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LX1606

Phase 1

Carcinoid Syndrome | Small molecule | Oncology |Lexicon Pharmaceuticals, Inc.|Last Updated: Oct 23, 2013

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment8

FDA Designations

No designations recorded

Clinical trial landscape

LX1606 · 1 trial · 1 indication

Phase 1 1
NCT01932528An Open-label Study to Evaluate the Absorption, Metabolism, and Excretion of [14C]-Telotristat Etiprate in MalesCarcinoid Syndrome
COMPLETED8 Analytics
PHASE1COMPLETED
An Open-label Study to Evaluate the Absorption, Metabolism, and Excretion of [14C]-Telotristat Etiprate in Males
Carcinoid SyndromeUnlock trial analytics

Study Endpoints

Primary Endpoints

Maximum plasma concentration of LX1606 and LX1033
7 days

Secondary Endpoints

Time to maximum plasma concentration of and LX1033
7 days
Determination of total radioactivity in blood and plasma
7 days
Mass balance recovery of total radioactivity in urine and feces
7 days
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
500 mg LX606EXPERIMENTALAll subjects will receive a single oral 500 mg dose of \[14C\]-LX1606.

Interventions

NameTypeDescription
500 mg [14C]-LX1606DRUG500 mg dose of LX1606 containing a target dose of 3.32 Megabecquerel (MBq) of radiation as \[14C\]-LX1606.
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Eligibility Criteria

Age Range30 Years to 65 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male subjects aged 30 to 65 years of age. * Male subjects and their partners must agree to use an adequate method of contraception * Historically able to produce a minimum of 1 bowel movement every day on most days Exclusion Criteria: * Female subjects * Use of any m...

Countries:United Kingdom
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Frequently asked questions about LX1606

What is LX1606 used for?

LX1606 is an investigational small molecule being developed for carcinoid syndrome, a condition that can occur in patients with neuroendocrine tumors. It is currently in Phase 1 clinical development and has not been approved by regulatory authorities.

Who makes LX1606?

LX1606 is being developed by Lexicon Pharmaceuticals, Inc., a biopharmaceutical company traded on the Nasdaq under the ticker symbol LXRX. The company is conducting clinical trials to evaluate the drug's safety and pharmacokinetics.

What phase is LX1606 in?

LX1606 is in Phase 1 clinical development. It is an investigational drug and has not been approved for any use. One Phase 1 trial has been completed, and the drug is not currently in active clinical trials.

What clinical trials is LX1606 in?

LX1606 has one completed clinical trial, NCT01932528, an open-label study evaluating the absorption, metabolism, and excretion of [14C]-Telotristat Etiprate in males. The trial enrolled 8 participants in the United Kingdom and was not randomized or double-blinded.

Is LX1606 the same as telotristat etiprate?

LX1606 is also known as telotristat etiprate. The completed clinical trial NCT01932528 specifically studied [14C]-Telotristat Etiprate, which is the radiolabeled form of the drug used to track its absorption and metabolism in the body.