Recent Updates
Recently added Catalysts

Clavamox

Phase 1

Bioequivalence | Small molecule | Other |Ligand Pharmaceuticals Incorporated|Last Updated: May 14, 2019

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedACTIVE_CONTROLLEDBiomarker
Total Trials2
Total Enrollment112

FDA Designations

No designations recorded

Clinical trial landscape

Clavamox · 2 trials · 1 indication

Phase 1 2
NCT03702894Bioequivalence Study of Clavamox, Film-coated Tablets, 875 mg + 125 mg Pharmtechnology LLC, Belarus), and Augmentin®, Film-coated Tablets, 875 mg + 125 mg (GlaxoSmithKline Trading CJSC, Russia), in Healthy Volunteers Under Fasting ConditionsBioequivalence
COMPLETED56 Analytics
NCT03616301Bioequivalence Study of Clavamox, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml (Pharmtechnology LLC, Belarus), and Augmentin®, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml (GlaxoSmithKline Trading CJSC, Russia), in Healthy Volunteers Under Fasting ConditionsBioequivalence
COMPLETED56 Analytics
PHASE1COMPLETED
Bioequivalence Study of Clavamox, Film-coated Tablets, 875 mg + 125 mg Pharmtechnology LLC, Belarus), and Augmentin®, Film-coated Tablets, 875 mg + 125 mg (GlaxoSmithKline Trading CJSC, Russia), in Healthy Volunteers Under Fasting Conditions
BioequivalenceUnlock trial analytics
PHASE1COMPLETED
Bioequivalence Study of Clavamox, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml (Pharmtechnology LLC, Belarus), and Augmentin®, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml (GlaxoSmithKline Trading CJSC, Russia), in Healthy Volunteers Under Fasting Conditions
BioequivalenceUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax of amoxicillin for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing

Maximum concentration in plasma among observed concentrations at pre-specified time points

AUC0-t of amoxicillin for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing

Area under the plasma concentration versus time curve from time 0 to the last measured concentration

Cmax of clavulanic acid for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing

Maximum concentration in plasma among observed concentrations at pre-specified time points

AUC0-t of clavulanic acid for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing

Area under the plasma concentration versus time curve from time 0 to the last measured concentration

Secondary Endpoints

AUC0-∞ of amoxicillin for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing
AUC0-∞ of clavulanic acid for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing
Tmax of amoxicillin for the test and the reference products
Time points: 0,00 (within 30 minutes before dosing) and 0.25, 0.5, 0.75, 1.00, 1.25, 1.5, 1.75, 2.00, 2.33, 2.67, 3.00, 3.5, 4.00, 5.00, 6.00, 7.00, 8.00, 10.00 hours after dosing
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Clavamox,Coated Tablets, 875 mg + 125 mgEXPERIMENTALClavamox, Film-coated Tablets, 875 mg + 125 mg, is the test product. 14 of 28 subjects in each of two cohorts (total number of enrolled volunteers - 56) were given a single tablet (containing 875 mg mg of amoxicillin and 125 mg of clavulanic acid) in period 1 and period 2 of the clinical part of the study.
Augmentin®, Coated Tablets, 875 mg + 125 mgACTIVE_COMPARATORAugmentin®, Film-coated Tablets, 875 mg + 125 mg, is the reference product. 14 of 28 subjects in each of two cohorts (total number of enrolled volunteers - 56) were given a single tablet (containing 875 mg mg of amoxicillin and 125 mg of clavulanic acid) in period 1 and period 2 of the clinical part of the study.
Clavamox, Powder for Oral Suspension, 400 mg + 57 mg / 5 mlEXPERIMENTALClavamox, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml is the test product. 14 of 28 subjects in each of two cohorts (total number of enrolled volunteers - 56) will be given single oral dose (5 ml containing 400 mg of amoxicillin and 57 mg of clavulanic acid) in period 1 and period 2 of the clinical part of the study.
Augmentin®, Powder for Oral Suspension, 400 mg + 57 mg / 5 mlACTIVE_COMPARATORAugmentin®, Powder for Oral Suspension, 400 mg + 57 mg / 5 ml is the reference product. 14 of 28 subjects in each of two cohorts (total number of enrolled volunteers - 56) will be given single oral dose (5 ml containing 400 mg of amoxicillin and 57 mg of clavulanic acid) in period 1 and period 2 of the clinical part of the study.

Interventions

NameTypeDescription
ClavamoxDRUGClavamox, Film-coated Tablets, 875 mg + 125 mg, manufactured by Pharmtechnology LLC, Belarus
Augmentin®DRUGAugmentin®, Film-coated Tablets, 875 mg + 125 mg, marketed by GlaxoSmithKline Trading CJSC, Russia
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 45 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Caucasian men or women aged between 18 to 45 years * Subjects having no clinically significant medical history and no clinically significant abnormalities in general physical examination, laboratory assessments and imaging studies. * Body mass index 18.5-29.9 kg/m² with body m...

Countries:Russia
Unlock Eligibility Criteria

Frequently asked questions about Clavamox

What is Clavamox used for?

Clavamox is an investigational small molecule being studied for bioequivalence. It is a powder for oral suspension and film-coated tablets being compared to Augmentin in healthy volunteers under fasting conditions. The drug is in Phase 1 clinical development and is not FDA approved.

Who makes Clavamox?

Clavamox is being developed by Ligand Pharmaceuticals Incorporated, which trades under the ticker LGND. The company is conducting bioequivalence studies of Clavamox against Augmentin in healthy volunteers in Russia.

What phase is Clavamox in?

Clavamox is in Phase 1 clinical development. Two Phase 1 bioequivalence studies have been completed, with a total of 112 participants enrolled. The drug is investigational and has not been approved by the FDA.

What clinical trials is Clavamox in?

Clavamox has two completed Phase 1 trials: NCT03616301, a bioequivalence study of the oral suspension 400 mg + 57 mg per 5 ml, and NCT03702894, a bioequivalence study of film-coated tablets 875 mg + 125 mg. Both compared Clavamox to Augmentin in healthy volunteers under fasting conditions in Russia.

Is Clavamox the same as Augmentin?

Clavamox is being studied as a potential generic equivalent to Augmentin. The bioequivalence trials compare Clavamox formulations to Augmentin products from GlaxoSmithKline. However, Clavamox is a distinct product being developed by Ligand Pharmaceuticals and is not yet approved.