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Tropifexor

Phase 2

Non-alcoholic Steatohepatitis (NASH) | Small molecule | Infectious Disease |Novartis AG|Last Updated: Apr 29, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment193
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03517540Study of Safety, Tolerability, and Efficacy of a Combination Treatment of LJN452 and CVC in Adult Patients With NASH and Liver FibrosisPHASE2 COMPLETED 193Sep 11, 2018Oct 15, 2020Apr 29, 202265 United States, Argentina +15
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Study Endpoints
Primary Endpoints
Number of Participants With Adverse Events
AEs were collected from first dose of study treatment until end of study treatment at week 48 and then up to maximum duration of 66 weeks

Occurrence of adverse events and serious adverse events Adverse Events (AEs) are any untoward sign or symptom that occurs during the study treatment and then up to 66 weeks

Secondary Endpoints
Proportion of Participants Who Have at Least a One Point Improvement in Fibrosis
baseline to 48 Weeks
Proportion of Participants With Resolution of Steatohepatitis
baseline to 48 weeks
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Arm A: Tropifexor (LJN452) - Dose 1EXPERIMENTALtropifexor 140 mcg, once daily; given orally
Arm B: Cenicriviroc (CVC)EXPERIMENTALCVC 150 mg, once daily; given orally
Arm C: Tropifexor (LJN452) Dose 1 + CVCEXPERIMENTALtropifexor 140 mcg + CVC 150 mg, once daily; given orally
Arm D: Tropifexor Dose 2 + CVCEXPERIMENTALtropifexor 90 mcg + CVC 150 mg, once daily; given orally
Interventions
NameTypeDescription
Tropifexor (LJN452)DRUGComparison with monotherapy and different combination doses
Cenicriviroc (CVC)DRUGComparison with monotherapy and different combination doses
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites65

Inclusion Criteria: Written informed consent Male and female patients 18 years or older (at the time of the screening visit). Patients must weigh at least 50 kg (110 lb) and no more than 200 kg (440 lb) to participate in the study. Able to communicate well with the investigator, to understand and ...

Countries:United StatesArgentinaBelgiumCanadaCzechiaEgyptFranceGermanyIndiaIsraelItalyLatviaRussiaSingaporeSpainTurkey (Türkiye)United Kingdom
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