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Aceclofenac film-coated

Phase 1

Bioequivalence | Small molecule | Other |Ligand Pharmaceuticals Incorporated|Last Updated: Jun 28, 2023

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment36

FDA Designations

No designations recorded

Clinical trial landscape

Aceclofenac film-coated · 1 trial · 1 indication

Phase 1 1
NCT05339373Bioequivalence Study of Two Formulations of Tablets Aceclofenac 100 mg in Healthy Volunteers Under Fasting ConditionsBioequivalence
COMPLETED36 Analytics
PHASE1COMPLETED
Bioequivalence Study of Two Formulations of Tablets Aceclofenac 100 mg in Healthy Volunteers Under Fasting Conditions
BioequivalenceUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax of aceclofenac in plasma after administration of the test and the reference products.
Time points 0.00 (prior to each drug administration) and 0.15, 0.30, 0.45, 1.00, 1.15, 1.30, 1.45, 2.00, 2.20, 2.40, 3.00, 3.30, 4.00, 5.00, 6.00, 8.00, 10.00, 12.00, 24.00 hours after each drug administration.

Maximum observed concentration in plasma.

AUC0-t of aceclofenac in plasma after administration of the test and the reference.
Time points 0.00 (prior to each drug administration) and 0.15, 0.30, 0.45, 1.00, 1.15, 1.30, 1.45, 2.00, 2.20, 2.40, 3.00, 3.30, 4.00, 5.00, 6.00, 8.00, 10.00, 12.00, 24.00 hours after each drug administration.

Cumulative area under the concentration time curve calculated from 0 to time of last observed quantifiable concentration using the linear trapezoidal method.

Secondary Endpoints

Tmax of aceclofenac in plasma after administration of the test and the reference products.
Time points 0.00 (prior to each drug administration) and 0.15, 0.30, 0.45, 1.00, 1.15, 1.30, 1.45, 2.00, 2.20, 2.40, 3.00, 3.30, 4.00, 5.00, 6.00, 8.00, 10.00, 12.00, 24.00 hours after each drug administration.
TLQC of aceclofenac in plasma after administration of the test and the reference products.
Time points 0.00 (prior to each drug administration) and 0.15, 0.30, 0.45, 1.00, 1.15, 1.30, 1.45, 2.00, 2.20, 2.40, 3.00, 3.30, 4.00, 5.00, 6.00, 8.00, 10.00, 12.00, 24.00 hours after each drug administration.
AUC0-INF of aceclofenac in plasma after administration of the test and the reference products.
Time points 0.00 (prior to each drug administration) and 0.15, 0.30, 0.45, 1.00, 1.15, 1.30, 1.45, 2.00, 2.20, 2.40, 3.00, 3.30, 4.00, 5.00, 6.00, 8.00, 10.00, 12.00, 24.00 hours after each drug administration.
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Sequence TROTHER18 subjects assigned to the sequence TR will receive a single 100 mg dose of the test product Aceclofenac (1 x 100 mg tablet), marked as T in the sequence, in Period 1 and a single 100 mg dose of the reference product Airtal ® (1 x 100 mg tablet), marked as R in the sequence, in period 2. These treatments will be administered orally with approximately 200 mL of water, in the morning, following a 10-hour overnight fast. The tablet must be swallowed whole and must not be chewed or broken.
Sequence RTOTHER18 subjects assigned to the sequence RT will receive a single 100 mg dose of the test product Airtal ® (1 x 100 mg tablet), marked as R in the sequence, in Period 1 and a single 100 mg dose of thetest product Aceclofenac (1 x 100 mg tablet), marked as T in the sequence, in period 2. These treatments will be administered orally with approximately 200 mL of water, in the morning, following a 10-hour overnight fast. The tablet must be swallowed whole and must not be chewed or broken.

Interventions

NameTypeDescription
Aceclofenac film-coated tablet 100 mgDRUGAceclofenac is manufactured by Pharmtechnology LLC, Republic of Belarus. Each tablet contains 100 mg of aceclofenac.
Airtal® film-coated tablet 100 mgDRUGAirtal ® is manufactured by Gedeon Richter- RUS", Russia / Gedeon Richter, Hungary. Each tablet contains 100 mg of aceclofenac.
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Eligibility Criteria

Age Range18 Years to 45 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Healthy european men or women aged between 18 to 45 years 2. The written consent of the volunteer to be included in the study 3. Verified diagnosis "healthy" according to the anamnesis data and the results of standard clinical, laboratory and instrumental examination methods,...

Countries:Russia
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Frequently asked questions about Aceclofenac film-coated

What is Aceclofenac film-coated used for?

Aceclofenac film-coated is a small molecule drug being studied for bioequivalence, meaning it is evaluated to confirm that a new formulation of aceclofenac 100 mg tablets matches an existing reference product in how it is absorbed and behaves in the body. It is intended for use in healthy volunteers under fasting conditions.

Who makes Aceclofenac film-coated?

Aceclofenac film-coated is being developed by Ligand Pharmaceuticals Incorporated, a company traded on the NASDAQ under the ticker LGND. The drug is currently in Phase 1 clinical development for a bioequivalence study.

What phase is Aceclofenac film-coated in?

Aceclofenac film-coated is in Phase 1 clinical development. It is an investigational drug, not yet approved, and is being studied in a single completed Phase 1 bioequivalence trial. The study enrolled 36 healthy volunteers and was conducted in Russia.

What clinical trials is Aceclofenac film-coated in?

Aceclofenac film-coated has one completed clinical trial, registered as NCT05339373, titled "Bioequivalence Study of Two Formulations of Tablets Aceclofenac 100 mg in Healthy Volunteers Under Fasting Conditions." This Phase 1 study enrolled 36 participants, was randomized and controlled, and took place in Russia.

Is Aceclofenac film-coated the same as aceclofenac?

Aceclofenac film-coated is a formulation of aceclofenac, a nonsteroidal anti-inflammatory drug. The film-coated version refers to the tablet coating, and the study compares two formulations of aceclofenac 100 mg tablets to assess their bioequivalence. No other alternative names are provided.