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ropinirole controlled release-RLS

Phase 2

Restless Legs Syndrome | Small molecule | Neurology |GSK plc|Last Updated: Sep 26, 2018

Success Probability

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment35

FDA Designations

No designations recorded

Clinical trial landscape

ropinirole controlled release-RLS · 1 trial · 1 indication

Phase 2 1
NCT00530790Clinical Evaluation of Ropinirole CR-RLS ( SK&F101468)Tablets in Restless Legs SyndromeRestless Legs Syndrome
COMPLETED35 Analytics
PHASE2COMPLETED
Clinical Evaluation of Ropinirole CR-RLS ( SK&F101468)Tablets in Restless Legs Syndrome
Restless Legs SyndromeUnlock trial analytics

Study Endpoints

Primary Endpoints

Drug Related Adverse Events-On-Therapy
Weeks 1 - 12 Treatment Period
Haematology Clinical Lab Values Change From Baseline
Baseline - Week 13 (Follow-up)

Standard units of measure vary. Therefore, Mean Change is represented in Standard Units: Hematocrit = SI unit of GSK; Hemoglobin = G/L; Platelet count, White Blood Cell count = GI/L; Red Blood Cell count = TI/L. n = number of subjects evaluated. EW = Early Withdrawal.

Blood Chemistry Clinical Lab Values Change From Baseline
Baseline - Week 13 (Follow-up)

Mean Change in Standard Units of Measure: Albumin, Total Protein=G/L; Alkaline Phosphatase, Alanine Amino Transferase, Aspartate Amino Transferase, Lactate Dehydrogenase, Creatine Phosphokinase, Gamma Glutamyl Transferase=IU/L; Total Bilirubin, Creatinine=UMOL/L; Blood Urea Nitrogen, Cholesterol, Chloride, Sodium, Potassium=MMOL/L; Prolactin=MCG/L

Urinalysis Clinical Lab Values
Baseline - Week 13 (Follow-up)

Dipstick test values: Neg Value, Trace, +1, +2, +3. No subjects tested higher than +3.

12-Lead Electrocardiogram (ECG) Findings Transitions From Baseline
Baseline, Week 4, 8, 12, 13 (Follow-up)

Baseline Finding/Time Period Finding. Abbreviations: N = normal; A = abnormal; CS = clinically significant; NCS = not clinically significant. Options include N/N, N/ANCS, N/ACS, ANCS/N, ANCS/ANCS, ANCS/ACS, ACS/N, ACS/ANCS, and ACS/ACS.

Vital Signs and Body Weight Change From Baseline
Baseline to Week 12/EW

Units of Measure Vary: Weight = kg; Semi-supine and Standing Systolic and Diastolic BP = mmHg; Semi-supine and Standing Pulse Rate = bpm; EW = early withdrawal; Semi-supine = lying down; Orthostatic = lying, sitting, and standing.

Secondary Endpoints

Change From Baseline to Week 12 in International Restless Leg Syndrome (IRLS) Rating Scale Total Score
Baseline and after Week 12
Clinical Global Impression Scale - Severity of Illness (CGI-S)
Baseline - Final assessment point
Clinical Global Impression Global Improvement (CGI-GI)
Baseline - Final assessment point
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ropinirole CR-RLSEXPERIMENTALSubjects will orally take ropinirole CR-RLS tablet(s) once daily 1-2 hours before the onset of RLS symptoms at about the same time of the day. The time of taking ropinirole must be after 16:00.Adjustment of the Ropinirole CR-RLS tablets should be completed after the Week 1 visit up to the Week 10 visit. The dose will be increased at intervals of at least one week until sufficient efficacy is obtained (use "much improved" as a guide) without safety problem. Dose escalation will start at the initial dose 0.5 mg/day to 1 mg/day; after 1 mg/day, the dose will be increased by 1 mg/day to the maximum 6 mg/day.

Interventions

NameTypeDescription
ropinirole controlled release (CR)-RLSDRUGWhite film-coated round-shaped tablet
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Eligibility Criteria

Age Range18 Years to 79 Years
SexALL
Healthy VolunteersNo
Study Sites11

Inclusion Criteria: * A subject will be considered eligible for inclusion in this study only if all of the following criteria apply: At Week -1 (at the start of Screening period) * Patients who are diagnosed with RLS according to the International RLS Study Group's (IRLSSG) Diagnostic Criteria. *...

Countries:Japan
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Frequently asked questions about ropinirole controlled release-RLS

What is ropinirole controlled release-RLS used for?

Ropinirole controlled release-RLS is an investigational small molecule being studied for Restless Legs Syndrome and Parkinson's Disease. It is a controlled-release formulation of ropinirole, a dopamine agonist. The drug is in clinical development for these neurological conditions, though it is not yet approved.

Who makes ropinirole controlled release-RLS?

Ropinirole controlled release-RLS is being developed by GSK plc, which trades under the ticker GSK. The company is conducting clinical trials to evaluate the drug's safety and efficacy in Restless Legs Syndrome and Parkinson's Disease.

What phase is ropinirole controlled release-RLS in?

Ropinirole controlled release-RLS is in Phase 2 clinical development for Restless Legs Syndrome. A Phase 3 trial was also completed for Parkinson's Disease. The drug remains investigational and has not been approved by regulatory authorities.

What clinical trials is ropinirole controlled release-RLS in?

Ropinirole controlled release-RLS has been evaluated in two completed trials. NCT00363727 was a Phase 3 study in Parkinson's Disease with 209 participants, and NCT00530790 was a Phase 2 study in Restless Legs Syndrome with 35 participants. Both trials are completed.

Is ropinirole controlled release-RLS the same as REQUIP CR?

Yes, ropinirole controlled release-RLS is also known as REQUIP CR, as referenced in the clinical trial NCT00363727. This controlled-release formulation of ropinirole is being studied for Restless Legs Syndrome and Parkinson's Disease.