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ISIS 301012

Phase 2

Hypercholesterolemia, Familial | Small molecule | Metabolic |Ionis Pharmaceuticals, Inc.|Last Updated: Aug 3, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLED
Total Trials1
Total Enrollment12
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00280995Dose-escalating Safety Study of ISIS 301012 in Homozygous Familial Hypercholesterolemia Subjects on Lipid Lowering TherapyPHASE2 COMPLETED 12Jan 1, 2006Aug 1, 2007Aug 3, 20166 United States, Netherlands
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Study Endpoints
Primary Endpoints
Percent reduction in LDL-cholesterol from baseline
Week 7 (Cohorts A-C), Week 15 (Cohort D)
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Cohort AEXPERIMENTALLoading doses followed by weekly maintenance doses
Cohort BEXPERIMENTALLoading doses followed by weekly maintenance doses
Cohort CEXPERIMENTALLoading doses followed by weekly maintenance doses
Cohort DEXPERIMENTALLoading doses followed by extended weekly maintenance doses
Interventions
NameTypeDescription
ISIS 301012DRUG100 mg subcutaneous injections on days 1, 4, 8, 11, 15, 22, 29, and 36
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites6

Inclusion Criteria: * Weight ≥ 40 kg for Cohorts A, B, \& C; Weight ≥ 50 kg for Cohort D * Diagnosis of Homozygous Familial Hypercholesterolemia. * Female must be non-pregnant and non-lactating. * On stable lipid lowering therapy for at least 4 weeks. * Lipid values that meet the pre-specified crit...

Countries:United StatesNetherlands
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