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Human ADME

Phase 1

Healthy | Small molecule | Other |Merck & Company, Inc.|Last Updated: Nov 15, 2019

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLEDBiomarker
Total Trials1
Total Enrollment6

FDA Designations

No designations recorded

Clinical trial landscape

Human ADME · 1 trial · 1 indication

Phase 1 1
NCT01442831Evaluate the Absorption, Metabolism, And Excretion Of Orally Administered [14C] TR 701 In Healthy Adult Male SubjectsHealthy
COMPLETED6 Analytics
PHASE1COMPLETED
Evaluate the Absorption, Metabolism, And Excretion Of Orally Administered [14C] TR 701 In Healthy Adult Male Subjects
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Study Endpoints

Primary Endpoints

To describe the single dose plasma PK of TR-700, the microbiologically active molecule
pre dose, 0.5, 1, 1.5, 2, 3, 4, 6, 8, 12, 24, 36, 48, 72, 96, then daily up to 312 hours post dose

To describe the single dose pharmacokinetics (Cmax, Tmax, AUC, t 1/2, CL/F) of total radioactivity in plasma, whole blood, urine and feces following oral (PO) administration of \[14C\] TR 701 in healthy adult male subjects

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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Human ADMEEXPERIMENTAL -

Interventions

NameTypeDescription
Human ADMEDRUGOral single dose
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Eligibility Criteria

Age Range18 Years to 50 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Males, between 18 and 50 years of age, inclusive. 2. Body mass index (BMI) of 20 kg/m2 to 29.9 kg/m2, inclusive. 3. In good health, determined by no clinically significant findings from medical history, physical examination (Check-in), 12-lead ECG, and vital signs. Exclusion...

Countries:United States
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Frequently asked questions about Human ADME

What is Human ADME used for?

Human ADME is an investigational small molecule being studied in healthy adult male subjects. It is being evaluated in a Phase 1 clinical trial to assess the absorption, metabolism, and excretion of orally administered [14C] TR 701. The drug is not approved and remains in clinical development.

Who makes Human ADME?

Human ADME is being developed by Merck & Company, Inc., which trades under the ticker symbol MRK. The company is conducting clinical research on this investigational small molecule in the United States.

What phase is Human ADME in?

Human ADME is in Phase 1 clinical development. The single trial listed for this drug has been completed. It is an investigational drug and has not been approved for any use.

What clinical trials is Human ADME in?

Human ADME has one completed Phase 1 trial, NCT01442831, titled 'Evaluate the Absorption, Metabolism, And Excretion Of Orally Administered [14C] TR 701 In Healthy Adult Male Subjects.' The trial enrolled 6 participants in the United States and was not randomized or blinded.

Is Human ADME the same as TR 701?

Human ADME is the name of the study drug in the clinical trial, and the trial evaluates [14C] TR 701, which is the radiolabeled form of the drug. The drug is referred to as TR 701 in the trial title, indicating it is the same compound being studied.