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MK-0822

Phase 1

Hepatic Insufficiency | Small molecule | Gastrointestinal |Merck & Company, Inc.|Last Updated: Aug 29, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment17
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01512693Assessment of Pharmacokinetics of Single Dose Odanacatib (MK-0822) in Participants With Moderate Hepatic Insufficiency (MK-0822-070)PHASE1 COMPLETED 17Feb 23, 2012Apr 24, 2012Aug 29, 2018 -
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Study Endpoints
Primary Endpoints
Area Under the Concentration-time Curve of MK-0822 From Time 0 to Infinity (AUC0-∞) After Single Dose
Pre-dose and 1, 2, 4, 6, 9, 12, 16, 24, 32, 48, 72, 96, 120, 168, 240, and 336 hours postdose

For healthy and moderate hepatic insufficiency participants, plasma samples were collected from predose to 336 hours postdose for determination of AUC0-∞ (Total AUC). AUC0-∞ is a measure of total drug exposure.

Secondary Endpoints
Maximum Concentration (Cmax) of MK-0822 After Single Dose
Pre-dose and 1, 2, 4, 6, 9, 12, 16, 24, 32, 48, 72, 96, 120, 168, 240, and 336 hours postdose
Time to Maximum Concentration (Tmax) of MK-0822 After Single Dose
Pre-dose and 1, 2, 4, 6, 9, 12, 16, 24, 32, 48, 72, 96, 120, 168, 240, and 336 hours postdose
Apparent Terminal Half-life (t1/2) of MK-0822 After Single Dose
Pre-dose and 1, 2, 4, 6, 9, 12, 16, 24, 32, 48, 72, 96, 120, 168, 240, and 336 hours postdose
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Moderate Hepatic Insufficiency GroupEXPERIMENTALSingle-dose administration of odanacatib 50 mg to participants with moderate hepatic insufficiency.
Healthy Matched Control GroupEXPERIMENTALSingle-dose administration of odanacatib 50 mg to healthy matched control participants.
Interventions
NameTypeDescription
MK-0822DRUGA single oral dose (50 mg tablet) of MK 0822 will be administered on Day 1 after an overnight fast.
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersYes

Inclusion Criteria: * Not currently pregnant, nursing or planning to be pregnant through-out the course of the study; agree to use specified contraception per protocol requirement * Body Mass Index (BMI) of ≤ 39 kg/m\^2 (not obese) * Judged to be in good health (for healthy participant population) ...

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