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GLPG3121

Phase 1

Healthy | Small molecule | Other |Lakefront Biotherapeutics|Last Updated: Sep 19, 2024

Target and mechanism

ModalitySmall molecule

Also known as GLPG3121 SAD, GLPG3121 MAD

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials2
Total Enrollment81

FDA Designations

No designations recorded

Clinical trial landscape

GLPG3121 · 2 trials · 1 indication

Phase 1 2
NCT04856358A Study to Evaluate How Well Single and Multiple Doses of GLPG3121-modified Release Formulation Are Tolerated in Healthy, Adult SubjectsHealthy
COMPLETED50 Analytics
NCT03899909A Study to Evaluate the Effects of a Single and Multiple Oral Doses of GLPG3121 in Adult, Healthy, Male SubjectsHealthy
COMPLETED31 Analytics
PHASE1COMPLETED
A Study to Evaluate How Well Single and Multiple Doses of GLPG3121-modified Release Formulation Are Tolerated in Healthy, Adult Subjects
HealthyUnlock trial analytics
PHASE1COMPLETED
A Study to Evaluate the Effects of a Single and Multiple Oral Doses of GLPG3121 in Adult, Healthy, Male Subjects
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Frequency and severity of treatment emergent adverse events (TEAEs), treatment-emergent serious adverse events, and TEAEs leading to treatment discontinuations
From screening through study completion, an average of 8 months

To evaluate the safety and tolerability of single and multiple ascending oral doses of GLPG3121-modified-release formulation (GLPG3121-MR), in adult, healthy, male subjects compared with placebo

Frequency and severity of treatment emergent adverse events (TEAEs), treatment-emergent serious adverse events, and TEAEs leading to treatment discontinuations.
From screening through study completion, an average of 6 months.

To evaluate the safety and tolerability of single and multiple ascending oral doses of GLPG3121, in adult, healthy, male subjects compared with placebo.

Secondary Endpoints

Maximum observed plasma concentration (Cmax) of GLPG3121 in SAD
Between Day 1 pre-dose and Day 6
Cmax of GLPG3121's main metabolite in SAD
Between Day 1 pre-dose and Day 6
Cmax of GLPG3121 in MAD
Between Day 1 pre-dose and Day 19
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
GLPG3121 SADEXPERIMENTALSingle doses of GLPG3121 at up to 3 dose levels in ascending order
Placebo SADPLACEBO_COMPARATORSingle doses of placebo
GLPG3121 MADEXPERIMENTALMultiple doses of GLPG3121 at up to 3 dose levels in ascending order
Placebo MADPLACEBO_COMPARATORMultiple doses of placebo
GLPG3121 FE fedEXPERIMENTALSingle dose of GLPG3121 in fed state
GLPG3121 FE fastedEXPERIMENTALSingle dose of GLPG3121 in fasted state

Interventions

NameTypeDescription
GLPG3121DRUGGLPG3121 modified-release tablet
PlaceboDRUGMatching placebo
GLPG3121 SADDRUGGLPG3121 oral suspension, single ascending doses
Placebo SADDRUGPlacebo oral suspension
GLPG3121 MADDRUGGLPG3121 oral suspension, multiple ascending doses, daily for 13 days
Placebo MADDRUGPlacebo oral suspension, daily for 13 days
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Eligibility Criteria

Age Range18 Years to 55 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male between 18 and 55 years of age (extremes included), on the date of signing the informed consent form (ICF). * A body mass index (BMI) between 18.0 and 30.0 kg/m2, inclusive. * Judged to be in good health by the investigator based upon the results of a medical history, phy...

Countries:GermanyBelgium
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