subjects With Chronic Rhinosinusitis Without the Presence of Nasal Polyps
Chronic RhinosinusitisUnlock trial analytics
PHASE3ACTIVE NOT_RECRUITING
OPN-375 Efficacy and Safety in Adolescents With Bilateral Nasal Polyps
Bilateral Nasal PolyposisUnlock trial analytics
PHASE3COMPLETED
Study Evaluating the Efficacy and Safety of Intranasal Administration of OPN-375 in Subjects With Chronic Rhinosinusitis With or Without the Presence of Nasal Polyps
Chronic RhinosinusitisUnlock trial analytics

Study Endpoints

Primary Endpoints

Change from baseline to the end of Week 4 in the average instantaneous CSS (evaluation of symptom severity immediately preceding the time of scoring).
4 Weeks

The CSS consists of the sum of the scores (0-3) assigned to each of the following symptoms of CRS: nasal congestion, nasal discharge (anterior and/or posterior), facial pain/pressure sensation, where 0 = no symptoms, 1 = mild symptoms, 2 = moderate symptoms, and 3 = severe symptoms. The total CSS for each day can range from 0 to 9. Participants will report symptom severity immediately preceding the time of scoring every morning (AM). The baseline CSS is the average of the CSS's over the last 7 days of the single-blind run-in period. The end of Week 4 CSS is the average of the CSS's over the 7 days before Week 4.

Change From Baseline in Symptoms as Measured by a Composite Score for Each Symptom of Nasal Congestion, Facial Pain or Pressure Sensation, and Nasal Discharge (Anterior and/or Posterior) at the End of Week 4
4 Weeks

Change from baseline to the end of Week 4 in average total instantaneous AM scores (evaluation of symptom severity immediately preceding the time of scoring) for each symptom: nasal congestion, nasal discharge (anterior and/or posterior), facial pain/pressure sensation. Baseline scores are the averaged total instantaneous AM scores over the last 7 days of the single blind run in period, and the end of Week 4, scores are averaged over the 7 days from the subject diary. Range of scores for each nasal symptom is 0= none, 1 = mild, 2 = moderate, 3 = severe. Composite score is a sum of the 3 symptom scores and will range from 0 to 9.

Change From Baseline to Week 24/Early Termination (ET) in the Average Percent of the Volume Opacified (APOV) in the Ethmoid and Maxillary Sinuses.
Baseline, Week 24

Change from baseline to Week 24/ET in the average percent of ethmoid and maxillary sinus volume opacified as measured by CT. Percent volume opacified can range from 0% to 100%. Outcome measure is the percentage change from percent opacification at baseline to percent opacification at Week 24; therefore, change in opacification volume can range from -100% to 100%. For example, if Baseline opacification was 68.22% and Week 24 opacification was 66.11%, then the change would be reported as -2.11%.

Change in nasal congestion/obstruction symptoms (mild, moderate, severe) at the end of Week 4
4 Weeks

Change in nasal congestion/obstruction symptoms at the end of Week 4 measured by the 7-day average instantaneous morning (AM) diary symptom scores (ADS7-IA). The nasal symptom scale is what is used to score the nasal congestion/obstruction score, which is recorded in the diary. Nasal symptom scale is graded on a scale of 0=no symptom, 1=mild symptom, 2=moderate symptom, 3=severe symptom.

Mean change from baseline at Week 16 in total polyp grade
16 Weeks

Change in total polyp grade (sum of scores from both nasal cavities) at Week 16 as determined by a nasal polyp grading scale score measured using a 0 to 6 point severity grading scale, with 0 (no polyps) to 3 (severe polyps) points per nostril

Change From Baseline to Week 24/Early Termination (ET) in the Average Percent of the Volume Opacified in the Ethmoid and Maxillary Sinuses
Baseline, Week 24

Change from baseline to Week 24/ET in the average percent of ethmoid and maxillary sinus volume opacified as measured by CT. Percent volume opacified can range from 0% to 100%. Outcome measure is the percentage change from percent opacification at baseline to percent opacification at Week 24; therefore, change in opacification volume can range from -100% to 100%. For example, if Baseline opacification was 68.22% and Week 24 opacification was 66.11%, then the change would be reported as -2.11%.

Secondary Endpoints

Frequency of acute exacerbations of CRS over the 12-week treatment period
12 weeks
Change from baseline to the end of Week 4 on CSS score in subjects using an intranasal steroid treatment for CRS within 30 days of Visit 1/Screening
4 Weeks
Change from baseline to the end of Weeks 8 and 12 in CSS
8 Weeks; 12 Weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Placebo BIDPLACEBO_COMPARATORDouble-Blind Treatment Phase: Intranasal administration of matching placebo BID x 12 weeks
OPN-375 186 µg BIDACTIVE_COMPARATORDouble-Blind Treatment Phase: Intranasal administration of OPN-375 186 µg x 12 weeks
OPN-375 186 μg BIDACTIVE_COMPARATOROPN-375 186 μg BID x 24 Weeks
OPN-375 372 μg BIDACTIVE_COMPARATOROPN-375 372 μg BID x 24 Weeks
PlaceboPLACEBO_COMPARATORMatching Placebo BID x 24 Weeks

Interventions

NameTypeDescription
OPN-375DRUGOPN-375 (fluticasone propionate) delivered via exhalation delivery system (EDS) BID
PlaceboDRUGPlacebo solution administered via exhalation delivery system (EDS).
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Eligibility Criteria

Age Range12 Years to 17 Years
SexALL
Healthy VolunteersNo
Study Sites21

Inclusion Criteria: 1. Male or female subjects aged 12 to 17 years, inclusive, at time of Visit 1 (Screening) 2. Female subjects, if sexually active, must: 1. be practicing an effective method of birth control (e.g., prescription oral contraceptives, contraceptive injections, contraceptive patc...

Countries:United StatesAustraliaBulgariaCzechiaGeorgiaNew ZealandPolandRomaniaSpainUnited KingdomArgentinaCanadaRussiaSweden
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Frequently asked questions about OPN-375

What is OPN-375 used for?

OPN-375 is an investigational small molecule being developed for chronic rhinosinusitis, chronic rhinosinusitis without nasal polyps, and bilateral nasal polyposis. It is administered as an intranasal spray and is currently in Phase 3 clinical trials for these ENT conditions.

Who makes OPN-375?

OPN-375 is being developed by OptiNose, Inc., a biopharmaceutical company traded on the NASDAQ under the ticker symbol OPTN. The company is conducting Phase 3 clinical trials to evaluate the drug's efficacy and safety in patients with chronic rhinosinusitis and nasal polyps.

What phase is OPN-375 in?

OPN-375 is in Phase 3 clinical development. It is not FDA approved and remains investigational. Multiple Phase 3 trials are ongoing or completed, including studies in adolescents and adults with chronic rhinosinusitis with or without nasal polyps.

What clinical trials is OPN-375 in?

OPN-375 has been studied in several Phase 3 trials. NCT03747458 evaluated efficacy and safety in adolescents with bilateral nasal polyps. NCT03781804 and NCT03960580 studied adults with chronic rhinosinusitis with or without nasal polyps. NCT06850805 is currently recruiting adolescents with chronic rhinosinusitis without nasal polyps.

Is OPN-375 the same as other nasal sprays for sinusitis?

OPN-375 is a distinct investigational drug developed by OptiNose. It is not known to be the same as any other marketed product. Its mechanism of action is not disclosed in available information, and it is being studied specifically for chronic rhinosinusitis and nasal polyposis.