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LFX453 H1

Phase 1

Healthy | Small molecule | Other |Novartis AG|Last Updated: May 15, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLED
Total Trials1
Total Enrollment41
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02052687A First-in-human Study to Evaluate the Safety, Tolerability and Pharmacokinetics of LFX453PHASE1 COMPLETED 41Jan 1, 2014Jun 1, 2014May 15, 20151 United Kingdom
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Study Endpoints
Primary Endpoints
General safety (number of subjects with adverse events)
14 days

Summarized statistics on adverse events will be reported under categories such as total adverse events, serious adverse events and death.

Local skin tolerability (tolerability score)
14 days

Summarized statistics on 5-point scale tolerability scores over 14 days of treatment.

Secondary Endpoints
All parts: Amount (ng/mL) of LFX453 in plasma
14 days
Part 1 and 2: LFX453 concentrations (ng/g) in the skin
Day 14 and between days 18-21
All parts: LFX453 concentration (ng/mL) in urine
Day 14
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelSINGLE_GROUP
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Part 1: LFX453/placeboEXPERIMENTALonce daily: LFX453 cream 1 high dose / LFX453 cream 1 low dose /Placebo 1 / LFX453 cream 2 high dose / LFX453 cream 2 low dose / Placebo 2
Part 2 groupA: LFX453/placeboEXPERIMENTALonce daily: LFX453 cream 1 / Placebo 1
Part 2 groupB: LFX453/placeboEXPERIMENTALonce daily: LFX453 cream 2 / Placebo 2
Part 2 groupC: LFX453/LFX453EXPERIMENTALonce daily: LFX453 cream 1 / LFX453 cream 2
Part 2 groupD: ImiquimodOTHERonce daily: imiquimod cream
Part 3: LFX453/placeboEXPERIMENTALtwice daily: LFX453 cream 1 high dose / LFX453 cream 1 low dose /Placebo 1 / LFX453 cream 2 high dose / LFX453 cream 2 low dose / Placebo 2
Interventions
NameTypeDescription
LFX453 H1DRUGLFX453 high dose cream 1
LFX453 L1DRUGLFX453 low dose cream 1
LFX453 H2DRUGLFX453 high dose cream 2
LFX453 L2DRUGLFX453 low dose cream 2
ImiquimodDRUGImiquimod cream
Placebo 1DRUGPlacebo cream 1
Placebo 2DRUGPlacebo cream 2
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male and female subjects of non-childbearing potential, 18 to 65 years of age inclusive (at the time of the screening visit), and in good health as determined by past medical history, physical examination, vital signs, electrocardiogram, and laboratory tests at screeni...

Countries:United Kingdom
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