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Sitagliptin anhydrous formulation

Phase 1

Type 2 Diabetes Mellitus | Small molecule | Metabolic |Merck & Company, Inc.|Last Updated: Aug 19, 2015

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment12

FDA Designations

No designations recorded

Clinical trial landscape

Sitagliptin anhydrous formulation · 1 trial · 1 indication

Phase 1 1
NCT00944450Study of the Bioequivalence of Two Tablet Forms of MK0431 (0431-027)Type 2 Diabetes Mellitus
COMPLETED12 Analytics
PHASE1COMPLETED
Study of the Bioequivalence of Two Tablet Forms of MK0431 (0431-027)
Type 2 Diabetes MellitusUnlock trial analytics

Study Endpoints

Primary Endpoints

Area Under the Curve (AUC(0 to Infinity)) Following Single Dose Administration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)
Through 72 Hours Following the Administration of the Medication

Area Under the Plasma Concentration-Time Curve and peak concentration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)

Peak Plasma Concentration (Cmax) Following Single Dose Administration of the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)
Through 72 Hours Following the Administration of the Medication

Peak Plasma concentration (Cmax) for the Anhydrous and Monohydrate Forms of MK0431 (Sitagliptin)

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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
1ACTIVE_COMPARATORSitagliptin anhydrous formulation
2ACTIVE_COMPARATORSitagliptin monohydrate FMI formulation

Interventions

NameTypeDescription
Sitagliptin phosphate anhydrous formulationDRUGSingle dose sitagliptin 100 mg tablets (anhydrous form) in one of two treatment periods.
Comparator: sitagliptin phosphate monohydrate formDRUGSingle dose sitagliptin 100 mg tablets \[monohydrate Final Market Image (FMI) form\] in one of two treatment periods.
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes

Inclusion Criteria: * Subject is in good health * Female subjects must have a negative pregnancy test * Subject is within 30% of ideal body weight * Subject does not smoke * Subject agrees to follow the study guidelines Exclusion Criteria: * Subject has a history of any illness that might confoun...

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Frequently asked questions about Sitagliptin anhydrous formulation

What is Sitagliptin anhydrous formulation used for?

Sitagliptin anhydrous formulation is used for Type 2 Diabetes Mellitus. It is a small molecule being developed by Merck & Company, Inc. (MRK) as an investigational treatment for this condition. The drug is currently in Phase 1 clinical development.

Who makes Sitagliptin anhydrous formulation?

Merck & Company, Inc. (MRK) is developing Sitagliptin anhydrous formulation. The company is conducting clinical trials to evaluate this small molecule for the treatment of Type 2 Diabetes Mellitus. The drug is currently in Phase 1 development.

What phase is Sitagliptin anhydrous formulation in?

Sitagliptin anhydrous formulation is in Phase 1 clinical development. It is an investigational drug for Type 2 Diabetes Mellitus and has not been approved by regulatory authorities. One Phase 1 trial has been completed.

What clinical trials is Sitagliptin anhydrous formulation in?

Sitagliptin anhydrous formulation has one completed clinical trial, NCT00944450, titled "Study of the Bioequivalence of Two Tablet Forms of MK0431 (0431-027)". This Phase 1 trial enrolled 12 participants with Type 2 Diabetes Mellitus and was active-controlled.

Is Sitagliptin anhydrous formulation the same as MK0431?

Sitagliptin anhydrous formulation is also known as MK0431. The clinical trial NCT00944450 refers to the drug as MK0431, confirming that these names refer to the same investigational compound being developed by Merck & Company, Inc. for Type 2 Diabetes Mellitus.