Recent Updates
Recently added Catalysts

Sitagliptin anhydrous formulation

Phase 1

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Merck & Company, Inc.|Last Updated: Aug 19, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment12
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00944450Study of the Bioequivalence of Two Tablet Forms of MK0431 (0431-027)PHASE1 COMPLETED 12Aug 1, 2004Nov 1, 2004Aug 19, 2015 -
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Area Under the Curve (AUC(0 to Infinity)) Following Single Dose Administration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)
Through 72 Hours Following the Administration of the Medication

Area Under the Plasma Concentration-Time Curve and peak concentration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)

Peak Plasma Concentration (Cmax) Following Single Dose Administration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)
Through 72 Hours Following the Administration of the Medication

Peak Plasma concentration (Cmax) for the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)

Unlock Study Endpoints
Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
1ACTIVE_COMPARATORSitagliptin anhydrous formulation
2ACTIVE_COMPARATORSitagliptin monohydrate FMI formulation
Interventions
NameTypeDescription
Sitagliptin phosphate anhydrous formulationDRUGSingle dose sitagliptin 100 mg tablets (anhydrous form) in one of two treatment periods.
Comparator: sitagliptin phosphate monohydrate formDRUGSingle dose sitagliptin 100 mg tablets \[monohydrate Final Market Image (FMI) form\] in one of two treatment periods.
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes

Inclusion Criteria: * Subject is in good health * Female subjects must have a negative pregnancy test * Subject is within 30% of ideal body weight * Subject does not smoke * Subject agrees to follow the study guidelines Exclusion Criteria: * Subject has a history of any illness that might confoun...

Unlock Eligibility Criteria