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ACE-083

Phase 1

Musculoskeletal Diseases | Small molecule | Musculoskeletal |Merck & Company, Inc.|Last Updated: Sep 23, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials1
Total Enrollment58
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02257489Phase 1 Study of ACE-083 in Healthy SubjectsPHASE1 COMPLETED 58Sep 1, 2014Apr 1, 2016Sep 23, 20221 United States
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Study Endpoints
Primary Endpoints
ACE-083 Safety and Tolerability: Number of Subjects With Adverse Events
From initiation of treatment (Study Day 1) to end of follow up period (up to Study Day 106)

Safety/tolerability assessment, following intramuscular administration, includes adverse events, injection site reactions, laboratory measurements, vital signs, etc.

Secondary Endpoints
ACE-083 Pharmacokinetics: Maximum Measured Plasma Concentrations
PK samples were collected predose, and at 3 hours and 6 hours postdose.
ACE-083 Pharmacodynamics
From initiation of treatment (Study Day 1) to end of follow up period (up to Study Day 106)
ACE-083 Pharmacokinetics: Time of the Maximum Measured Plasma Concentration
PK samples were collected predose, and at 3 hours and 6 hours postdose.
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
50 mg single doseEXPERIMENTAL8 subjects in total; 6 subjects to received ACE-083 (50 mg) and 2 subjects to receive placebo, single injection, intramuscularly
100 mg single doseEXPERIMENTAL8 subjects in total; 6 subjects to received ACE-083 (100 mg) and 2 subjects to receive placebo, single injection, intramuscularly
200 mg single doseEXPERIMENTAL8 subjects in total; 6 subjects to received ACE-083 (200 mg) and 2 subjects to receive placebo, single injection, intramuscularly
100 mg multiple doseEXPERIMENTAL8 subjects in total; 6 subjects to received ACE-083 (100 mg) and 2 subjects to receive placebo, two injections 3 weeks apart, intramuscularly
200 mg multiple doseEXPERIMENTAL8 subjects in total; 6 subjects to received ACE-083 (200 mg) and 2 subjects to receive placebo, two injections 3 weeks apart, intramuscularly
100 mg (multiple dose)EXPERIMENTAL9 subjects in total; 6 subjects to received ACE-083 (100 mg) and 3 subjects to receive placebo, two injections 3 weeks apart, intramuscularly
150 mg multiple doseEXPERIMENTAL9 subjects in total; 6 subjects to received ACE-083 (150 mg) and 3 subjects to receive placebo, two injections 3 weeks apart, intramuscularly
Interventions
NameTypeDescription
ACE-083DRUGrecombinant fusion protein
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Eligibility Criteria
Age Range45 Years — 75 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Postmenopausal women, defined by follicle stimulating hormone (FSH) level \> 40 IU/L and either 12 months of spontaneous amenorrhea or at least 6 months post-surgical bilateral oophorectomy and/or hysterectomy * BMI 18.5-32 kg/m2 * Clinical laboratory values that meet the foll...

Countries:United States
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