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Schedule A

Phase 1

Healthy | Small molecule | Other |Lexicon Pharmaceuticals, Inc.|Last Updated: May 19, 2011

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment14
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01334242A Study to Determine the Pharmacodynamics of LX4211 Relative to Meals in Healthy SubjectsPHASE1 COMPLETED 14Mar 1, 2011 -May 19, 20111 United States
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Study Endpoints
Primary Endpoints
Urinary glucose excretion
24 hours collection on Day -1 and Days 7-13
Fasting Plasma Glucose
Day -1 and Days 7-12
Postprandial Glucose
Day -1 and Days 7-12
Insulin
Day -1 and Days 7-12
Glucagon-like peptide 1 (total and active)
Day -1 and Days 7-12
Peptide YY
Day -1 and Days 7-12
Secondary Endpoints
Number of Participants with Adverse Events
Day 1 to Day 14
Blood chemistry
Day -2, Day 7 and Day 13
Hematology
Day -2, Day 7 and Day 13
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
LX4211EXPERIMENTAL400 mg of LX4211 administered orally
PlaceboPLACEBO_COMPARATORNonidentical placebo administered orally
Interventions
NameTypeDescription
Schedule ADRUGDosing 1 hour before breakfast
Schedule BDRUGDosing 0.5 hour before breakfast
Schedule CDRUGDosing immediately before breakfast
Schedule DDRUGDosing immediately before lunch
Schedule EDRUGSplit dose, dosing 1 hour before breakfast and dinner
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Adults ≥18 and ≤55 years of age * Vital signs at Screening in the following ranges: systolic blood pressure, 90-140 mm Hg; diastolic blood pressure, 50-90 mm Hg; heart rate, 50-100 bpm * Body mass index (BMI) ≥18 and ≤35 kg/sq m * Able to provide written informed consent Excl...

Countries:United States
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