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Sulopenem-Etzadroxil/Probenecid

Phase 3

Intra Abdominal Infections | Small molecule | Other |Iterum Therapeutics plc|Last Updated: Dec 1, 2020

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindACTIVE_CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment674
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03358576Sulopenem Versus Ertapenem for Complicated Intra-abdominal Infection (cIAI)PHASE3 COMPLETED 674Sep 18, 2018Oct 2, 2019Dec 1, 202042 United States, Bulgaria +5
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Study Endpoints
Primary Endpoints
Percentage of Participants With Clinical Success
Day 28 +/- 1 day

Clinical response is defined as resolution in signs and symptoms of the index infection and no new symptoms, without the need for additional antibiotics or interventions

Secondary Endpoints
Percentage of Participants With Clinical Success
Day 11-14 +/- 1 day
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
SulopenemEXPERIMENTALSulopenem 1000 mg IV once daily for at least 5 days, followed by Sulopenem-Etzadroxil/Probenecid 500 mg PO twice daily to complete 7-10 days of treatment
ErtapenemACTIVE_COMPARATORErtapenem 1000 mg IV once daily for at least 5 days, followed by ciprofloxacin 500 mg PO twice daily along with metronidazole 500 mg PO four times daily. If patient is found to have causative pathogens that are resistant to ciprofloxacin they will receive amoxicillin-clavulanate 875 mg PO twice daily instead
Interventions
NameTypeDescription
ErtapenemDRUGAntibiotic for complicated intra-abdominal infection
Sulopenem-Etzadroxil/ProbenecidDRUGAntibiotic for complicated intra-abdominal infection
CiprofloxacinDRUGAntibiotic for complicated intra-abdominal infection
MetronidazoleDRUGAntibiotic for complicated intra-abdominal infection
Amoxicillin-ClavulanateDRUGAntibiotic for complicated intra-abdominal infection
SulopenemDRUGAntibiotic for complicated intra-abdominal infection
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites42

Inclusion Criteria: 1. Patient or the patient's legally acceptable representative able to provide a signed written informed consent prior to any study-specific procedures. 2. Adult patients ≥18 years of age 3. EITHER: a. Intra-operative/post-operative enrollment with visual confirmation (presen...

Countries:United StatesBulgariaEstoniaGeorgiaHungaryLatviaPoland
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