Recent Updates
Recently added Catalysts

LML134

Phase 1

Healthy Volunteers | Small molecule | Other |Novartis AG|Last Updated: Oct 27, 2016

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

Double-BlindCONTROLLED
Total Trials1
Total Enrollment133

FDA Designations

No designations recorded

Clinical trial landscape

LML134 · 1 trial · 1 indication

Phase 1 1
NCT02334449First-in-human Study to Assess the Safety and Pharmacokinetics of LML134 in Healthy VolunteersHealthy Volunteers
COMPLETED133 Analytics
PHASE1COMPLETED
First-in-human Study to Assess the Safety and Pharmacokinetics of LML134 in Healthy Volunteers
Healthy VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

Adverse events assessments after single and multiple ascending dose administration at baseline and repeatedly until study completion
Starting about 24 hours before dosing and continued until about 7-14 days after last dose

This safety outcome combines the measure of the number of subjects experiencing adverse events (AEs), the nature and severity of those AEs and their relationship to the study treatments.

Cardiovascular safety assessments after single and multiple ascending dose administration at baseline and repeatedly until study completion
Starting about 24 hours before dosing and continued until about 7-14 days after last dose

This safety outcome combines the measure of a set of cardiovascular safety parameters extracted from ECGs, 25 hours-Holter ECGs and from vital signs assessments

Central nervous system safety assessments after single and multiple ascending dose administration at baseline and repeatedly until study completion
Starting about 24 hours before dosing and continued until about 7-14 days after last dose

This safety outcome combines the measure of a set of central nervous system safety parameters extracted from EEGs and neurological examinations

Ocular safety assessments after single and multiple ascending dose administration at baseline and repeatedly until study completion
Starting about 24 hours before dosing and continued until about 7-14 days after last dose

This safety outcome combined the measure of a set of ocular parameters including best corrected visual acuity and other parameters assessed by the mean of slit lamp biomicroscopy and dilated ophthalmoscopy examinations and by optical coherence tomography and electroretinography

General safety assessments after single and multiple ascending dose administration at baseline and repeatedly until study completion
Starting about 24 hours before dosing and continued until about 7-14 days after last dose

This general safety outcome combines the measure of blood laboratory parameters and the outcome of physical examinations

Secondary Endpoints

Pharmacokinetics (PK) of LML134: time to reach the maximum concentration after a single drug administration (Tmax) in Part 1 and in Part 3
Starting 1hour prior to dosing on Day 1 and until 72 hours after dosing (Day 4)
PK of LML134: Observed maximum serum concentration following single drug administration (Cmax) in Part 1 and Part 3
Starting 1hour prior to dosing on Day 1 and until 72 hours after dosing (Day 4)
PK of LML134: Area under the serum concentration-time curve from time zero to the time of last quantifiable concentration (AUClast) in Part 1 and Part 3
Starting 1hour prior to dosing on Day 1 and until 72 hours after dosing (Day 4)
Unlock Study Endpoints

Study Design & Arms

MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Single dose study partEXPERIMENTALthere will be 8 cohorts of healthy volunteers dosed with single doses of LML134 (8 planned dose levels) or with placebo and 2 potential additional cohorts (also dosed with single dose of LML134 or placebo)
Multiple dose study partEXPERIMENTALthere will be 3 cohorts of healthy volunteers dosed with multiple doses of LML134 (3 planned dose levels) or placebo and one potential additional cohort (also dosed with multiple doses of LML134 or placebo)

Interventions

NameTypeDescription
LML134DRUGLML134 will be administered first as single doses and then as multiple doses
PlaceboDRUGAll study cohorts (except food effect cohort) are placebo controlled
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male and female subjects age 18 to 55 years of age included, and in good health as determined by medical history, physical examination, vital signs, electrocardiogram, and laboratory tests. * Written informed consent must be obtained before any assessment is performed....

Countries:Germany
Unlock Eligibility Criteria

Frequently asked questions about LML134

What is LML134 used for?

LML134 is an investigational small molecule being studied in healthy volunteers. It is not approved for any disease and is in early clinical development. The only completed trial assessed its safety and pharmacokinetics in healthy participants, meaning it has not yet been tested for a specific medical condition.

Who makes LML134?

LML134 is being developed by Novartis AG, which trades under the ticker NVS. The company sponsored a first-in-human study of the drug in healthy volunteers. As of the available data, LML134 remains an investigational asset in Phase 1 development.

What phase is LML134 in?

LML134 is in Phase 1 clinical development. A single first-in-human study has been completed, and no active trials are currently listed. The drug is investigational and has not been approved by regulatory authorities. Its safety and pharmacokinetics were evaluated in healthy volunteers.

What clinical trials is LML134 in?

LML134 has one completed clinical trial, registered as NCT02334449. This was a first-in-human study to assess the safety and pharmacokinetics of LML134 in healthy volunteers. The trial enrolled 133 participants in Germany and was double-blind and controlled, though it was not randomized.

Is LML134 FDA approved?

No, LML134 is not FDA approved. It is an investigational drug that has completed a Phase 1 trial in healthy volunteers. The drug is still in clinical development and has not been evaluated for any disease indication. Approval status cannot be confirmed beyond the available trial data.