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Ruxolitinib IR

Phase 1

Healthy Participants | Small molecule | Other |Incyte Corporation|Last Updated: Feb 13, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials2
Total Enrollment192
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06555081A Study to Evaluate the Bioequivalence of Ruxolitinib Extended Release (XR) Tablets With Ruxolitinib Immediate Release (IR) Tablets Administered Orally in Healthy ParticipantsPHASE1 COMPLETED 168Sep 25, 2024Nov 7, 2024Feb 13, 20251 United States
NCT06310304A Study to Evaluate the Relative Bioavailability of Ruxolitinib Extended Release (XR) Tablets Compared With Ruxolitinib Immediate Release (IR) Tablets Administered Orally in Healthy Participants.PHASE1 COMPLETED 24Mar 26, 2024May 15, 2024Jun 5, 20241 United States
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Study Endpoints
Primary Endpoints
INCB018424 pharmacokinetic (PK) in Plasma
Up to Day 16

INCB018424 concentration in plasma.

Secondary Endpoints
Number of participants with Treatment Emergent Adverse Events (TEAEs)
Up to Day 33
Additional INCB018424 pharmacokinetic (PK) in Plasma
Up to Day 16
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Period 1: Dose Treatment AEXPERIMENTALRuxolitinib IR will be administered at protocol defined dose.
Period 1: Dose Treatment BEXPERIMENTALRuxolitinib XR will be administered at protocol defined dose.
Period 2: Dose Treatment AEXPERIMENTALRuxolitinib IR will be administered at protocol defined dose.
Period 2: Dose Treatment BEXPERIMENTALRuxolitinib XR will be administered at protocol defined dose.
Cohort 1: Dose Treatment AEXPERIMENTALRuxolitinib IR will be administered at protocol defined dose.
Cohort 1: Dose Treatment BEXPERIMENTALRuxolitinib XR will be administered at protocol defined dose.
Cohort 2: Dose Treatment AEXPERIMENTALRuxolitinib IR will be administered at protocol defined dose.
Cohort 2: Dose Treatment BEXPERIMENTALRuxolitinib XR will be administered at protocol defined dose.
Interventions
NameTypeDescription
Ruxolitinib IRDRUGTablet
Ruxolitinib XRDRUGTablet
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Ability to comprehend and willingness to sign a written ICF for the study. * Healthy adult participants aged 18 to 55 years, inclusive at screening. * Body mass index between 18.0 and 32.0 kg/m2, inclusive, at screening. Note: Only up to 25% of the participants may be enrolled...

Countries:United States
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