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Telotristat Ethyl

Phase 1

Hepatic Impairment | Small molecule | Gastrointestinal |Lexicon Pharmaceuticals, Inc.|Last Updated: Oct 15, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment16
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03423446Study to Evaluate the Pharmacokinetics of Telotristat Ethyl in Subjects With Severe Hepatic ImpairmentPHASE1 COMPLETED 16Nov 28, 2017Jun 15, 2018Oct 15, 20183 United States
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Study Endpoints
Primary Endpoints
Maximum observed concentration of telotristat ethyl
4 days
Time of maximum observed concentration of telotristat ethyl
4 days
Area under the plasma concentration-time curve beginning from the first dose until the last quantifiable concentration of telotristat ethyl
4 days
Secondary Endpoints
Number of adverse events
Up to 9 days
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Severe Hepatic ImpairmentEXPERIMENTALUp to 8 subjects with severe hepatic impairment (Child-Pugh Class C, score of 10 to 15 points)
Healthy ControlEXPERIMENTALUp to 8 healthy control subjects with normal hepatic function
Interventions
NameTypeDescription
Telotristat EthylDRUGTelotristat ethyl (TE) 250 mg (1 x 250-mg tablet), single dose
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersYes
Study Sites3

Inclusion Criteria: * Adult male and female subjects ≥18 to ≤70 years of age, inclusive, at the time of Screening: 1. Females of non-childbearing potential are to be surgically sterile (documented hysterectomy, tubal ligation, or bilateral salpingo-oophorectomy) or postmenopausal (defined as at ...

Countries:United States
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